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Cat. No.	Product Name	Target	Signaling Pathways
TP1104L	Melanin Concentrating Hormone, salmon acetate MCH (salmon),Melanin Concentrating Hormone, salmon acetate(87218-84-6 free base)	Others; Melanin-concentrating Hormone Receptor (MCHR)	GPCR/G Protein; Others
	Melanin Concentrating Hormone, salmon acetate (MCH (salmon))(87218-84-6 free base) 是一种 19 个氨基酸的环状肽，主要在下丘脑中表达。
TP1104	Melanin Concentrating Hormone, salmon MCH (salmon)
	Melanin Concentrating Hormone (MCH), a 19 amino acid cyclic peptide, is largely expressed in the hypothalamus.
T11966	MCHR1 antagonist 2	HER; Melanin-concentrating Hormone Receptor (MCHR)	Angiogenesis; GPCR/G Protein; JAK/STAT signaling; Tyrosine Kinase/Adaptors
	MCHR1 antagonist 2 是有效的黑色素聚集激素受体 1 拮抗剂，IC50为 65 nM。它也抑制hERG，在IMR-32 细胞中的IC50为 4.0 nM。
T75970	Melanin Concentrating Hormone, salmon TFA
	Melanin Concentrating Hormone, salmon TFA (MCH (salmon) TFA) 是在硬骨鱼的垂体中发现的 19 个氨基酸组成的神经肽，它调节食物摄入，能量平衡，睡眠状态和心血管系统。Melanin Concentrating Hormone, salmon TFA (MCH (salmon) TFA) 是 SLC-1/GPR24和 MCHR2的配体。
TP1102	MCH (salmon) TFA (87218-84-6 free base) Melanin Concentrating Hormone, salmon TFA,MCH (salmon) TFA
	Melanin Concentrating Hormone (MCH), a 19 amino acid cyclic peptide, is largely expressed in the hypothalamus. Melanin Concentrating Hormone is implicated in the control of general arousal and goal-orientated behaviours in mammals, and appears to be a key
T8004	SNAP 94847 hydrochloride	GPR; Melanin-concentrating Hormone Receptor (MCHR)	Endocrinology/Hormones; GPCR/G Protein
	SNAP 94847 hydrochloride 是一种选择性黑色素浓缩激素受体1 拮抗剂，Ki 为 2.2 nM，具有抗抑郁样活性。它是 MCH 诱发的肌醇磷酸形成的高亲和力拮抗剂，pA2为 7.81。
TP1996	MCH(human, mouse, rat) MCH (human, mouse, rat),黑色素聚集激酶素(MCH)( 大鼠)	GPR; Melanin-concentrating Hormone Receptor (MCHR)	Endocrinology/Hormones; GPCR/G Protein
	MCH(human, mouse, rat) 是MCH-R 肽激动剂，对 CHO 细胞系中 MCH-2R 高度敏感，激活 MCH-1R 和 MCH-2R 的IC50 值分别为 0.3 和 1.5 nM，EC50值对分别为 3.9 和 0.1 nM。
T5406	SNAP 94847 SNAP-94847	GPR; Melanin-concentrating Hormone Receptor (MCHR)	Endocrinology/Hormones; GPCR/G Protein
	SNAP 94847 (SNAP-94847) 是一种选择性黑色素浓缩激素受体1 拮抗剂，Ki 为 2.2 nM。它具有抗焦虑和抗抑郁活性，可减少小鼠的食物摄入。
T22591	ATC 0175 hydrochloride	GPR; 5-HT Receptor; Melanin-concentrating Hormone Receptor (MCHR)	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	ATC 0175 hydrochloride 是一种具有口服活性的黑色素细胞浓缩激素1受体拮抗剂，具有强效性和选择性，ATC 0175 hydrochloride 对MCH1R、MCH2R、MCH1、5-HT2B 受体和5-HT1A 受体具有亲和力，IC50分别为为13.5nM、>10,000 nM、13 nM、9.66 nM 和16.9 nM。ATC 0175 hydrochloride 在动物模型中表现出抗抑郁和抗焦虑作用。ATC0175可用于研究抑郁症和/或焦虑症。
T28902	T-226296 T 226296,T226296
	T-226296 is a antagonist of melanin concentrating hormone receptor 1 (MCHR1).
T69170	ATC0065 HCl
	ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.
T11965	MCHR1 antagonist 3	Others	Others
	MCHR1 antagonist 3, a potent antagonist of the melanin-concentrating hormone receptor-1 (MCHR1), is employed for the regulation of energy metabolism.
T28823	SNAP-7941 SNAP7941
	SNAP-7941 is a selective antagonist of the melanin concentrating hormone receptor MCH1 with promising anxiolytic, antidepressant and anorectic effects in initial animal studies.
T26677	ATC0175 ATC 0175,ATC-0175
	ATC0175 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.
T26676	ATC0065 ATC 0065,ATC-0065
	ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.
T16293	NGD-4715	Others	Others
	NGD-4715 is a selective and orally active antagonist of melanin-concentrating hormone receptor 1.
T26703	AZ13483342 AZ-13483342,AZ 13483342
	AZ13483342 is an antagonist of the melanin concentrating hormone receptor 1 (MCH1) with a potential diabetes therapeutic activity.
T16852	SB-568849	Others	Others
	SB-568849 is a melanin-concentrating hormone receptor 1 antagonist (pKi: 7.7).
T10173	MCHR1 antagonist 1	Others	Others
	MCHR1 antagonist 1 is a selective antagonist of melanin-concentrating hormone-1 (MCH1) receptor (Kb: 1 nM, Ki: 4 nM at human MCH1).
T23719	AMG-076
	AMG-076 is an antagonist of melanin-concentrating hormone receptor 1. It also reduced hERG inhibition.
T14372	AZD1979	Others	Others
	AZD1979 is an antagonist of Melanin-concentrating hormone receptor 1 (MCHr1) (IC50: 12 nM).
T15450	GW-803430 GW-3430	Others	Others
	GW-803430 is a potent and selective antagonist of melanin-concentrating hormone receptor 1 (MCH R1) (pIC50: 9.3). GW-803430 is orally active in an animal model of obesity.
T11964	MCH-1 antagonist 1	P450	Metabolism
	MCH-1 antagonist 1 also inhibits CYP3A4 (IC50: 10μM).MCH-1 antagonist 1 is a potent melanin concentrating hormone (MCH-1) antagonist (Ki: 2.6 nM).
T7749	ALB-127158
	ALB-127158(a) 是一种有效的选择性黑色素浓缩激素 1 (MCH1) 受体拮抗剂，可能是炎症性肠病 (IBD) 的潜在治疗方法
T82140	Hypertrehalosemic neuropeptide (Nauphoeta cinerea)
	Hypertrehalosemic neuropeptide (Nauphoeta cinerea) 属于脂动激素/红色素浓缩激素 (AKH/RPCH) 家族，具有促进海藻糖合成的功能。
TP1997	[Ala17]-MCH
	Potent melanin-concentrating hormone (MCH) receptor agonist (EC50 values are 17 and 54 nM at MCH1 and MCH2 receptors respectively). Displays some selectivity towards MCH1 over MCH2 (Ki values are 0.16 and 34 nM respectively).
T76640	hMCH-1R antagonist 1
	hMCH-1R antagonist 1 (Compound 30)为高效且具有选择性的hMCHR1拮抗剂，KB值仅为3.6 nM。它与hMCHR1和hMCHR2的结合能力强，IC50值分别为65 nM与49 nM，主要用于代谢研究领域。
T81319	Quizalofop-P	Acetyl-CoA Carboxylase	Metabolism
	Quizalofop-P被杂草通过茎叶吸收，能在植株内实现向上和向下的双向运输，并在顶端和分生区域累积，通过抑制脂肪酸合成，进而导致杂草死亡。此外，Quizalofop-P对禾本科杂草与双子叶作物具有显著的选择性。
T64692	AMY-101 acetate
	Complement component C3 plays a particularly versatile role in this process by keeping the cascade alert, acting as a point of convergence of activation pathways, fueling the amplification of the complement response, exerting direct effector functions, and helping to coordinate downstream immune responses[3]. In C3-/- mice alcohol-induced liver steatosis is absent or strongly reduced after chronic or acute alcohol exposure. This suggests that the complement system and its component C3 contribute...

