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9

抑制剂 & 化合物

1

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Cat. No. Product Name Target Signaling Pathways
T23686 AHR-activator-1023

Branching Morphogenesis Modulator 1023,Cpd 1023,Compound 1023,BMM 1023

AHR-activator-1023 is the aryl hydrocarbon receptor activator. It is also a specific FGF2-induced branching morphogenesis modulator.
T6351 MGCD-265 analog

MGCD-265,Glesatinib

Apoptosis; VEGFR; c-Met/HGFR Angiogenesis; Apoptosis; Tyrosine Kinase/Adaptors
MGCD-265 analog (Glesatinib) 是一种口服生物可利用的多靶点酪氨酸激酶抑制剂,具有抗肿瘤活性,对 c-Met 和 VEGFR2 的 IC50 分别为 29 nM 和 10 nM。
T8389 Trifluoperazine

三氟拉嗪,trifluoroperazine

CaMK; Dopamine Receptor; Influenza Virus; Adrenergic Receptor; P-gp; Autophagy Autophagy; GPCR/G Protein; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
Trifluoperazine (trifluoroperazine) 是一种多巴胺 D2 受体抑制剂,可治疗精神分裂症。它是NUPR1抑制剂,具有抗癌活性。它是α1-adrenergic 受体拮抗剂,是流感病毒形态发生的可逆抑制剂。
T1222 Trifluoperazine dihydrochloride

Trifluoperazine 2HCl,盐酸三氟拉嗪,SKF5019,Urinox

CaMK; Dopamine Receptor; Influenza Virus; Adrenergic Receptor; P-gp; Autophagy Autophagy; GPCR/G Protein; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
Trifluoperazine dihydrochloride (SKF5019) 是一种抗精神病药物,靶向中枢多巴胺受体。它是流感病毒形态发生的可逆抑制剂,是NUPR1抑制剂,具有抗癌活性。它是钙调蛋白抑制剂,还可抑制 P-糖蛋白,可研究精神分裂症。
T71508 TCSA

TCSA is an inhibitor of fungal morphogenesis, biofilm formation, and host cell invasion.
T27089 CRT0066854

CRT0066854 HCl,CRT-0066854 HCl,CRT 0066854,CRT-0066854

CRT-0066854 is a PKCι and PKCζ inhibitor. CRT0066854 was able to restore polarized morphogenesis in the dysplastic H-Ras spheroids.
T27590 IHVR-11029

IHVR 11029

IHVR-11029 is a potent inhibitor of ER α-glucosidase. IHVR-11029 is active against multiple hemorrhagic fever viruses and efficiently disrupts the morphogenesis of a broad spectrum of enveloped viruses.
T78030 GRGESP

GRGESP为胶原凝胶收缩抑制剂,能够抑制人成纤维细胞在胶原凝胶中的扩散,显著减少凝胶收缩,适用于结缔组织形态发生研究。
T38336 W140 (trifluoroacetate salt)

W140 (trifluoroacetate salt)

Sphingosine-1-phosphate (S1P) is a bioactive lipid that exhibits a broad spectrum of biological activities including cell proliferation, survival, migration, cytoskeletal organization, and morphogenesis. It exerts its activity by binding to five distinct G protein-coupled receptors, S1P1/EDG-1, S1P2/EDG-5, S1P3/EDG-3, S1P4/EDG-6, and S1P5/EDG-8. W140 is an inactive enantiomer of W146, a selective S1P1 antagonist (Ki = 77 nM), that binds to the S1P1 receptor with a Ki of 4.6 μM (2a = W146; 2b = W...

化合物

AHR-activator-1023
Cat.No: T23686
Synonym: Branching Morphogenesis Modulator 1023,Cpd 1023,Compound 1023,BMM 1023
Target:
MGCD-265 analog
Cat.No: T6351
Synonym: MGCD-265,Glesatinib
Target: Apoptosis, VEGFR, c-Met/HGFR
Trifluoperazine
Cat.No: T8389
Synonym: 三氟拉嗪,trifluoroperazine
Target: CaMK, Dopamine Receptor, Influenza Virus, Adrenergic Receptor, P-gp, Autophagy
Trifluoperazine dihydrochloride
Cat.No: T1222
Synonym: Trifluoperazine 2HCl,盐酸三氟拉嗪,SKF5019,Urinox
Target: CaMK, Dopamine Receptor, Influenza Virus, Adrenergic Receptor, P-gp, Autophagy
TCSA
Cat.No: T71508
Synonym:
Target:
CRT0066854
Cat.No: T27089
Synonym: CRT0066854 HCl,CRT-0066854 HCl,CRT 0066854,CRT-0066854
Target:
IHVR-11029
Cat.No: T27590
Synonym: IHVR 11029
Target:
GRGESP
Cat.No: T78030
Synonym:
Target:
W140 (trifluoroacetate salt)
Cat.No: T38336
Synonym: W140 (trifluoroacetate salt)
Target:
Cat. No. Product Name Target Signaling Pathways
T72867 Fusarisetin A

Fusarisetin A 是一种五环真菌代谢物,是一种腺泡形态发生抑制剂。

天然产物

Fusarisetin A
Cat.No: T72867
Synonym:
Target:
TargetMol Loading
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