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Cat. No. Product Name Target Signaling Pathways
T18893 5(6)-Carboxyfluorescein

5(6)-羧基荧光素,5-(and-6)-Carboxyfluorescein mixed isomers,5(6)-FAM

Others Others
5(6)-Carboxyfluorescein (5-(and-6)-Carboxyfluorescein mixed isomers) 是一种胺反应性 pH 敏感的绿色荧光标记物,能够标记蛋白质、多肽和氨基酸,可用于体内实验检测肿瘤位置。
T77456 Lumiliximab

IDEC-152,ST-152

Lumiliximab (IDEC-152) 是一种灵长类化的靶向 CD23 猕猴/人嵌合抗体,对 IgE 抗体的产生有抑制作用,用于研究过敏性疾病。
T76844 Abciximab

C7E3

Integrin Cytoskeletal Signaling
Abciximab (C7E3) 是一种小鼠/人嵌合单克隆抗体,是一种有效的糖蛋白 IIb/IIIa (glycoprotein IIb/IIIa) 抑制剂。 Abciximab 具有抗血小板聚集和白细胞粘附的作用,通过与糖蛋白 IIb/IIIa、vitronectin 和 Mac-1 受体结合发挥作用。
T9910 Rituximab

Others Others
Rituximab 是抗 CD20 嵌合单克隆抗体,用于研究某些自身免疫疾病和癌症。
T22889 KF38789

KF 38789

Others Others
KF38789 特异性的抑制P-selectin 与PSGL-1结合。它对 U937 细胞与 P-selectin 免疫球蛋白 G 嵌合蛋白 (P-selectin-Ig) 的结合具有抑制作用 (IC50:1.97 μM) 。
T76671 Amatuximab

MORab-009

Others Others
Amatuximab (MORab-009) 是一种人源化针对细胞表面间皮素 (MSLN) 的嵌合 IgG1/k 单抗,具有抗肿瘤活性,可用于治疗实体肿瘤。
T73698 Basiliximab

CHI 621

Interleukin Immunology/Inflammation
Basiliximab (CHI 621) 是一种嵌合鼠/人 IgG1 单克隆抗白细胞介素 2 受体 (interleukin-2 receptor) 重组抗体。Basiliximab 具有良好的免疫抑制活性,可用于研究肾移植。
T76718 Brentuximab

TNF Apoptosis
Brentuximab 是靶向 CD30 的嵌合抗体,是 Brentuximab vedotin 的裸抗。Brentuximab 具有抗肿瘤活性,可用于研究复发或难治性霍奇金淋巴瘤。
T76773 Rolinsatamab

IL Receptor Immunology/Inflammation
Rolinsatamab 是一种完全人源化的选择性单克隆抗体,是一种有效的 IL-4 和 IL-13 双重抑制剂。Rolinsatamab 嵌合抗原受体序列 T 细胞。Rolinsatamab 可用于预防和治疗免疫疾病。
T76830 Teneliximab

Chi220,Anti-Human CD40 Recombinant Antibody,BMS 224819

TNF Apoptosis
Teneliximab (Chi220) 是一种嵌合的单克隆抗体,也是一种肿瘤坏死因子受体超家族成员5(CD40)抑制剂,可阻断CD40-CD40L 的相互作用。Teneliximab 通过CD40 和外周B细胞损耗发挥部分激动剂活性,可用于研究器官移植排斥和类风湿关节炎。
TP1991L M 1145 acetate

Neuropeptide Y Receptor GPCR/G Protein; Neuroscience
M1145 acetate 是一种嵌合肽,是一种选择性甘丙肽受体 2 (GAL2) 激动剂,Ki 为 6.55 nM。它对 GAL2 的亲和力比 GAL1 高 90 倍以上(Ki=587 nM),比 GalR3 的亲和力高 76 倍(Ki=497 nM)。 它对甘丙肽的信号转导具有累加作用。
T77484 Atibuclimab

TNF Apoptosis
Atibuclimab 是一种靶向 CD14 的嵌合单克隆抗体,由小鼠可变区和人类 IgG4 Fc 区构成。Atibuclimab 可用于治疗肌萎缩侧索硬化症。Atibuclimab 可减少 LPS 诱导的病症,并对 LPS 诱导的促炎细胞因子释放有抑制作用,可延迟抗炎细胞因子可溶性 TNF 受体 I 型的释放,
T39954 AU-15330

Epigenetic Reader Domain; PROTACs Chromatin/Epigenetic; PROTAC
AU-15330是SWI/SNF ATPase亚基SMARCA2和SMARCA4的蛋白水解靶向嵌合体(PROTAC)降解剂。AU-15330 能有效抑制肿瘤在前列腺癌异种移植模型中的生长,并与 AR 拮抗剂恩杂鲁胺具有协同作用。AU-15330在去势抵抗性前列腺癌(CRPC)模型中显示出部分治疗效果和AU-15330具有无毒性的特点。
T15517 Hydroxy-PEG2-C2-PFP ester

