70
5
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0116 |
Balofloxacin
|
DNA gyrase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Balofloxacin 是一种具有口服活性的氟喹诺酮类抗生素,可通过干扰 DNA 促旋酶来抑制细菌 DNA 的合成,对革兰氏阴性,革兰氏阳性和厌氧菌具有广谱抗菌活性。它可研究呼吸道,肠道和泌尿道感染。 | |||
T3117 |
Marbofloxacin
马波沙星,Marbofloxacine,Zeniquin,Marbocyl |
Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Marbofloxacin (Zeniquin) 是一种具有口服活性的氟喹诺酮类广谱抗菌剂。它可研究革兰氏阳性和革兰氏阴性细菌以及支原体引起的感染。 | |||
T6349 |
Sitafloxacin Hydrate
西他沙星水合物,DU-6859a,DU6859a hydrate |
Antibacterial; Antibiotic | Microbiology/Virology |
Sitafloxacin Hydrate (DU-6859a) 是一种口服有效的氟喹诺酮类抗生素,在体外可对抗广泛的革兰氏阳性和阴性细菌有活性。Sitafloxacin 可研究呼吸道感染和尿路感染。 | |||
T9066 |
Merafloxacin
CI 934 |
SARS-CoV | Microbiology/Virology |
Merafloxacin (CI 934) 是一种氟喹诺酮类抗菌药物,也被确定为 SARS-CoV-2 的 1 PRF 抑制剂。它对革兰氏阳性菌和革兰氏阴性菌具有体外活性。 | |||
T7865 |
Danofloxacin
达氟沙星,达诺沙星,Danofloxacino,Danofloxacin free base,Danofloxacine |
Others; DNA/RNA Synthesis; Antibacterial; Antibiotic | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others |
Danofloxacin (Danofloxacin free base) free base 是一种具有口服活性第三代氟喹诺酮抗菌剂,对大多数革兰氏阴性和革兰氏阳性细菌,支原体和衣原体物种具有广谱的活性,并通过抑制细菌的 DNA 回转酶发挥抗菌作用。它可用于牛,猪和鸡呼吸道疾病的研究。 | |||
T6406 |
Besifloxacin Hydrochloride
BOL-303224-A,Besivance hydrochloride,Besifloxacin HCl,盐酸贝西沙星 |
Antibacterial; Antibiotic | Microbiology/Virology |
Besifloxacin Hydrochloride (BOL-303224-A) 是一种氟喹诺酮类抗生素。 | |||
T1620 |
Pazufloxacin Mesylate
Pazucross,Pazufloxacin mesilate,甲磺酸帕珠沙星,T-3762,帕珠沙星甲磺酸盐,Pazufloxacin methanesulfonate |
Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Pazufloxacin Mesylate (T-3762) 是一种喹诺酮类抗生素。 | |||
T1444 |
Lomefloxacin
洛美沙星,SC47111A |
Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Lomefloxacin (SC47111A) 是一种广谱喹诺酮类抗生素,具有抗菌活性。它可研究支气管炎、尿路感染、结膜炎、外耳炎和中耳炎。 | |||
T8173 |
Delafloxacin meglumine
ABT492 meglumine,德拉沙星葡甲胺,WQ-3034 meglumine,RX-3341 meglumine |
Antibacterial; Antibiotic | Microbiology/Virology |
Delafloxacin meglumine (RX-3341 meglumine) 是一种广谱氟喹诺酮类抗生素。Delafloxacin 对耐药性的金黄色葡萄球菌,肺炎克雷伯菌和肺炎链球菌有活性。 | |||
T1294 |
Fleroxacin
AM-833,氟罗沙星,RO 23-6240 |
DNA gyrase; Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Fleroxacin (RO 23-6240) 是一种广谱氟喹诺酮类抗菌素。 | |||
TQ0221 |
Rufloxacin hydrochloride
MF-934 hydrochloride,盐酸芦氟沙星 |
Antibacterial | Microbiology/Virology |
Rufloxacin hydrochloride (MF-934 hydrochloride) 是一种氟喹诺酮类抗菌剂,可抑制拓扑异构酶。 Rufloxacin hydrochloride 抑制人单核细胞中的 B 细胞分化。 | |||
