Powder: -20°C for 3 years | In solvent: -80°C for 1 year
BW-A 78U 抑制 PDE4,其 IC50值为 3 μM。
规格 | 价格/CNY | 货期 | 数量 | |
---|---|---|---|---|
1 mg | ¥ 498 | 现货 | ||
2 mg | ¥ 727 | 现货 | ||
5 mg | ¥ 1,190 | 现货 | ||
10 mg | ¥ 1,780 | 现货 | ||
25 mg | ¥ 2,970 | 现货 | ||
50 mg | ¥ 4,380 | 现货 | ||
100 mg | ¥ 6,190 | 现货 | ||
1 mL * 10 mM (in DMSO) | ¥ 638 | 现货 |
产品描述 | BW-A 78U is a PDE4 inhibitor (IC50: 3 μM). It is not inhibition on the lipopolysaccharide (LPS)-induced TNF-α release. |
靶点活性 | PDE4:3 μM |
细胞实验 | Mononuclear cells were incubated for 30 min with BW-A 78U (0.01-10 μM). The cells were then stimulated with lipopolysaccharide (10 μg/mL) overnight at 37°C in an atmosphere of 5% CO2 at 100% humidity. Cell-free supernatants were collected, centrifuged (2000 g), and stored frozen at -20°C before TNF-α determination. TNF-α concentrations in cell culture supernatants were determined by specific ELISA using a commercial kit. The sensitivity of the assay was 1 pg/mL. The absorbance at 450 nm was assessed with an ELISA reader. |
别名 | BW-A78U |
分子量 | 257.27 |
分子式 | C13H12FN5 |
CAS No. | 101155-02-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 45 mg/mL (174.91 mM)
可选溶剂 | 浓度 体积 质量 | 1 mg | 5 mg | 10 mg | 25 mg |
DMSO | 1 mM | 3.887 mL | 19.4348 mL | 38.8697 mL | 97.1742 mL |
5 mM | 0.7774 mL | 3.887 mL | 7.7739 mL | 19.4348 mL | |
10 mM | 0.3887 mL | 1.9435 mL | 3.887 mL | 9.7174 mL | |
20 mM | 0.1943 mL | 0.9717 mL | 1.9435 mL | 4.8587 mL | |
50 mM | 0.0777 mL | 0.3887 mL | 0.7774 mL | 1.9435 mL | |
100 mM | 0.0389 mL | 0.1943 mL | 0.3887 mL | 0.9717 mL |
对于不同动物的给药剂量换算,您也可以参考 更多...
请在以下方框中输入您的动物实验信息后点击计算,可以得到母液配置方法和体内配方的制备方法: 比如您的给药剂量是10 mg/kg,每只动物体重20 g,给药体积100 μL,一共给药动物10 只,您使用的配方为5% DMSO+30% PEG300+5% Tween 80+60% ddH2O。那么您的工作液浓度为2 mg/mL。
母液配置方法:2 mg 药物溶于 50 μL DMSO (母液浓度为 40 mg/mL), 如您需要配置的浓度超过该产品的溶解度,请先与我们联系。
体内配方的制备方法:取 50 μL DMSO 主液,加入 300 μL PEG300, 混匀澄清,再加 50 μL Tween 80,混匀澄清,再加 600 μL ddH2O, 混匀澄清。
您可能有的问题的答案可以在抑制剂处理说明中找到,包括如何准备库存溶液,如何存储产品,以及基于细胞的分析和动物实验需要特别注意的问题。
BW-A 78U 101155-02-6 Metabolism PDE inhibit Inhibitor BW A 78U BW-A78U Phosphodiesterase (PDE) BWA 78U inhibitor