Others Others
Hydroxy-PEG2-C2-PFP ester, a PEG/Alkyl/ether-based PROteolysis TArgeting Chimeric (PROTAC) linker, is suitable for the synthesis of PROTACs.
T31949 Glutathione amide

GASH cpd,L-gamma-Glutamyl-L-cysteinylglycinamide

Glutathione amide is a enzyme of a chimeric protein.
T78339 Human IgG4 (S228P) kappa, Isotype Control

HumanIgG4(S228P) kappa, Isotype Control为人-鼠嵌合型单克隆抗体,作为humanIgG4(S228P)κ抗体的同型对照使用。
T82159 Human IgG1 (K214R) kappa, Isotype Control

HumanIgG1(K214R) kappa, Isotype Control为HumanIgG1(K214R)κ 抗体的人源化同型对照,属于人-鼠嵌合型抗体。
T39364 Desthiobiotin-PEG4-propargyl

Desthiobiotin-PEG4-propargyl

Desthiobiotin-PEG4-propargyl is a PEG-coupled PROteolysis TArgeting Chimeric (PROTAC) linker, employed for PROTAC synthesis.
T34858 THIQ-20c

THIQ 20c

THIQ-20c is a steroidomimetic and chimeric microtubule disruptor.
T15512 Hydroxy-PEG1-(CH2)2-Boc

Others Others
Hydroxy-PEG1-(CH2)2-Boc is a polyethylene glycol (PEG)-based linker used in the synthesis of proteolysis-targeting chimeric molecules (PROTACs)[1].
T76689 Margetuximab

Margetuximab (MGAH22)为优化Fc结构域的嵌合抗HER2单克隆抗体,EC50值为39.33 ng/mL,适用于转移性HER2阳性乳腺癌研究。
T81247 Runimotamab

Runimotamab为针对CD3E和HER2的IgG1-κ型人源化嵌合单克隆抗体。
T18857 Tri(Amino-PEG3-amide)-amine

Others Others
Tri(Amino-PEG3-amide)-amine is a polyethylene glycol (PEG)-derived linker employed for the synthesis of proteolysis-targeting chimeric molecules (PROTACs)[1].
T80564 Vamikibart

Vamikibart为针对IL-6的人源化嵌合IgG2κ抗体。
T40886 Onzigolide

BIM-23A760,TBR-760,Onzigolide

Onzigolide (BIM-23A760), a chimeric compound combining properties of both dopamine and somatostatin, exhibits strong agonistic activity towards the D2 subtype of dopamine receptors (D2R) as well as type 2 somatostatin receptors (SSTR2).
T39191 DSTYSLSSTLTLSK

DSTYSLSSTLTLSK is a generic human peptide and can be used for infliximab quantitative detection. Infliximab (Avakine) is a chimeric monoclonal IgG1 antibody that specifically binds to TNF-α.
T27461 GSK2336805

GSK 2336805,GSK-2336805,JNJ-56914845,GSK-805,GSK805

GSK-2336805 is a HCV NS5A inhibitor. GSK2336805 retained activity on chimeric replicons containing NS5A patient sequences from genotype 1 and patient and consensus sequences for genotypes 4 and 5 and part of genotype 6.
T17363 β-Naphthoflavone-CH2-OH

β-NF-CH2-OH

Others Others
β-Naphthoflavone-CH2-OH (β-NF-CH2-OH) serves as an AhR E3 ligase ligand, forming chimeric molecules when connected to a protein ligand through a linker, resulting in PROTACs or SNIPERs (e.g., β-naphthoflavone-JQ1). These chimeric molecules recruit the AhR E3 ligase complex by incorporating AhR ligands. By inducing ubiquitination-mediated degradation, PROTACs effectively target and degrade cancer-promoting proteins [1].
T77496L AZD 1775 Linker Conjugate 1 TFA

AZD 1775 Linker Conjugate 1 TFA( 2101954-45-2 Free base)

AZD 1775 Linker Conjugate 1 TFA 是一种参与泛素酶靶向嵌合体实验的化合物。
T16190 N-(Azido-PEG3)-N-Boc-PEG4-Boc

Others Others
N-(Azido-PEG3)-N-Boc-PEG4-Boc is a polyethylene glycol (PEG)-based proteolysis targeting chimeric (PROTAC) linker employed in PROTAC synthesis[1].
T39521 LEESGGGLVQPGGSMK

LEESGGGLVQPGGSMK, a proteolysis peptide, is a constituent of Infliximab, a chimeric monoclonal IgG1 antibody that selectively binds to TNF-α. It can be employed for quantitative assessment of Infliximab.
T17458 Azide-PEG-amine (MW 3500)

