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Cat. No.	Product Name	Target	Signaling Pathways
T38111	Dimethyl-W84 (dibromide) Dimethyl-W84 (dibromide)
	Dimethyl-W84 is a selective allosteric modulator of the M2 muscarinic acetylcholine receptor. It hinders the dissociation of the orthosteric antagonist N-methylscopolamine from the M2 receptor with an EC50 value of 3 nM.
T23524	W-84 dibromide HDMPPA	AChR	Neuroscience
	W-84 dibromide (HDMPPA) 是 M2胆碱受体的强变构调节剂，是一种非竞争性毒蕈碱乙酰胆碱受体拮抗剂，具有变构效应。它联合阿托品时，可有效地防止有机磷中毒。它阻碍 [3H]N-甲基东莨菪碱解离，能稳定胆碱能拮抗剂-受体复合物。
T15454	GW843682X GW843682	VEGFR; PLK; CDK; PDGFR; Aurora Kinase	Angiogenesis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Tyrosine Kinase/Adaptors
	GW843682X (GW843682) 是 PLK1 和 PLK3 的特异性和 ATP 竞争性抑制剂，IC50 分别为 2.2 nM 和 9.1 nM。
T6527	GW842166X 2-(2,4-二氯苯基氨基)-4-三氟甲基嘧啶-5-羧酸[(四氢吡喃-4-基)甲基]酰胺	Cannabinoid Receptor	GPCR/G Protein
	GW842166X 是一种选择性 cannabinoid receptor 2 激活剂，IC50=63 nM。
T69571	SEW84
	SEW84 是 Aha1 刺激的 Hsp90(ASH) ATP 酶活性的抑制剂。SEW84 抑制 Aha1 刺激的 Hsp90(ASH) 活性，IC50值为 0.3 μM。SEW84 可用于蛋白质沉积疾病的研究。
T27517	GW848687X GW-848687X,GW 848687X
	GW848687X, a potent and selective prostaglandin EP1 receptor antagonist, is used for the treatment of inflammatory pain.
T27516	GW844520
	GW844520 is a potent and selective inhibitor of the cytochrome bc1 complex of mitochondrial electron transport in P. falciparum.
T36574	GW841819X GW841819X
	GW841819X is an analogue of (+)-JQ1 and a novel inhibitor of BET bromodomains. GW841819X was a single enantiomer but of undefined chirality at the 4-position of the benzodiazepine ring3. GW841819X and JQ1 were recently discovered that bind to the acetyl-lysine binding pocket of BET bromodomains with Kd ranges from 50 to 370 nM [1]. GW841819X bounded to both the individual BD1 and BD2 domains with affinities of 46 and 52.5 nM, respectively. GW841819X-Brd3 interaction was estimated to be around 70...

化合物

Dimethyl-W84 (dibromide)

Cat.No: T38111

Synonym: Dimethyl-W84 (dibromide)

Cat.No: T23524

Synonym: HDMPPA

Target: AChR

Cat.No: T15454

Synonym: GW843682

Target: VEGFR, PLK, CDK, PDGFR, Aurora Kinase

Cat.No: T6527

Synonym: 2-(2,4-二氯苯基氨基)-4-三氟甲基嘧啶-5-羧酸[(四氢吡喃-4-基)甲基]酰胺

Target: Cannabinoid Receptor

Cat.No: T69571

Cat.No: T27517

Synonym: GW-848687X,GW 848687X

Cat.No: T27516

Cat.No: T36574

Synonym: GW841819X

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