219
14
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T40840 |
H-Tyr-Ala-OH
H-Tyr-Ala-OH,Tyrosylalanine |
Others | Others |
H-Tyr-Ala-OH (Tyrosylalanine) 是一种L-酪氨酸和L-丙氨酸组成的二肽。 | |||
T36352 |
Suc-Leu-Tyr-AMC
|
||
Suc-Leu-Tyr-AMC 是钙蛋白酶 I 和 II 以及木瓜蛋白酶(另一种半胱氨酸蛋白酶)的荧光底物,用于测量 20S 蛋白酶体的糜蛋白酶样肽酶活性(Ex-max:360 nm;Em-max:460 nm)。Suc-Leu-Tyr-AMC 也能被大肠杆菌的 Ti 蛋白酶裂解。 | |||
T78223 |
γ-Glu-Tyr
gamma-Glutamyltyrosine,gamma-GLU-TYR |
||
γ-Glu-Tyr (gamma-Glutamyltyrosine) 是一种对二肽基肽酶-IV (DPP-IV) 具有竞争性抑制作用的 kokumi 肽,可用于研究糖尿病。 | |||
TP2333 |
cyclo(L-Pro-L-Tyr)
|
Others | Others |
cyclo(L-Pro-L-Tyr) 是真菌和细菌的次生代谢产物。 | |||
TP1164 |
N-Formyl-Nle-Leu-Phe-Nle-Tyr-Lys TFA
For-Nle-Leu-Phe-Nle-Tyr-Lys-OH (TFA) |
Others | Others |
N-Formyl-Nle-Leu-Phe-Nle-Tyr-Lys TFA (For-Nle-Leu-Phe-Nle-Tyr-Lys-OH (TFA)) (71901-21-8 free base) 是一种甲酰肽受体 (FPR) 激动剂 。人类中性粒细胞。放射性碘化分子具有充分的生物活性。 | |||
TP1790L |
Tyr-Somatostatin-14 acetate(58100-03-1 free base)
|
Others | Others |
Tyr-Somatostatin-14 acetate(58100-03-1 free base) 是一种定制肽,可在 Somatostatin-14 中添加酪氨酸氨基酸。 | |||
T7211 |
Tyr-Gly-Gly-Phe-Met-OH
Methionine enkephalin,蛋氨酸脑啡肽,Met-Enkephalin,[MET5]脑啡肽 |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin) 是天然存在的内源性阿片肽、metenkephalin 和 zeta-和 delta-阿片受体激动剂的合成形式,是 mu-阿片受体激动剂,具有潜在的镇痛、神经调节、免疫调节、抗炎、抗肿瘤作用以及镇痛、抗抑郁和胃肠运动调节活性。 | |||
TP1708L |
H-Ala-Ala-Tyr-OH acetate(67131-52-6 free base)
|
Others | Others |
H-Ala-Ala-Tyr-OH acetate(67131-52-6 free base) 可以合成突变肽。 | |||
T36347 |
Ac-YVAD-CMK
Caspase-1 Inhibitor II,Ac-Tyr-Val-Ala-Asp-chloromethylketone,Ac-Tyr-Val-Ala-Asp-CMK |
IL Receptor; Caspase; Immunology/Inflammation related; Pyroptosis | Apoptosis; Immunology/Inflammation; Proteases/Proteasome |
Ac-YVAD-CMK (Ac-Tyr-Val-Ala-Asp-CMK) 是一种选择性的、不可逆的Caspase-1抑制剂,并能抑制焦亡作用、IL-1β和IL-18。Ac-YVAD-CMK 显示出神经保护和抗炎的能力。 | |||
TP1790 |
Tyr-Somatostatin-14
|
||
Tyr-Somatostatin-14 is a modified peptide incorporating an additional Tyrosine (amino acid) into the structure of Somatostatin-14. | |||
T40666 |
Cyclo(Gly-Tyr)
|
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Cyclo(Gly-Tyr) is a cyclic dipeptide. | |||
T31636 |
Enkephalin-met, tyr-O-sulfate
METOS,Met-enkephalin, tyr-O-sulfate-,Tyr-O-sulfate-met-enkephalin |
||
Enkephalin-met, tyr-O-sulfate is a opioid peptide. | |||
TP1251L |
N-terminally acetylated Endomorphin-1 acetate
Ac-L-Tyr-L-Pro-L-Trp-L-Phe-CONH2 |
Others | Others |
N-terminally acetylated Endomorphin-1 acetate (Ac-L-Tyr-L-Pro-L-Trp-L-Phe-CONH2) 是一种修饰的 Endomorphin-1。 | |||
T30557 |
Boc-Gly-Tyr-Lys
|
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Boc-Gly-Tyr-Lys is a peptide. | |||
T36555 |
Tyr-α-CGRP (human) (trifluoroacetate salt)
|
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Tyr-α-CGRP is an N-terminal extended tyrosinated analogue of α-calcitonin gene-related peptide . It binds to amylin receptors AMY1 and AMY3 in COS-7 cells expressing the human receptors (IC50s = 141 and 1.86 nM, respectively). Tyr-α-CGRP also binds to and stimulates cAMP accumulation in rat L6 myocytes (IC50 = 4 nM; EC50 = 12 nM). It also binds to rat brain and spleen membrane preparations (IC50s = 0.2 and 0.5 nM, respectively), induces positive chronotropic and inotropic effects in isolated rig... | |||
T38190 |
Tyr-α-CGRP (rat) (trifluoroacetate salt)
|
||
