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Cat. No. Product Name Target Signaling Pathways
T6283 Wortmannin

SL-2052,渥曼青霉素,KY-12420

ATM/ATR; DNA-PK; Serine/threonin kinase; PLK; PI3K; Antibiotic; Autophagy Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology; PI3K/Akt/mTOR signaling
Wortmannin (SL-2052) 是一种 PI3K 抑制剂 (IC50=3 nM),具有共价性和不可逆性。Wortmannin 也是一种 PlK1 和 PlK3 的抑制剂 (IC50=5.8/48 nM),可以阻断自噬。
T36314 Wortmannin-Rapamycin Conjugate

Phosphoinositide 3-kinase (PI3K) and mammalian target of rapamycin (mTOR) act synergistically in promoting cancer. Wortmannin is a potent inhibitor of PI3K enzymes, while rapamycin blocks mTOR Complex 1 TORC1. Wortmannin-rapamycin conjugate consists of analogs of 17-hydroxy wortmannin and rapamycin conjugated via a prodrug linker. Hydrolysis of the prodrug linker in vivo releases the inhibitors. The wortmannin-rapamycin conjugate inhibits the growth of HT-29 colon tumors and A498 renal tumors in...
T12870 SCH79797 dihydrochloride

Apoptosis; Others; Protease-activated Receptor Apoptosis; GPCR/G Protein; Others
SCH79797 dihydrochloride 是一种有效的特异性蛋白酶激活受体 1 (PAR1) 拮抗剂,IC50 为 70 nM,Ki 为 35 nM。SCH79797 dihydrochloride 具有抗增殖和促凋亡作用。
T4079 LY-294002 hydrochloride

SF 1101,LY 294002,NSC 697286

PI3K PI3K/Akt/mTOR signaling
LY-294002 hydrochloride (NSC 697286) 是一种合成的 PI3Kα/δ/β 分子抑制剂(IC50:0.5/0.57/0.97 μM,在无细胞试验中);在溶液中比 Wortmannin 更稳定,也是自噬体形成的阻断剂。

化合物

Wortmannin
Cat.No: T6283
Synonym: SL-2052,渥曼青霉素,KY-12420
Target: ATM/ATR, DNA-PK, Serine/threonin kinase, PLK, PI3K, Antibiotic, Autophagy
Wortmannin-Rapamycin Conjugate
Cat.No: T36314
Synonym:
Target:
SCH79797 dihydrochloride
Cat.No: T12870
Synonym:
Target: Apoptosis, Others, Protease-activated Receptor
LY-294002 hydrochloride
Cat.No: T4079
Synonym: SF 1101,LY 294002,NSC 697286
Target: PI3K
TargetMol Loading
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