T0292 |
Orbifloxacin
CP-104354,奥比沙星 |
Antibacterial; Antibiotic | Microbiology/Virology |
Orbifloxacin (CP-104354) 是一种可用于犬类的氟喹诺酮类合成广谱抗生素。 | |||
T1095 |
Sparfloxacin
AT-4140,PD 131501,Zagam,司帕沙星,CI-978 |
DNA gyrase; Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Sparfloxacin (CI-978) 是一种氟喹诺酮类抗菌素。 | |||
T1640 |
Ciprofloxacin
Ciproxan,环丙沙星,Ciprobay,Bay o 9867,Bay-09867 |
Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Ciprofloxacin (Bay-09867) 是一种有高抗菌活性的氟喹诺酮类抗生素。 | |||
T1492 |
Gemifloxacin mesylate
LB-20304a,甲磺酸吉米沙星,SB-265805S,Gemifloxacin mesylate |
DNA gyrase; Topoisomerase; Antibacterial | DNA Damage/DNA Repair; Microbiology/Virology |
Gemifloxacin mesylate (Gemifloxacin mesylate) 是一种喹诺酮类口服广谱抗菌剂,可研究轻中度肺炎和慢性支气管炎的急性细菌性发作。 | |||
T1293 |
Gatifloxacin
BMS 206584-01,PD 135432,CG5501,BMS-206584,AM-1155,加替沙星 |
Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Gatifloxacin (CG5501) 是一种具有广谱抗菌活性的氟喹诺酮类抗生素。它可抑制大肠杆菌 DNA 解旋酶 (IC50=0.109 μg/ml) 和细菌 II 型拓扑异构酶(IC50=13.8 μg/ml)。在动物模型中,它有抗细菌性结膜炎作用。 | |||
T0425 |
Pefloxacin Mesylate
Pefloxacinium mesylate,甲磺酸培氟沙星 |
Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Pefloxacin Mesylate (Pefloxacinium mesylate) 是一种抗菌化合物,可抑制DNA 旋转酶阻断DNA 复制。 | |||
T13231L |
Trovafloxacin mesylate
|
Others; DNA/RNA Synthesis; Topoisomerase; Antibacterial | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others |
Trovafloxacin是一种广谱氟喹诺酮类抗生素,可阻断 DNA 促旋酶 (DNA gyrase) 和拓扑异构酶 IV (topoisomerase IV) 的活性,也是一种有效的特异性 pannexin 1 通道抑制剂 (PANX1, IC50 = 4 μM)。 | |||
T4063 |
Delafloxacin
ABT492,WQ-3034,德拉沙星,RX-3341 |
Antibacterial; Antibiotic | Microbiology/Virology |
Delafloxacin (WQ-3034) 是一种广谱氟喹诺酮类抗生素,抑制耐药性的金黄色葡萄球菌,肺炎链球菌和肺炎克雷伯菌。 | |||
T8142 |
Difloxacin hydrochloride
Difloxacin HCl,盐酸二氟沙星 |
Antibacterial; Antibiotic | Microbiology/Virology |
Difloxacin hydrochloride (Difloxacin HCl) 是一种广谱抗菌药物。它干扰 DNA 促旋酶和拓扑异构酶 IV 的活性,抑制细菌 DNA 促旋酶并显示出浓度依赖性的杀菌作用。 | |||
T12649 |
Ibafloxacine
S25930,Ibafloxacin,R835 |
Antifungal | Microbiology/Virology |
Ibafloxacine (R835) 是一种氟喹诺酮类抗生素,专门用于兽类,对巴氏杆菌显示出良好的抑菌效果。 | |||
T13346L |
WQ3810 TFA
WQ3810 TFA(888032-58-4 Free base),KPI-10 TFA |
Antifungal | Microbiology/Virology |
WQ3810 TFA 是一种可口服的氟喹诺酮,具有抗菌活性,对结核分枝杆菌有抑制作用,抑制氧氟沙星耐药麻风分枝杆菌的 DNA 旋转酶活性。 | |||
T8835 |
Tosufloxacin hydrochloride
A-61827 hydrochloride,盐酸妥舒沙星,T-3262 hydrochloride |
