Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0154 |
Nebivolol hydrochloride
R 065824 hydrochloride,盐酸奈必洛尔,Nebivolol HCl,R-65824 |
Apoptosis; Adrenergic Receptor | Apoptosis; GPCR/G Protein; Neuroscience |
Nebivolol hydrochloride (R 065824 hydrochloride) 是一种β1-肾上腺素受体选择性抑制剂,IC50为0.8 nM。 | |||
T20843 |
Aplodan
Nergize,Creatinolfosfate,磷酸肌肉醇,creatinol-O-phosphate,Creatinolfosfate, Creatinol Phosphate |
Others | Others |
Aplodan (creatinol-O-phosphate) 表现出抗缺血和抗心律失常的能力以及对细胞膜的保护作用。 Aplodan 可用于缺血性心脏病或伴有持续性室性早搏的缺血性心脏病的研究。 | |||
T29687 |
Afacifenacin
Afacifenacin fumarate,SMP-986,NS 986,NS-986,SMP 986,NS986,SMP986 |
AChR | Neuroscience |
Afacifenacin (SMP-986) fumarate 是一种 M3 毒蕈碱受体选择性拮抗剂,可用于研究缺血性心脏病,尿失禁和膀胱炎和其他疾病。 | |||
T0080 |
Trapidil
唑嘧胺,乐可安,Rocornal,Trapymine,Avantrin,Trapymin,AR-12008 |
PDGFR; PDE | Angiogenesis; Metabolism; Tyrosine Kinase/Adaptors |
Trapidil (Avantrin) 是一种抗血小板药物,是一种血管扩张剂,有特异性血小板衍生生长因子。 | |||
T0988 |
Trimetazidine dihydrochloride
盐酸曲美他嗪,Yoshimilon,Kyurinett,Vastarel F |
Autophagy; Fatty Acid Synthase | Autophagy; Metabolism |
Trimetazidine dihydrochloride (Vastarel F) 是细胞保护性抗缺血剂,也用作缺血性心脏病或心绞痛的血管扩张剂,具有抗氧化,抗炎,抗伤害和胃保护作用。它可通过抑制脂肪酸代谢提高心肌葡萄糖利用率。 | |||
T26279 |
Tiracizine HCl
AWD-19-166,AWD19166,Bonnecor,AWD 19 166,Tiracizine Hydrochloride |
||
Tiracizine HCl 是一种新的I 类抗心律失常药物,对缺血性心脏病患者进行了研究,结果表明该药物可降低心肌收缩功能。 | |||
T33673 |
Niludipine
Niludipina,BAY-a 7168,Bay a 7168,Niludipinum |
||
Nirudipine is a double (2-propoxyethyl) analogist of nifedipine and a calcium channel blocker, which is also a safe anti-angina Ca2+ antagonist with a broad range of efficacy for all types of angina. At the same time, Niludipine is a highly effective drug |