Others Others
Azide-PEG-amine (MW 3500) is a polyethylene glycol (PEG) derived linker compound, specifically designed for the synthesis of proteolysis targeting chimeric molecules (PROTACs)[1].
T80606 Duvortuxizumab

MGD 011

Duvortuxizumab (MGD 011) 是一种嵌合人源化IG抗体,特异性靶向CD19和CD3E。
T16310 NH2-PEG1-CH2CH2-Boc

Others Others
NH2-PEG1-CH2CH2-Boc is a polyethylene glycol (PEG) and alkyl/ether-based proteolysis targeting chimeric (PROTAC) linker, commonly employed in the synthesis of PROTACs[1].
T77051 Larcaviximab

Larcaviximab (c4G7-N) 是一种IgG1kappa 抗Ebola virus 糖蛋白嵌合单克隆抗体。
T18603 PROTAC BRD4 degrader for PAC-1

Others Others
PROTAC BRD4 degrader for PAC-1 (compound 5) is a chimeric BET degrader GNE-987 conjugated with a disulfide-containing linker[1]. This PROTAC-linker conjugate specifically targets and degrades BRD4, enabling selective proteolysis of PAC-1.
T82575 Devextinetug

IXT-M200

Devextinetug (IXT-M200) 是一种小鼠源IgG2κ抗体,其特异性针对嵌合抗甲基苯丙胺 (Methamphetamine)。
T80610 Romilkimab

SAR156597

Romilkimab (SAR156597),一种特异性结合IL-4与IL-13的嵌合人源化IG抗体。
T82157 Human IgG1 lambda1, Isotype Control

HumanIgG1lambda1, Isotype Control为人-鼠嵌合型单克隆抗体,作为human IgG1λ1抗体的同型对照物。
T75103 CD19 CAR mRNA

CD19CAR mRNA 能够编码CD19car蛋白,适用于CAR-T细胞免疫治疗(CAR-CD19)。CD19car作为嵌合抗原受体,针对B细胞表面的CD19,一种关键参与B细胞增殖、分化、活化及产生抗体的CD分子(即白细胞分化抗原),进而增强BCR信号传递。
T77150 Cosfroviximab

Cosfroviximab(c13C6-FR1)是一种抗埃博拉病毒糖蛋白(EBOV-GP)的鼠/人嵌合单克隆抗体。
T77015 Futuximab

Futuximab 是一种嵌合单克隆抗体,靶向 EGFR 上的非重叠表位。Futuximab 具有抗肿瘤活性。
T82961 ASB20123

ASB20123 是一款融合了CNP/ghrelin序列的嵌合肽,具有促进骨骼生长的效能,适用于研究生长障碍和侏儒症。
T81174 Setoxaximab

Setoxaximab是一种IgG1-κ型的人源化嵌合单克隆抗体,专门针对shiga toxin 1。
T36091 LEESGGGLVQPGGSMK acetate

LEESGGGLVQPGGSMK acetate is a proteolysis peptide found in Infliximab, a chimeric monoclonal IgG1 antibody. It serves as a component of Infliximab and can be employed for the quantitative analysis of this antibody. Infliximab is specifically designed to bind to TNF-α[1].
T76209 DSTYSLSSTLTLSK TFA

DSTYSLSSTLTLSK TFA 是用于 Infliximab (Avakine) 定量检测的通用肽。Infliximab (Avakine) 是一种嵌合单克隆IgG1抗体,能特异性地结合到 TNF-α。
T82161 Human IgG1 (D265A) kappa, Isotype Control

HumanIgG1(D265A) kappa, Isotype Control是一种人鼠嵌合型抗体,用作HumanIgG1(D265A)κ抗体的同型对照。
T80871 Veligrotug

IGF-1R Tyrosine Kinase/Adaptors
Veligrotug为IgG1-kappa型抗IGF1R(胰岛素样生长因子1受体,CD221)嵌合单克隆抗体。
T80567 Boserolimab

MK-5890

Boserolimab (MK-5890)为一款嵌合人源化IgG1κ抗体,其特异性靶向小鼠CD27信号调节蛋白。
T82155 Human IgG4 (S228P) lambda1, Isotype Control

HumanIgG4(S228P) lambda1, Isotype Control,为人-鼠嵌合型抗体,作为humanIgG4(S228P) λ1抗体同型对照使用。

