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8

抑制剂 & 化合物

8

天然产物

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Cat. No. Product Name Target Signaling Pathways
T30159 ASL-7003

ASL 7003,ASL7003,

ASL-7003 is a dopamine analog with cardian stimulating properties.
T3575 Acecainide hydrochloride

ASL 601,NAPA

Others Others
Acecainide hydrochloride (NAPA) 是 PROCAINAMIDE 的主要代谢物。其抗心律失常作用可能导致肾衰竭时的心脏毒性。
T20458 Aspirin DL-lysine

DL-Lysine acetylsalicylic acid salt,Aspegic,ASL,Aspisol

Aspirin DL-lysine is a non-steroidal anti-inflammatory drug. It also may inhibit cancer growth. Aspirin DL-lysine is a water-soluble, injectable aspirin derivative.
T81852 Maslimomab

Maslimomab为针对T细胞受体的鼠源性单克隆抗体,亦作为免疫抑制剂。
T80906 TYVPANASL TFA

TYVPANASL TFA,一种由HER2/neu的9个氨基酸组成,可结合MHC I并与CD8 T细胞表位相关的化合物。该化合物可用于制备J-LEAPS疫苗。
T80907 TYVPANASL

TYVPANASL为由HER2/neu的9个氨基酸组成的MHC I结合CD8 T细胞表位,可用于制备J-LEAPS疫苗。
T37039 Betulinic Aldehyde oxime

Betulinic aldehyde oxime is a pentacyclic triterpenoid and derivative of the cholesterol biosynthesis inhibitor betulin .1It is active againstE. aerogenes,E. coli,E. faecalis,P. aeruginosa,S. aureus, andC. albicans, as well asL. donovaniamastigotes, when used at a concentration of 50 μM.1,2Betulinic aldehyde oxime (50 μM) is cytotoxic to Huh7 hepatocellular carcinoma cells.2
T82972 Argininosuccinic acid disodium

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
Argininosuccinic acid disodium 在尿素循环的第四步起关键作用,由ASL(精氨酸琥珀酸裂解酶)催化裂解生成精氨酸和富马酸。此外,该化合物能够降低GSH(还原型谷胱甘肽)浓度,并提升大脑皮层与纹状体中的活性氧产生。Argininosuccinic acid disodium 还可能导致脂质过氧化和蛋白质氧化,并在发育中的大鼠脑内触发氧化应激。

化合物

ASL-7003
Cat.No: T30159
Synonym: ASL 7003,ASL7003,
Target:
Acecainide hydrochloride
Cat.No: T3575
Synonym: ASL 601,NAPA
Target: Others
Aspirin DL-lysine
Cat.No: T20458
Synonym: DL-Lysine acetylsalicylic acid salt,Aspegic,ASL,Aspisol
Target:
Maslimomab
Cat.No: T81852
Synonym:
Target:
TYVPANASL TFA
Cat.No: T80906
Synonym:
Target:
TYVPANASL
Cat.No: T80907
Synonym:
Target:
Betulinic Aldehyde oxime
Cat.No: T37039
Synonym:
Target:
Argininosuccinic acid disodium
Cat.No: T82972
Synonym:
Target: Reactive Oxygen Species
Cat. No. Product Name Target Signaling Pathways
T1644 Dopamine hydrochloride

盐酸多巴胺,Dopamine HCl,ASL279

Ferroptosis; Dopamine Receptor; 5-HT Receptor; Endogenous Metabolite Apoptosis; GPCR/G Protein; Metabolism; Neuroscience
Dopamine hydrochloride (ASL279) 是在脑黑质、脑腹侧被盖区和下丘脑中产生的一种天然儿茶酚胺,由二羟基苯丙氨酸脱羧形成,是去甲肾上腺素和肾上腺素的前体。它通过 D2 多巴胺受体来诱导 VEGFR2 的内吞作用,有促进血管生成活性。
TN2130 Manghaslin

槲皮素-3-O-芸香糖-(1→2)-O-鼠李糖苷,Quercetin 3-O-rutinoside-(1->2)-O-rhamnoside

AChE; Glucosidase Metabolism; Neuroscience
Manghaslin (Quercetin 3-O-rutinoside-(1->2)-O-rhamnoside) 是具有抗炎活性的黄酮苷,对 AChE 具有抑制活性,IC50=94.92 µM。
TN7129 Methyl maslinate

马斯里酸甲酯,Maslinic acid methyl ester,Crategolic acid methyl ester

Adrenergic Receptor GPCR/G Protein; Neuroscience
Methyl maslinate (Maslinic acid methyl ester) 是一种具有强心和抗心律失常特性的 β-肾上腺素受体拮抗剂。Methyl maslinate 可用于高血压研究。
T3772 Maslinic acid

2α-Hydroxyoleanoic Acid,山楂酸,2α-Hydroxyoleanolic acid,Crategolic acid

NF-κB; HIV Protease; DNA/RNA Synthesis; Antibacterial Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; NF-κB; Proteases/Proteasome
Maslinic acid (Crategolic acid) 是一种 DNA 聚合酶 B 抑制剂,抑制 NF-κB p65的 DNA 结合活性并消除 IκB-α磷酸化。
TN6163 3-O-cis-p-Coumaroylmaslinic acid

3-beta-O-(trans-p-Coumaroyl)maslinic acid shows antimicrobial activity on Gram-positive bacteria and yeasts.
TN6148 3-O-trans-p-Coumaroylmaslinic acid

3-beta-O-(trans-p-Coumaroyl)maslinic acid is a DNA polymerase B" inhibitor. It shows antimicrobial activity on Gram-positive bacteria and yeasts.
TN5558 Jaslanceoside B

Jaslanceoside B 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5558,CAS号为 188300-82-5。
T37977 Succinyladenosine

Succinyladenosine is a biochemical marker of adenylosuccinase (ASL) deficiency. It is formed through the dephosphorylation of intracellular adenylosuccinic acid (S-AMP) by cytosolic 5-nucleotidase [1].

天然产物

Dopamine hydrochloride
Cat.No: T1644
Synonym: 盐酸多巴胺,Dopamine HCl,ASL279
Target: Ferroptosis, Dopamine Receptor, 5-HT Receptor, Endogenous Metabolite
Manghaslin
Cat.No: TN2130
Synonym: 槲皮素-3-O-芸香糖-(1→2)-O-鼠李糖苷,Quercetin 3-O-rutinoside-(1->2)-O-rhamnoside
Target: AChE, Glucosidase
Methyl maslinate
Cat.No: TN7129
Synonym: 马斯里酸甲酯,Maslinic acid methyl ester,Crategolic acid methyl ester
Target: Adrenergic Receptor
Maslinic acid
Cat.No: T3772
Synonym: 2α-Hydroxyoleanoic Acid,山楂酸,2α-Hydroxyoleanolic acid,Crategolic acid
Target: NF-κB, HIV Protease, DNA/RNA Synthesis, Antibacterial
3-O-cis-p-Coumaroylmaslinic acid
Cat.No: TN6163
Synonym:
Target:
3-O-trans-p-Coumaroylmaslinic acid
Cat.No: TN6148
Synonym:
Target:
Jaslanceoside B
Cat.No: TN5558
Synonym:
Target:
Succinyladenosine
Cat.No: T37977
Synonym:
Target:
TargetMol Loading
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