Tyr-α-CGRP (rat) is an N-terminally tyrosinated analog of the neuropeptide α-CGRP that induces a fall in resting tension of isolated opossum internal anal sphincter (IAS) with an EC50 value of 178 nM. | |||
T38697 |
[Tyr(P)4] Angiotensin II
|
||
[Tyr(P)4] Angiotensin II is a peptide that exerts a multitude of effects on vascular smooth muscle. These effects include the contraction of normal arteries, as well as the induction of hypertrophy or hyperplasia in cultured cells or diseased vessels. | |||
T35753 |
Z-Phe-Tyr(tBu)-diazomethylketone
|
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Irreversible cathepsin L inhibitor which is ca 10'000 times more effective in inactivating cathepsin L than cathepsin S. | |||
TP1708 |
H-Ala-Ala-Tyr-OH
|
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H-Ala-Ala-Tyr-OH can be synthesized mutant peptides. | |||
T36352L |
Suc-Leu-Tyr-AMC Acetate
Suc-Leu-Tyr-AMC Acetate(94367-20-1 Free base) |
Others | Others |
Suc-Leu-Tyr-AMC Acetate 在高浓度时抑制酪蛋白分解。 | |||
T39793 |
Fmoc-Tyr(3-F,tBu)-OH
|
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Fmoc-Tyr(3-F, tBu)-OH is a cyclic peptide compound possessing high membrane permeability and exhibiting specific binding affinity towards a target molecule. | |||
T36353 |
Suc-Tyr-Val-Ala-Asp-pNA
|
||
Suc-YVAD-pNA, a chromogenic caspase-1 substrate. | |||
T21521L |
Papain Inhibitor acetate
乙氨酸-乙氨酸-酪氨酸-精氨酸,GGYR,Gly-Gly-Tyr-Arg,Papain Inhibitor acetate (70195-20-9 free base) |
Others | Others |
Papain Inhibitor acetate (Gly-Gly-Tyr-Arg) 是木瓜蛋白酶的亲和配体。 | |||
TP1308 |
Suc-Leu-Leu-Val-Tyr-AMC
|
||
Suc-Leu-Leu-Val-Tyr-AMC is a fluorescent substrate for the 20S proteasome, other chymotrypsin-like proteases. | |||
T7376 |
Dihexa
PNB-0408,Hexanoyl-Tyr-Ile-Ahx-NH2,N-hexanoic-Try-Ile-(6)-amino hexanoic amide |
c-Met/HGFR | Tyrosine Kinase/Adaptors |
Dihexa (Hexanoyl-Tyr-Ile-Ahx-NH2) 是肝细胞生长因子/c-Met (HGF/c-Met) 系统的激活剂,它与 HGF (Kd = 65 pM) 结合,是肽血管紧张素 IV 的类似物。 | |||
T7339 |
Angiotensin (1-7)
Ang-(1-7),Angiotensin 1-7,ASP-ARG-VAL-TYR-ILE-HIS-PRO |
RAAS; Endogenous Metabolite | Endocrinology/Hormones; Metabolism |
Angiotensin (1-7) (ASP-ARG-VAL-TYR-ILE-HIS-PRO) 是肾素-血管紧张素系统中的内源性七肽。Angiotensin 1-7在心肌细胞中具有抗炎和抗纤维化活性,因此具有心脏保护作用。它能抑制血管紧张素转换酶和释放一氧化氮,是激肽诱导的血管舒张的局部协同调节剂。它阻断 Ang II 诱导的平滑肌细胞增殖和肥大,并显示对内皮的抗血管生成和生长抑制作用。它显示出抗炎活性。 | |||
TQ0143 |
N-Formyl-Nle-Leu-Phe-Nle-Tyr-Lys
For-Nle-Leu-Phe-Nle-Tyr-Lys-OH |
Others | Others |
N-Formyl-Nle-Leu-Phe-Nle-Tyr-Lys TFA is a formyl peptide receptor (FPR) agonist. | |||
TP2085 |
Ac-Tyr(PO3H2)-Glu-Glu-Ile-Glu-OH
N-Acetyl-O-phosphono-Tyr-Glu-Glu-Ile-Glu |
||
Phosphopeptide ligand for the src SH2 domain (IC50 = 1 μM). Blocks src interactions with EGFR and FAK. | |||
TP2136 |
(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
|
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Selective vasopressin V1A receptor antagonist. Inhibits vasopressin and oxytocin-induced increases in intracellular calcium concentrations in vitro (IC50 values are 5 and 30 nM respectively). Exhibits potent and prolonged antivasopressor activity and indu | |||
TP2084 |
N-Acetyl-O-phosphono-Tyr-Glu Dipentylamide
|
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Phosphopeptide; binds to the src SH2 domain. | |||
T21459 |
Splenopentin diacetate
