Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T9022 |
AZD9977
AZD 9977 |
Glucocorticoid Receptor | Endocrinology/Hormones |
AZD9977 是一种选择性的,有效的,具有口服活性的盐皮质激素受体 (MR) 调节剂,可用于研究心力衰竭和慢性肾病。 | |||
T0083 |
Eplerenone
Epoxymexrenone,CGP 30083,依普利酮,SC-66110 |
Glucocorticoid Receptor | Endocrinology/Hormones |
Eplerenone (CGP 30083) 是一种竞争性的、选择性的、具有口服活性的醛固酮 (aldosterone) 拮抗剂,IC50=138 nM。它对孕酮,雄激素,雌激素和糖皮质激素受体的亲和力低,可用于研究高血压和心肌梗死后的心力衰竭。 | |||
T6542 |
Imidapril hydrochloride
Novaloc,Imidapril HCl,盐酸咪达普利,Tanapril,TA-6366 |
RAAS | Endocrinology/Hormones |
Imidapril hydrochloride (Tanapril) 是一种血管紧张素转换酶 (ACE) 抑制剂,具有抗高血压活性。 | |||
T2006 |
Omecamtiv mecarbil
CK-1827452 |
ATPase; Myosin | Cytoskeletal Signaling; Membrane transporter/Ion channel |
Omecamtiv mecarbil (CK-1827452) 是一种心脏特异性的肌球蛋白激活剂,用于研究心脏相关疾病。 | |||
T10631 |
Bucindolol
BMY 13105,MJ 131051,MJ 13105 |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Bucindolol (BMY 13105) 是一种新型有效的 β1 肾上腺素能受体 (β1-adrenergic receptor) 阻滞剂,可介导血管舒张,可用于研究慢性心力衰竭。 | |||
T27596 |
Imazodan hydrochloride
CI914 HCl,CI-914 HCl,CI 914 HCl,Imazodan HCl |
PDE | Metabolism |
Imazodan hydrochloride (CI-914 HCl) 是一种强效的选择性 III 型磷酸二酯酶抑制剂,用于治疗慢性充血性心力衰竭。 | |||
T6486 |
Enalapril Maleate
MK-421 Maleate,Renitec Maleate,Glioten Maleate,MK-421 (maleate),Vasotec Maleate,马来酸依那普利 |
RAAS | Endocrinology/Hormones |
Enalapril Maleate (MK-421 Maleate) 一种是血管紧张素转化酶(ACE)抑制剂。 | |||
T33711L |
Nolomirole HCl
CHF 1035 HCl,CHF 1035,CHF1035,CHF1035 HCl,CHF-1035 HCl,CHF-1035,Nolomirole Hydrochloride |
Dopamine Receptor; Norepinephrine | GPCR/G Protein; Neuroscience |
Nolomirole HCl(CHF 1035) 是一种具有口服活性的新型选择性多巴胺激动剂,对去甲肾上腺素的释放有抑制作用,可用于研究轻度慢性心力衰竭。 | |||
T0154 |
Nebivolol hydrochloride
R 065824 hydrochloride,盐酸奈必洛尔,Nebivolol HCl,R-65824 |
Apoptosis; Adrenergic Receptor | Apoptosis; GPCR/G Protein; Neuroscience |
Nebivolol hydrochloride (R 065824 hydrochloride) 是一种β1-肾上腺素受体选择性抑制剂,IC50为0.8 nM。 | |||
T21395 |
Finerenone
BAY948862,BAY-948862,BAY94-8862,非奈利酮,BAY 94-8862,BAY-94-8862,BAY 948862 |
Glucocorticoid Receptor | Endocrinology/Hormones |
Finerenone (BAY-948862) 是一种选择性、具有口服活性的、非甾体类盐皮质激素受体拮抗剂 (IC50=18 nM)。与糖皮质激素受体、雄激素受体和孕酮受体相比,它表现出良好的选择性 (>500-fold)。它在心肾疾病研究中具有潜在的应用前景,如 2 型糖尿病和慢性肾脏疾病。 | |||
T68138 |
Saterinone
|
Adrenergic Receptor; PDE | GPCR/G Protein; Metabolism; Neuroscience |
Saterinone 是一种强效且具有选择性的磷酸二酯酶III 抑制剂,是血管α - 1-肾上腺素受体的有效拮抗剂。Saterinone 具有血管舒张作用,可用于慢性心力衰竭的急性治疗。Saterinone 对豚鼠右心室匀浆中粗cAMP 磷酸二酯酶(PDE)活性具有抑制作用,ic50值为2.3 × 10(-5) mol/l。 | |||
T13599 |
Benzofurodil
CB4091,Benfurodil,Eudilat |
Others | Others |
Benzofurodil is cardiotonic used for the chronic treatment of congestive heart failure. | |||
T39063 |
Azilsartan mepixetil
|
||
Azilsartan mepixetil is a potent angiotensin II receptor antagonist with enhanced efficacy and prolonged duration of action. It exhibits more prominent and sustained effects in lowering blood pressure and heart rate, while maintaining a high level of safety. Furthermore, Azilsartan mepixetil demonstrates optimal protective efficacy for cardiovascular and renal functions. Hence, it holds promise for the research and treatment of hypertension, chronic heart failure, and diabetic nephropathy. | |||
T61407 |
TRPC3/6-IN-1
|
||
TRPC3/6-IN-1 is a highly potent and selective inhibitor that specifically blocks the activity of the canonical transient receptor channels TRPC3 and TRPC6. It exhibits a significant blocking potency against the human isoforms hTRPC3 and hTRPC6, with IC50 values of 1260 nM and 500 nM, respectively. This compound, TRPC3/6-IN-1, is particularly valuable for conducting research on chronic models of heart failure [1]. | |||
T78657 |
Azilsartan mepixetil potassium
QR-01019K |
||
Azilsartan mepixetil potassium (QR-01019K),是一种高效安全的血管紧张素 II 受体拮抗剂,展现出卓越的持久降压效应以及显著且持续的降心率功能,有望用于治疗高血压、慢性心力衰竭和糖尿病肾病。 | |||
T21485 |
Perindopril
|
||
Perindopril (S-9490) 是一种长效血管紧张素转换酶(ACE)抑制剂,用于治疗高血压、心力衰竭或稳定性冠状动脉疾病。 | |||
T62005 |
Imidapril
|
||
Imidapril (TA-6366 free base) 是口服有效的血管紧张素转换酶(ACE)和MMP-9抑制剂。Imidapril 通过抑制血管紧张素 I 向血管紧张素 II 转化从而降低总外周阻力和血压。Imidapril 在高血压、1 型糖尿病、肾病和慢性心力衰竭中有研究价值。 | |||
T72213 |
Efonidipine hydrochloride
NZ-105 hydrochloride |
||
Efonidipine(NZ-105)盐酸盐是T 型和L 型钙离子通道双重阻断剂。 |