化合物

5(6)-Carboxyfluorescein
Cat.No: T18893
Synonym: 5(6)-羧基荧光素,5-(and-6)-Carboxyfluorescein mixed isomers,5(6)-FAM
Target: Others
Lumiliximab
Cat.No: T77456
Synonym: IDEC-152,ST-152
Target:
Abciximab
Cat.No: T76844
Synonym: C7E3
Target: Integrin
Rituximab
Cat.No: T9910
Synonym:
Target: Others
KF38789
Cat.No: T22889
Synonym: KF 38789
Target: Others
Amatuximab
Cat.No: T76671
Synonym: MORab-009
Target: Others
Basiliximab
Cat.No: T73698
Synonym: CHI 621
Target: Interleukin
Brentuximab
Cat.No: T76718
Synonym:
Target: TNF
Rolinsatamab
Cat.No: T76773
Synonym:
Target: IL Receptor
Teneliximab
Cat.No: T76830
Synonym: Chi220,Anti-Human CD40 Recombinant Antibody,BMS 224819
Target: TNF
M 1145 acetate
Cat.No: TP1991L
Synonym:
Target: Neuropeptide Y Receptor
Atibuclimab
Cat.No: T77484
Synonym:
Target: TNF
AU-15330
Cat.No: T39954
Synonym:
Target: Epigenetic Reader Domain, PROTACs
Hydroxy-PEG2-C2-PFP ester
Cat.No: T15517
Synonym:
Target: Others
Glutathione amide
Cat.No: T31949
Synonym: GASH cpd,L-gamma-Glutamyl-L-cysteinylglycinamide
Target:
Human IgG4 (S228P) kappa, Isotype Control
Cat.No: T78339
Synonym:
Target:
Human IgG1 (K214R) kappa, Isotype Control
Cat.No: T82159
Synonym:
Target:
Desthiobiotin-PEG4-propargyl
Cat.No: T39364
Synonym: Desthiobiotin-PEG4-propargyl
Target:
THIQ-20c
Cat.No: T34858
Synonym: THIQ 20c
Target:
Hydroxy-PEG1-(CH2)2-Boc
Cat.No: T15512
Synonym:
Target: Others
Margetuximab
Cat.No: T76689
Synonym:
Target:
Runimotamab
Cat.No: T81247
Synonym:
Target:
Tri(Amino-PEG3-amide)-amine
Cat.No: T18857
Synonym:
Target: Others
Vamikibart
Cat.No: T80564
Synonym:
Target:
Onzigolide
Cat.No: T40886
Synonym: BIM-23A760,TBR-760,Onzigolide
Target:
DSTYSLSSTLTLSK
Cat.No: T39191
Synonym:
Target:
GSK2336805
Cat.No: T27461
Synonym: GSK 2336805,GSK-2336805,JNJ-56914845,GSK-805,GSK805
Target:
β-Naphthoflavone-CH2-OH
Cat.No: T17363
Synonym: β-NF-CH2-OH
Target: Others
AZD 1775 Linker Conjugate 1 TFA
Cat.No: T77496L
Synonym: AZD 1775 Linker Conjugate 1 TFA( 2101954-45-2 Free base)
Target:
N-(Azido-PEG3)-N-Boc-PEG4-Boc
Cat.No: T16190
Synonym:
Target: Others
LEESGGGLVQPGGSMK
Cat.No: T39521
Synonym:
Target:
Azide-PEG-amine (MW 3500)
Cat.No: T17458
Synonym:
Target: Others
Duvortuxizumab
Cat.No: T80606
Synonym: MGD 011
Target:
NH2-PEG1-CH2CH2-Boc
Cat.No: T16310
Synonym:
Target: Others
Larcaviximab
Cat.No: T77051
Synonym:
Target:
PROTAC BRD4 degrader for PAC-1
Cat.No: T18603
Synonym:
Target: Others
Devextinetug
Cat.No: T82575
Synonym: IXT-M200
Target:
Romilkimab
Cat.No: T80610
Synonym: SAR156597
Target:
Human IgG1 lambda1, Isotype Control
Cat.No: T82157
Synonym:
Target:
CD19 CAR mRNA
Cat.No: T75103
Synonym:
Target:
Cosfroviximab
Cat.No: T77150
Synonym:
Target:
Futuximab
Cat.No: T77015
Synonym:
Target:
ASB20123
Cat.No: T82961
Synonym:
Target:
Setoxaximab
Cat.No: T81174
Synonym:
Target:
LEESGGGLVQPGGSMK acetate
Cat.No: T36091
Synonym:
Target:
DSTYSLSSTLTLSK TFA
Cat.No: T76209
Synonym:
Target:
Human IgG1 (D265A) kappa, Isotype Control
Cat.No: T82161
Synonym:
Target:
Veligrotug
Cat.No: T80871
Synonym:
Target: IGF-1R
Boserolimab
Cat.No: T80567
Synonym: MK-5890
Target:
Human IgG4 (S228P) lambda1, Isotype Control
Cat.No: T82155
Synonym:
Target:
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