Thymopoietin III pentapeptide (32-36),SP5,Splenopentin Acetate,醋酸脾脏五肽,Splenin pentapeptide (32-36),Arg-lys-glu-val-tyr |
Others | Others |
Splenopentin diacetate (Splenin pentapeptide (32-36)) 是一种合成的免疫调节肽,可以再现脾和胸腺激素胸腺生成素的生物活性。 | |||
T80137 |
(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin
d(CH2)5[Tyr(Me)2, Dab5]AVP |
Vasopressin Receptor | GPCR/G Protein |
(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin (d(CH2)5[Tyr(Me)2, Dab5]AVP)作为针对加压素受体V1a的特异性拮抗剂,具有pA2值为6.71。 | |||
TP1654 |
H-Ala-Ala-Tyr-OH (TFA) (67131-52-6 free base)
H-Ala-Ala-Tyr-OH (TFA) |
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H-Ala-Ala-Tyr-OH TFA can be synthesized mutant peptides. | |||
TP2507 |
Leu-Tyr-Asp-Lys
|
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Leu-Tyr-Asp-Lys 是一种四肽化合物,可用于研究与代谢相关的疾病。 | |||
T41009 |
Fmoc-Tyr(tBu)-Ser(psi(Me,Me)pro)-OH
|
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Fmoc-Tyr(tBu)-Ser(psi(Me,Me)pro)-OH is a dipeptide. | |||
T20556 |
Tyrosyltyrosine
Tyr-tyr,Peptide tyrosine-tyrosine,Tyrosyl tyrosine |
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Tyrosyltyrosine is a dipeptide. | |||
T32529 |
Lactoferroxin-B
Arg-tyr-tyr-gly-tyr-och3,Lactoferroxin B |
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Lactoferroxin-B is a peptide that has an affinity for opioid receptors. | |||
T29595 |
Acetylalanyltyrosine
CH3CO-Ala-tyr,Acetyl-ala-tyr |
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Acetylalanyltyrosine is a peptide. | |||
TP2309 |
NEUROTENSIN TFA (39379-15-2 free base)
NEUROTENSIN TFA,神经加压素 |
Others | Others |
Neurotensin TFA (39379-15-2 free base) 是一种内源性 13 个氨基酸的神经肽,具有显着的阿片类非依赖性镇痛作用。它在大脑中充当神经递质,在肠道中充当激素,也充当神经调节剂。由于它与多种神经递质系统如多巴胺能、血清素能、谷氨酸能、GABA 能和胆碱能系统。它具有作为人体代谢物、有丝分裂原、神经递质和创伤的作用。 | |||
TP2362 |
Acetyl decapeptide-3
Rejuline,Ac-tyr-arg-ser-arg-lys-tyr-thr-ser-trp-tyr-NH2 |
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Acetyl decapeptide-3 is a peptide that can stimulate collagen and elastin to increase skin elasticity and increase cell growth and improve healing and repair. | |||
T25598 |
Lactoferroxin-A
Tyr-leu-gly-ser-gly-tyr-och3 |
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Lactoferroxin-A is used as an opioid antagonist. | |||
T25490 |
Hemorphin 4
Tyr-pro-trp-thr |
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Hemorphin 4 is an endogenous opioid peptide of the hemorphin family which has antinociceptive properties and is derived from the β-chain of hemoglobin in the bloodstream. | |||
TP2371 |
Asudemotide
Glu-tyr-tyr-glu-leu-phe-val-asn-ile |
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Asudemotide is a bioactive chemical. | |||
T29077 |
Urolinin
nWWK-Tyr(3-NO2)-Abu |
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Urolinin is a linear peptidic Urotensin-II Receptor Agonist with low nanomolar potency as well as improved metabolic stability. Urolinin is a hexameric UIIR agonist with an EC50 of 4.75 nM and a metabolic stability of 1319 min, 6.3-fold higher than wild-t | |||
T20496 |
TIPP
Tyr-Tic-Phe-Phe-OH |
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TIPP is an agent of delta opioid antagonist. | |||
T5092 |
AIM-100
AIM100 |
ACK | Tyrosine Kinase/Adaptors |