Antibacterial | Microbiology/Virology |
Tosufloxacin hydrochloride 是一种氟喹诺酮类抗菌剂,用于治疗细菌感染。 Tosufloxacin hydrochloride 也是一种细菌 Topo(DNA 促旋酶,拓扑异构酶)抑制剂。 | |||
T1283 |
Clinafloxacin
克林沙星,PD 127391,CI-960,AM-1091 |
Antibacterial; Antibiotic | Microbiology/Virology |
Clinafloxacin (CI-960) 是一种高效广谱氟喹诺酮类抗生素,抑制革兰氏阳性、革兰氏阴性和厌氧病原体。它对金黄色葡萄球菌的 DNA 促旋酶和拓扑异构酶 IV 有抑制作用,IC50值分别为 0.92 µg/ml 和 1.62 µg/ml。 | |||
T0902 |
Ofloxacin
DL8280,菲宁达,Hoe-280,氧氟沙星,Floxin,Tarivid,Oxaldin |
Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Ofloxacin (Oxaldin) 是可抑制细菌DNA 旋转酶的一种氟喹诺酮类抗生素。 | |||
T1625 |
Lomefloxacin hydrochloride
Lomefloxacin HCl,盐酸洛美沙星,Okacyn,Maxaquin |
Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Lomefloxacin hydrochloride (Okacyn) 是一种广谱喹诺酮类抗生素,具有抗菌活性。它可研究支气管炎、尿路感染、结膜炎、外耳炎和中耳炎。 | |||
T5394 |
Prulifloxacin
AF 3012,Pruvel,NM441,普卢利沙星 |
Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Prulifloxacin (NM441) 是一种口服有效的氟喹诺酮抗生素 ,对革兰氏阳性和阴性细菌具有广泛活性。它是噻唑喹啉羧酸衍生物 Ulifloxacin 的前药。它有潜力用于下尿路感染和慢性支气管炎。 | |||
T0331L |
Moxifloxacin
Avelox,Moxeza,莫西沙星 |
Others; Antibacterial; Antibiotic | Microbiology/Virology; Others |
Moxifloxacin (Avelox) 是一种8-甲氧基喹诺酮类口服有效抗菌药物,用于急性细菌性鼻窦炎,慢性支气管炎的急性细菌性加重和感染性肺炎的研究。 | |||
T1451 |
Levofloxacin hydrate
左氧氟沙星半水合物,Levaquin hydrate,Cravit hydrate,Quixin hydrate,Levofloxacin Hemihydrate,Tavanic hydrate,Iquix hydrate |
DNA gyrase; Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Levofloxacin hydrate (Cravit hydrate) 是抗生素化合物,抑制细菌DNA 旋转酶活性。 | |||
T0331 |
Moxifloxacin hydrochloride
盐酸莫西沙星,莫西沙星盐酸盐,BAY-128039,Moxifloxacin HCl,BAY12-8039 HCl |
Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Moxifloxacin hydrochloride (BAY12-8039 HCl) 是一种口服有效的 8-甲氧基喹诺酮类抗菌药物,可研究感染性肺炎,急性细菌性鼻窦炎和慢性支气管炎的急性细菌性加重。 | |||
T8747 |
Levofloxacin hydrochloride
|
DNA gyrase; Topoisomerase | DNA Damage/DNA Repair |
Levofloxacin hydrochloride 是一种广谱的第三代氟喹诺酮类抗生素,是氧氟沙星的光学活性 L-异构体,具有抗菌活性。左氧氟沙星通过细菌细胞壁扩散并通过抑制 DNA 促旋酶(细菌拓扑异构酶 II)起作用,这是一种 DNA 复制、RNA 转录和细菌 DNA 修复所需的酶。 DNA 促旋酶活性的抑制导致细菌细胞生长受阻。 | |||
T16703 |
Quarfloxin
CX-3543 |
DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Quarfloxin (CX-3543) 是一种氟喹诺酮衍生物,具有抗肿瘤活性,可靶向抑制RNA pol I 的活性,在神经母细胞瘤细胞中的 IC50 值在纳摩尔范围内。它破坏核糖体 DNA 模板中核仁蛋白和 G-四链体 DNA 结构之间的相互作用。 | |||
T13346 |
WQ3810
KPI-10 free base |
Others | Others |
WQ3810 is an orally active fluoroquinolone, has potent antibacterial activities. | |||
T22265 |
Balofloxacin Dihydrate