化合物

Melanin Concentrating Hormone, salmon acetate

Cat.No: TP1104L

Synonym: MCH (salmon),Melanin Concentrating Hormone, salmon acetate(87218-84-6 free base)

Target: Others, Melanin-concentrating Hormone Receptor (MCHR)

Melanin Concentrating Hormone, salmon

Cat.No: TP1104

Synonym: MCH (salmon)

MCHR1 antagonist 2

Cat.No: T11966

Target: HER, Melanin-concentrating Hormone Receptor (MCHR)

Melanin Concentrating Hormone, salmon TFA

Cat.No: T75970

MCH (salmon) TFA (87218-84-6 free base)

Cat.No: TP1102

Synonym: Melanin Concentrating Hormone, salmon TFA,MCH (salmon) TFA

SNAP 94847 hydrochloride

Cat.No: T8004

Target: GPR, Melanin-concentrating Hormone Receptor (MCHR)

MCH(human, mouse, rat)

Cat.No: TP1996

Synonym: MCH (human, mouse, rat),黑色素聚集激酶素(MCH)( 大鼠)

Target: GPR, Melanin-concentrating Hormone Receptor (MCHR)

Cat.No: T5406

Synonym: SNAP-94847

Target: GPR, Melanin-concentrating Hormone Receptor (MCHR)

ATC 0175 hydrochloride

Cat.No: T22591

Target: GPR, 5-HT Receptor, Melanin-concentrating Hormone Receptor (MCHR)

Cat.No: T28902

Synonym: T 226296,T226296

Cat.No: T69170

MCHR1 antagonist 3

Cat.No: T11965

Target: Others

Cat.No: T28823

Synonym: SNAP7941

Cat.No: T26677

Synonym: ATC 0175,ATC-0175

Cat.No: T26676

Synonym: ATC 0065,ATC-0065

Cat.No: T16293

Target: Others

Cat.No: T26703

Synonym: AZ-13483342,AZ 13483342

Cat.No: T16852

Target: Others

MCHR1 antagonist 1

Cat.No: T10173

Target: Others

Cat.No: T23719

Cat.No: T14372

Target: Others

Cat.No: T15450

Synonym: GW-3430

Target: Others

MCH-1 antagonist 1

Cat.No: T11964

Target: P450

Cat.No: T7749

Hypertrehalosemic neuropeptide (Nauphoeta cinerea)

Cat.No: T82140

Cat.No: TP1997

hMCH-1R antagonist 1

Cat.No: T76640

Cat.No: T81319

Target: Acetyl-CoA Carboxylase

AMY-101 acetate

Cat.No: T64692

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