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Cat. No. Product Name Target Signaling Pathways
TN2315 Xanthopurpurin

茜草红素,1,3-二羥蒽醌,异茜草素

Platelet aggregation; Antifection Microbiology/Virology; Others
Xanthopurpurin 是分离自Rubia akane 根茎的蒽醌苷。Xanthopurpurin 主要对胶原诱导的血小板聚集有较强的抑制作用。
T4241 Rubiadin

1,3-Dihydroxy-2-Methylanthracene-9,10-Dione,茜根定,茜草素

Free radical scavengers; PARP; Caspase Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; oxidation-reduction; Proteases/Proteasome
Rubiadin (1,3-Dihydroxy-2-Methylanthracene-9,10-Dione) 是一种二羟基蒽醌,提取自茜草,具有抗氧化剂作用。
T3673 Mollugin

大叶茜草素,Rubimaillin

HER; JAK Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors
Mollugin (Rubimaillin) 是Rubia cordifolia L.中主要的生物活性成分。它能通过 p38-Smad 信号通路增强 BMP-2 的成骨作用。它通过抑制 TNF-α 诱导的 NF-κB 激活起抗癌疗效。
T5648 Purpurin

吡啉,1,2,4-Trihydroxyanthraquinone,Hydroxylizaric acid,Verantin

MAO; Antibacterial; Antibiotic; Antifungal Metabolism; Microbiology/Virology; Neuroscience
Purpurin (Verantin) 是来自Rubia tinctorumL. 的天然蒽醌,具有抗抑郁样作用。
TN1316 6-Hydroxyrubiadin

6-羟基茜草素,1,3,6-三羟基-2-甲基蒽醌

Others Others
6-Hydroxyrubiadin has antioxidant activity, EC(50) is 14.7ug/ml.
TN2417 Furomollugin

5-羟基萘并[1,2-B]呋喃-4-甲酸甲酯,呋喃大叶茜草素

Antifection Microbiology/Virology
Furomollugin has antiviral activity, it can strongly suppress the secretion of hepatitis B surface antigen (HBsAg), with IC50 = 2.0 micrograms/mL, in human hepatoma Hep3B cells.
TN2163 Rubioncolin C

NF-κB NF-κB
Rubioncolin C shows good cytotoxicity with IC50 value of 1.53 μM and NF-κB inhibitory activity with IC50 value of 2.97 μM.
TN1886 Lucidin primeveroside

Lucidin 3-O-primeveroside,亮黄素3-桑色素酊

Topoisomerase DNA Damage/DNA Repair
Lucidin primeveroside (Lucidin 3-O-primeveroside) 是从茜草的根粉中分离得到的天然产物,可用作着色剂和食用色素。 Lucidin Primeveroside 可以在小鼠体内代谢转化为基因毒性化合物 Lucidin。
T6S1294 Nicotiflorin

Nictoflorin,Kaempferol-3-O-Rutinoside,山奈酚-3-O-芸香糖苷,Nicotifloroside

Others Others
Nicotiflorin (Kaempferol-3-O-Rutinoside) 是一种黄酮苷,从传统中药Flos Carthami 中提取得到。它有抗糖化活性和神经保护作用。

天然产物

Xanthopurpurin
Cat.No: TN2315
Synonym: 茜草红素,1,3-二羥蒽醌,异茜草素
Target: Platelet aggregation, Antifection
Rubiadin
Cat.No: T4241
Synonym: 1,3-Dihydroxy-2-Methylanthracene-9,10-Dione,茜根定,茜草素
Target: Free radical scavengers, PARP, Caspase
Mollugin
Cat.No: T3673
Synonym: 大叶茜草素,Rubimaillin
Target: HER, JAK
Purpurin
Cat.No: T5648
Synonym: 吡啉,1,2,4-Trihydroxyanthraquinone,Hydroxylizaric acid,Verantin
Target: MAO, Antibacterial, Antibiotic, Antifungal
6-Hydroxyrubiadin
Cat.No: TN1316
Synonym: 6-羟基茜草素,1,3,6-三羟基-2-甲基蒽醌
Target: Others
Furomollugin
Cat.No: TN2417
Synonym: 5-羟基萘并[1,2-B]呋喃-4-甲酸甲酯,呋喃大叶茜草素
Target: Antifection
Rubioncolin C
Cat.No: TN2163
Synonym:
Target: NF-κB
Lucidin primeveroside
Cat.No: TN1886
Synonym: Lucidin 3-O-primeveroside,亮黄素3-桑色素酊
Target: Topoisomerase
Nicotiflorin
Cat.No: T6S1294
Synonym: Nictoflorin,Kaempferol-3-O-Rutinoside,山奈酚-3-O-芸香糖苷,Nicotifloroside
Target: Others
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