Neuroquinoron,巴洛沙星/1-环丙基-7-(3-甲氨基-1-哌啶基)-8-甲氧基-6-氟-1,4-二氢-4-氧代-3-喹啉羧酸 |
Others | Others |
Balofloxacin is a fluoroquinolone antibiotic with oral activity. | |||
T30684 |
Cadrofloxacin
CS-940,CS 940,Cadrofloxacin hydrochloride,Caderofloxacin,CS940 |
||
Cadrofloxacin (Caderofloxacin, CS-940) is a novel fluoroquinolone antimicrobial agent. | |||
T27818 |
Levonadifloxacin Arginine Salt
WCK 771,WCK-771A,WCK 771A,WCK-771,WCK771A,WCK771 |
||
Levonadifloxacin, a broad-spectrum fluoroquinolone antibiotic, is used potentially for the treatment of staphylococci. | |||
T26449 |
A 80556
A-80556,A80556 |
||
A 80556, a fluoroquinolone antibiotic, has potent antibacterial activity against gram-positive, gram-negative, and anaerobic organisms. | |||
T25461 |
Grepafloxacin, (S)-
L-Grepafloxacin |
||
Grepafloxacin, (S)- is an oral broad-spectrum fluoroquinolone antibacterial used for the treatment of bacterial infections. | |||
T33899 |
PD 131628
PD131628,PD-131628 |
||
PD 131628 is a novel fluoroquinolone that is a bioactive form of PD 131112 or CI-990 for use against anaerobic bacteria. | |||
T23622 |
Acorafloxacin HCl
JNJ-32729463,JNJ-Q2 hydrochloride,Acorafloxacin hydrochloride,JNJ 32729463,JNJ-Q2 HCl |
||
Acorafloxacin is a broad-spectrum fluoroquinolone antibacterial drug being developed for the treatment of acute bacterial skin and skin structure infections and community-acquired pneumonia. | |||
T10420 |
Avarofloxacin
JNJ-Q2 |
Others | Others |
Avarofloxacin (JNJ-Q2) is a broad-spectrum fluoroquinolone antibacterial drug being developed for the treatment of acute bacterial skin and community-acquired pneumonia and skin structure infections. | |||
T36031 |
Desmethyl Ofloxacin (hydrochloride)
|
||
Desmethyl ofloxacin is a metabolite of the fluoroquinolone antibiotic ofloxacin .1 1.Sudo, K., Okazaki, O., Tsumura, M., et al.Isolation and identification of metabolites of ofloxacin in rats, dogs and monkeysXenobiotica16(8)725-732(1986) | |||
T81412 | Pradofloxacin | ||
Pradofloxacin是一种第三代的氟喹诺酮类抗菌化合物。 | |||
T1466L |
Difloxacin HCl
|
||
Difloxacin 是第二代合成的氟喹诺酮抗菌抗生素。 | |||
T71982 |
Ofloxacin HCl
|
||
Ofloxacin HCl is a synthetic fluoroquinolone ( FLUOROQUINOLONES) antibacterial agent that inhibits the supercoiling activity of bacterial DNA GYRASE, halting DNA REPLICATION. | |||
T38586 |
Grepafloxacin
dl-Grepafloxacin,OPC-17116 |
||
