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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6991 |
Nitroprusside disodium dihydrate
硝普钠二水合物,硝普钠,Sodium Nitroferricyanide(III) Dihydrate,Sodium Nitroprusside Dihydrate |
Guanylate cyclase; Autophagy | Autophagy; GPCR/G Protein |
Nitroprusside disodium dihydrate (Sodium Nitroprusside Dihydrate) 是一种血管扩张剂,通过在血液中自发释放 NO 发挥作用。它可在谷胱甘肽耗竭的成骨细胞中诱导自噬,用于急性高血压和心力衰竭的研究。 | |||
T2226 |
Pergolide mesylate
甲磺酸培高利特,Pergolide mesylate salt,LY127809,Pergolide methanesulfonate |
Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Pergolide mesylate salt(LY127809) 是一种有效的,具有口服活性的多巴胺 D1和 D2受体激动剂,是一种 Ergoline 衍生物,可用于帕金森氏病和高泌乳素血症的研究。 | |||
T24799 |
SKA-111
SKA 111,SKA111 |
Potassium Channel | Membrane transporter/Ion channel |
SKA-111 是一种选择性钙离子激活的钾离子通道 (potassium phannel ) KCa3.1 激活剂,可引起猪内皮细胞膜超极化。SKA-111结合在CaM N-瓣和S4-S5接头之间的界面中,能够改善 Bradykinin 诱导的离体大鼠心脏的冠状动脉扩张,可用于研究心血管疾病。 | |||
T73645 | ARL67156 triethylamine | ||
ARL67156 (FPL 67156) triethylamine 是一种ecto-ATPase 抑制剂。ARL67156 triethylamine 是竞争性 NTPDase1 (CD39),NTPDase3 和 NPP1 抑制剂,Ki 分别为 11,18 和 12 μM。ARL67156 triethylamine 可用于钙化性主动脉瓣疾病、哮喘等疾病的研究。 | |||
T73644 | ARL67156 trisodium hydrate | ||
ARL67156 (FPL 67156) trisodium hydrate 是一种ecto-ATPase 抑制剂。ARL67156 trisodium hydrate 是竞争性 NTPDase1 (CD39),NTPDase3 和 NPP1 抑制剂,Ki 分别为 11,18 和 12 μM。ARL67156 trisodium hydrate 可用于钙化性主动脉瓣疾病、哮喘等疾病的研究。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN2553 |
1-Methyl-2-undecyl-4(1H)-quinolone
1-Methyl-2-undecylquinolin-4(1H)-one |
MAO | Metabolism; Neuroscience |
1-Methyl-2-undecyl-4(1H)-quinolone, and dihydroevocarpine should also be served as the chemical markers together with evodiamine for the quality control of Evodia rutaecarpa (Juss.) Benth. 1-Methyl-2-undecyl-4(1H)-quinolone shows a selective inhibition of type B MAO (MAO-B) activity with the IC(50) value of 15.3 microM using a substrate kynuramine, but does not inhibit type A MAO (MAO-A) activity.It can mitigate high phosphate-induced human aortic valve interstitial cells (HAVICs) calcification ... |