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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T1296 4-Aminosalicylic acid

Aminosalicylic acid,4-aminosalicylate,para-aminosalicylic acid,对氨水杨酸,Aminopar

NF-κB; Lipoxygenase; COX; Glutathione Peroxidase; Antibacterial; Antibiotic Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience; NF-κB
4-Aminosalicylic acid (para-aminosalicylic acid) 是一种具有口服活性的抗生素,可研究肺结核病。
T0315 Acedoben

Others Others
Acedoben 是对氨基苯甲酸 (PABA) 的乙酰基衍生物。
T0836 Sulfadoxine

周效磺胺,磺胺多辛,Sulphadoxine

DHFR; HIV Protease; Antibiotic; Parasite; Autophagy Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology; Proteases/Proteasome
Sulfadoxine (Sulphadoxine) 是磺胺类化合物,常与pyrimethamine 结合起到抗疟疾作用。它抑制HIV 在外周血单核细胞中的复制。
T0930 Sulfadiazine

Sulphadiazine,磺胺嘧啶

Antibacterial; Antibiotic; Parasite; Autophagy Autophagy; Microbiology/Virology
Sulfadiazine (Sulphadiazine) 是一种磺胺类抗生素具有抗疟活性,可研究弓形虫病。
T0913 Sulfamerazine

磺胺甲基嘧啶,RP2632

Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology
Sulfamerazine (RP2632) 是磺胺类抗菌素。它是磺胺嘧啶的单甲基衍生物,是 2-磺胺基-4-甲基嘧啶。它是一种磺胺类药物,通过与对氨基苯甲酸 (PABA) 竞争结合二氢叶酸合成,抑制细菌合成二氢叶酸。
T0020 Sodium 4-aminosalicylate dihydrate

对氨基水杨酸钠二水合物,Sodium 4-Aminosalicylate,4-Amino-salicylic acid sodium salt

Free radical scavengers; NF-κB; Antibacterial; Antibiotic Microbiology/Virology; NF-κB; oxidation-reduction
Sodium 4-aminosalicylate dihydrate (4-Amino-salicylic acid sodium salt) 是一种抗耐药性结核化合物。
T13028 Sulfamerazine D4

Others Others
Sulfamerazine D4, a deuterium-labeled version of Sulfamerazine, acts as a sulfonamide antibacterial. It inhibits the bacterial synthesis of dihydrofolic acid by competing with para-aminobenzoic acid (PABA) for the binding site on dihydropteroate synthase.

化合物

4-Aminosalicylic acid
Cat.No: T1296
Synonym: Aminosalicylic acid,4-aminosalicylate,para-aminosalicylic acid,对氨水杨酸,Aminopar
Target: NF-κB, Lipoxygenase, COX, Glutathione Peroxidase, Antibacterial, Antibiotic
Acedoben
Cat.No: T0315
Synonym:
Target: Others
Sulfadoxine
Cat.No: T0836
Synonym: 周效磺胺,磺胺多辛,Sulphadoxine
Target: DHFR, HIV Protease, Antibiotic, Parasite, Autophagy
Sulfadiazine
Cat.No: T0930
Synonym: Sulphadiazine,磺胺嘧啶
Target: Antibacterial, Antibiotic, Parasite, Autophagy
Sulfamerazine
Cat.No: T0913
Synonym: 磺胺甲基嘧啶,RP2632
Target: Antibacterial, Antibiotic, Autophagy
Sodium 4-aminosalicylate dihydrate
Cat.No: T0020
Synonym: 对氨基水杨酸钠二水合物,Sodium 4-Aminosalicylate,4-Amino-salicylic acid sodium salt
Target: Free radical scavengers, NF-κB, Antibacterial, Antibiotic
Sulfamerazine D4
Cat.No: T13028
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T1311 4-aminobenzoic acid

PABA,Vitamin H1,Vitamin Bx,para-Aminobenzoic acid,对氨基苯甲酸

Endogenous Metabolite Metabolism
4-aminobenzoic acid (para-Aminobenzoic acid) 是一种具有紫外线吸收和抗纤维化特性的有机酸。当暴露在光线下时,4-aminobenzoic acid 吸收紫外线并通过光化学反应释放多余的能量,这可能会对DNA造成损害。4-aminobenzoic acid 还可以增加组织水平的摄氧量,并可能增强单胺氧化酶(MAO)活性以促进血清素的降解,过量可能导致纤维化变化。

天然产物

4-aminobenzoic acid
Cat.No: T1311
Synonym: PABA,Vitamin H1,Vitamin Bx,para-Aminobenzoic acid,对氨基苯甲酸
Target: Endogenous Metabolite
TargetMol Loading
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