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Targets Recommended: PKA PDE

5

抑制剂 & 化合物

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天然产物

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重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T1418 Bucladesine sodium

dbcAMP,Dibutyryl-cAMP sodium salt,布拉地新钠盐,Dibutyryl-cAMP,DC2797,Sodium dibutyryl cAMP,Bucladesine,Bucladesine sodium salt

PKA; PDE Metabolism; Tyrosine Kinase/Adaptors
Bucladesine sodium (DC2797) 是一种 cAMP 类似物,具有细胞渗透性。Bucladesine sodium 也是一种 cAMP 依赖性的蛋白激酶 (PKA) 激活剂,一种磷酸二酯 (PDE) 抑制剂。Bucladesine sodium 具有抗炎活性。
T25505 Homomoschatoline

Liridine,O-Methyl-moschatoline

Homomoschatoline is an antibacterial isolated from Artabotrys crassifolius.
T29602 Achatin I

Gfad peptide,Achatin II,Achatin-I,Achatin-II

Achatin I is a neuroexcitatory tetrapeptide from Achatina fulica Ferussac.
T14194 β-NETA

α-NETA

AChE Neuroscience
β-NETA(α-NETA) 是胆碱乙酰转移酶(ChA;IC50=76 μM) 和胆碱酯酶 (ChE;IC50=40 µM)的非竞争性抑制剂,对乙酰胆碱酯的作用微弱 (AChE;IC50=1 mM)。
T64672 Colivelin TFA

Colivelin (sequence SALLRSIPAPAGASRLLLLTGEIDLP) is composed of activity-dependent neurotrophic factor (ADNF) C-terminally fused to AGA-(C8R)HNG17, a potent HN derivative. It works as a neuroprotective peptide and activator of STAT3. Colivelin-induced neuroprotection has been confirmed to occur via two neuroprotective pathways: one mediated by Ca2+/calmodulin-dependent protein kinase IV, triggered by ADNF, and one mediated by signal transducer and activator of transcription 3, triggered by HN. Co...

化合物

Bucladesine sodium
Cat.No: T1418
Synonym: dbcAMP,Dibutyryl-cAMP sodium salt,布拉地新钠盐,Dibutyryl-cAMP,DC2797,Sodium dibutyryl cAMP,Bucladesine,Bucladesine sodium salt
Target: PKA, PDE
Homomoschatoline
Cat.No: T25505
Synonym: Liridine,O-Methyl-moschatoline
Target:
Achatin I
Cat.No: T29602
Synonym: Gfad peptide,Achatin II,Achatin-I,Achatin-II
Target:
β-NETA
Cat.No: T14194
Synonym: α-NETA
Target: AChE
Colivelin TFA
Cat.No: T64672
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN1653 Fustin

ERK; Beta Amyloid; AChR MAPK; Neuroscience
Fustin 是植物漆树 (Rhus verniciflua Stokes) 的植物性黄烷醇成分。 Fustin 对 6-羟基多巴胺诱导的神经元细胞死亡具有保护作用。
T3767 Polygalacic acid

Virgaureagenin G,毛果一枝黄花皂苷元G,远志酸

MMP; AChR; AChE Neuroscience; Proteases/Proteasome
Polygalacic acid (Virgaureagenin G) 是一种从远志 Polygala tenuifolia Willd 根中分离出来的三萜,可抑制 MMP 表达。它对认知障碍有显著的神经保护作用,PA 通过抑制乙酰胆碱酯酶活性,增加胆碱乙酰转移酶活性,提高海马和额皮质中的乙酰胆碱水平来提高胆碱能系统反应性。 它可以用于骨关节炎相关研究。
T13818 Phytohemagglutinin

PHA-M,植物血球凝集素,PHA,植物血凝素

Apoptosis Apoptosis
Phytohemagglutinin (PHA-M) 是一种普通豆菜豆的主要种子凝集素,聚集在子叶的薄壁细胞中。它是一种 T 细胞激活剂,能够刺激人单核白细胞,可诱导 ChAT mRNA 表达,增强 ACh 合成。

天然产物

Fustin
Cat.No: TN1653
Synonym:
Target: ERK, Beta Amyloid, AChR
Polygalacic acid
Cat.No: T3767
Synonym: Virgaureagenin G,毛果一枝黄花皂苷元G,远志酸
Target: MMP, AChR, AChE
Phytohemagglutinin
Cat.No: T13818
Synonym: PHA-M,植物血球凝集素,PHA,植物血凝素
Target: Apoptosis
Cat. No. Product Name Species Expression System
TMPH-01085 CHAT Protein, Human, Recombinant (His)

CHAT,Choline O-acetyltransferase,ChAT,CHOA...

Human E. coli
Catalyzes the reversible synthesis of acetylcholine (ACh) from acetyl CoA and choline at cholinergic synapses. CHAT Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 72.7 kDa and the accession number is P28329.

重组蛋白

CHAT Protein, Human, Recombinant (His)
Cat.No: TMPH-01085
Species: Human
Expression System: E. coli
TargetMol Loading
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