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Cat. No. | Product Name | Target | Signaling Pathways |
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T30159 |
ASL-7003
ASL 7003,ASL7003, |
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ASL-7003 is a dopamine analog with cardian stimulating properties. | |||
T3575 |
Acecainide hydrochloride
ASL 601,NAPA |
Others | Others |
Acecainide hydrochloride (NAPA) 是 PROCAINAMIDE 的主要代谢物。其抗心律失常作用可能导致肾衰竭时的心脏毒性。 | |||
T20458 |
Aspirin DL-lysine
DL-Lysine acetylsalicylic acid salt,Aspegic,ASL,Aspisol |
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Aspirin DL-lysine is a non-steroidal anti-inflammatory drug. It also may inhibit cancer growth. Aspirin DL-lysine is a water-soluble, injectable aspirin derivative. | |||
T81852 |
Maslimomab
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Maslimomab为针对T细胞受体的鼠源性单克隆抗体,亦作为免疫抑制剂。 | |||
T80906 |
TYVPANASL TFA
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TYVPANASL TFA,一种由HER2/neu的9个氨基酸组成,可结合MHC I并与CD8 T细胞表位相关的化合物。该化合物可用于制备J-LEAPS疫苗。 | |||
T80907 |
TYVPANASL
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TYVPANASL为由HER2/neu的9个氨基酸组成的MHC I结合CD8 T细胞表位,可用于制备J-LEAPS疫苗。 | |||
T37039 |
Betulinic Aldehyde oxime
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Betulinic aldehyde oxime is a pentacyclic triterpenoid and derivative of the cholesterol biosynthesis inhibitor betulin .1It is active againstE. aerogenes,E. coli,E. faecalis,P. aeruginosa,S. aureus, andC. albicans, as well asL. donovaniamastigotes, when used at a concentration of 50 μM.1,2Betulinic aldehyde oxime (50 μM) is cytotoxic to Huh7 hepatocellular carcinoma cells.2 | |||
T82972 |
Argininosuccinic acid disodium
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Reactive Oxygen Species | Immunology/Inflammation; Metabolism; NF-κB |
Argininosuccinic acid disodium 在尿素循环的第四步起关键作用,由ASL(精氨酸琥珀酸裂解酶)催化裂解生成精氨酸和富马酸。此外,该化合物能够降低GSH(还原型谷胱甘肽)浓度,并提升大脑皮层与纹状体中的活性氧产生。Argininosuccinic acid disodium 还可能导致脂质过氧化和蛋白质氧化,并在发育中的大鼠脑内触发氧化应激。 |
Cat. No. | Product Name | Target | Signaling Pathways |
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T1644 |
Dopamine hydrochloride
盐酸多巴胺,Dopamine HCl,ASL279 |
Ferroptosis; Dopamine Receptor; 5-HT Receptor; Endogenous Metabolite | Apoptosis; GPCR/G Protein; Metabolism; Neuroscience |
Dopamine hydrochloride (ASL279) 是在脑黑质、脑腹侧被盖区和下丘脑中产生的一种天然儿茶酚胺,由二羟基苯丙氨酸脱羧形成,是去甲肾上腺素和肾上腺素的前体。它通过 D2 多巴胺受体来诱导 VEGFR2 的内吞作用,有促进血管生成活性。 | |||
TN2130 |
Manghaslin
槲皮素-3-O-芸香糖-(1→2)-O-鼠李糖苷,Quercetin 3-O-rutinoside-(1->2)-O-rhamnoside |
AChE; Glucosidase | Metabolism; Neuroscience |
Manghaslin (Quercetin 3-O-rutinoside-(1->2)-O-rhamnoside) 是具有抗炎活性的黄酮苷,对 AChE 具有抑制活性,IC50=94.92 µM。 | |||
TN7129 |
Methyl maslinate
马斯里酸甲酯,Maslinic acid methyl ester,Crategolic acid methyl ester |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Methyl maslinate (Maslinic acid methyl ester) 是一种具有强心和抗心律失常特性的 β-肾上腺素受体拮抗剂。Methyl maslinate 可用于高血压研究。 | |||
T3772 |
Maslinic acid
2α-Hydroxyoleanoic Acid,山楂酸,2α-Hydroxyoleanolic acid,Crategolic acid |
NF-κB; HIV Protease; DNA/RNA Synthesis; Antibacterial | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; NF-κB; Proteases/Proteasome |
Maslinic acid (Crategolic acid) 是一种 DNA 聚合酶 B 抑制剂,抑制 NF-κB p65的 DNA 结合活性并消除 IκB-α磷酸化。 | |||
TN6163 |
3-O-cis-p-Coumaroylmaslinic acid
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3-beta-O-(trans-p-Coumaroyl)maslinic acid shows antimicrobial activity on Gram-positive bacteria and yeasts. | |||
TN6148 |
3-O-trans-p-Coumaroylmaslinic acid
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3-beta-O-(trans-p-Coumaroyl)maslinic acid is a DNA polymerase B" inhibitor. It shows antimicrobial activity on Gram-positive bacteria and yeasts. | |||
TN5558 |
Jaslanceoside B
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Jaslanceoside B 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5558,CAS号为 188300-82-5。 | |||
T37977 |
Succinyladenosine
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Succinyladenosine is a biochemical marker of adenylosuccinase (ASL) deficiency. It is formed through the dephosphorylation of intracellular adenylosuccinic acid (S-AMP) by cytosolic 5-nucleotidase [1]. |