Grepafloxacin (OPC-17116) is a fluoroquinolone antibiotic that is administered orally. It possesses strong efficacy against community-acquired respiratory pathogens, notably Streptococcus pneumonia. Grepafloxacin exhibits excellent tissue penetration and demonstrates a promising pharmacodynamic profile. | |||
T26368 |
Tosufloxacin tosylate
Tosufloxacin,T-3262,T3262,T 3262 |
||
Tosufloxacin is a fluoroquinolone antibiotic used to treat susceptible infections. | |||
T31031 |
CP 74667
UNII-D66A707X1B,CP74667,CP-74667 |
||
CP 74667 is a new fluoroquinolone that has good activity against several gram-positive and gram-negative pathogens. | |||
T3522 |
Tosufloxacin tosilate
|
Others | Others |
Tosufloxacin tosilate 是一种氟喹诺酮类抗生素。 | |||
T22797 |
Gatifloxacin mesylate
|
Others | Others |
Gatifloxacin (mesylate) is an antibiotic of the fourth-generation fluoroquinolone family. It also inhibits the bacterial enzymes DNA gyrase and topoisomerase IV. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6567 |
Levofloxacin
Levaquin,Cravit,Tavanic,Fluoroquinolone,左氧氟沙星,(-)-Ofloxacin |
Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Levofloxacin (Fluoroquinolone) 是合成的氟喹诺酮类抗生素,有抑制细菌DNA 旋转酶的超螺旋活性的作用,能阻止DNA 复制。 | |||
T8046 |
Tosufloxacin tosylate hydrate
Tosufloxacin p-Toluenesulfonate Hydrate,A-61827 tosylate hydrate,对甲苯磺酸妥舒沙星水合物,T-3262 Tosylate Hydrate |
Others; Antibacterial; Antibiotic | Microbiology/Virology; Others |
Tosufloxacin tosylate hydrate (A-61827 tosylate hydrate) 是一个氟喹诺酮类抗菌剂。 | |||
T8130 |
Ciprofloxacin hydrochloride monohydrate
Oftacilox,Ciprofloxacin hydrochloride hydrate,Bay-09867 hydrochloride monohydrate,环丙沙星盐酸盐一水合物,Ceprimax,盐酸环丙沙星(一水物),Ciloxan |
Antibacterial; Antibiotic | Microbiology/Virology |
Ciprofloxacin hydrochloride monohydrate (Bay-09867 hydrochloride monohydrate) 是一种具有高效抗菌活性的氟喹诺酮类抗生素。 | |||
T1276 |
Danofloxacin mesylate
甲磺酸达氟沙星,CP 76136-27 |
DNA/RNA Synthesis; Antibacterial; Antibiotic | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology |
Danofloxacin mesylate (CP 76136-27) 是一种兽医用氟喹诺酮类抗菌素。 | |||
T8384 |
Gatifloxacin hydrochloride
AM-1155 (hydrochloride),BMS-206584 (hydrochloride),PD135432 (hydrochloride),加替沙星盐酸盐 |
Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Gatifloxacin hydrochloride (AM-1155 hydrochloride) 是一种氟喹诺酮类抗生素,有广谱抗菌活性。它可抑制大肠杆菌 DNA 解旋酶 (IC50=0.109 μg/ml)和细菌 II 型拓扑异构酶(IC50=13.8 μg/ml) 。它在动物模型中,可研究细菌性结膜炎。 |