AIM-100 是选择性的 Ack1 抑制剂 (IC50:21.58 nM)。它还抑制 Tyr267磷酸化,但不抑制其他激酶,包括 PI3K 和 AKT 亚家族成员。它具有抗癌活性。 | |||
T31973 |
Glycyl-tyrosyl-alanine
Gly-tyr-ala |
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Glycyl-tyrosyl-alanine has a photooxidative effect. | |||
TP2478 |
WT-1 A1
Tyr-Met-Phe-Pro-agn-Ala-Pro-Tyr-Leu |
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WT-1 A1 is an attractive target for immunotherapy in patients with pancreatic adenocarcinoma. | |||
T40778 |
Tyrosylleucine TFA
Tyr-Leu TFA |
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Tyrosylleucine (Tyr-Leu, YL) TFA is a dipeptide compound with potent antidepressant-like activity. This orally active compound demonstrates effective modulation of depressive symptoms. | |||
T31634 |
[Des-Tyr1]-Met-Enkephalin
Met-enkephalin, des-tyr(1),1-De-tyr-met-enkephalin,Enkephalin-met, des-tyr(1)- |
||
Enkephalin-met, des-tyr(1)- ccauses retrograde amnesia in rats. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN6444 |
Cyclo(Tyr-Leu)
|
Antifungal | Microbiology/Virology |
Cyclo(Tyr-Leu) 是一种来自马齿苋 Portulaca oleracea Linn 的环状二肽,具有细胞毒性、抗真菌和抗凝血活性。 | |||
T5568 |
H-Tyr(3-I)-OH
3-碘-L-酪氨酸,3-Iodo-L-tyrosine |
Endogenous Metabolite | Metabolism |
H-Tyr(3-I)-OH (3-Iodo-L-tyrosine) 是酪氨酸羟化酶抑制剂和甲状腺激素 的中间体。 | |||
TN6678 |
Cyclo(Tyr-Pro)
|
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Cyclo(Tyr-Pro) shows antibacterial activity towards several marine bacterial species, it also shows weak antagonistic activity against VEGFR2 -CD. Cyclo(Tyr-Pro) and cyclo(Pro-Val) are toxic to both suspension cells and seedlings of Pinus thunbergii, whic | |||
TN6684 | Cyclo(Tyr-Hpro) | ||
Cyclo(Tyr-Hpro) 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6684,CAS号为 813461-21-1。 | |||
T5292 |
N-Acetyl-L-tyrosine
N-乙酰-L-酪氨酸,N-Acetyltyrosine,Ac-Tyr-OH |
Others; Endogenous Metabolite | Metabolism; Others |
N-Acetyl-L-tyrosine (Ac-Tyr-OH) 是一种来源于AA 乙酰酶作用下的酪氨酸,和芳香族氨基酸脱羧酶缺乏症以及酪氨酸血症有关,能够作为儿茶酚胺的前体,用于治疗神经递质。 | |||
TN6688 |
Cyclo(Ala-Tyr)
|
||
Cyclo(Val-Tyr) is a product from the culture of Pseudomonas putida. | |||
TN6689 |
Cyclo(Tyr-Phe)
|
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Cyclo-(Phe-Tyr) shows anticoagulant activities. | |||
TN6690 |
Cyclo(Tyr-Val)
|
||
Cyclo(Tyr-Val) 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6690,CAS号为 21754-25-6。 | |||
TN6687 |
Cyclo(Tyr-Gly)
|
||
Cyclo(Tyr-Gly) 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6687,CAS号为 5625-49-0。 | |||
T20555 |
Glycyltyrosine
NSC 118362,Gly Tyr,NSC-118362,Gly-Tyr,NSC118362,N-Glycyl-L-tyrosine |
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Glycyltyrosine, a dipeptide composed of tyrosine and glycine, is an incomplete breakdown product of protein catabolism or protein digestion. | |||
T4587 |
Mirificin
BCP10902,Puerarin Apioside,葛根素芹菜糖苷,芹糖葛根素苷 |
Tyrosinase | Proteases/Proteasome |
Mirificin (BCP10902) 是一种葛根中的异黄酮。它能够抑制酪氨酸酶(Tyrosinase),IC50=12.66 μM。 | |||
T66956 | H-Val-Tyr-OH | ||
H-Val-Tyr-OH 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 T66956,CAS号为 3061-91-4。 | |||
T3810 |
Saikosaponin B2
柴胡皂苷 B2,柴胡皂甙 B2 |
Others; HCV Protease | Microbiology/Virology; Others; Proteases/Proteasome |
Saikosaponin B2 是从柴胡根中分离得到的一种活性成分,可抑制 HCV 病毒感染的侵入,有抗癌作用。 | |||
T13762 |
Luteolin 7-sulfate
|
Others | Others |
Luteolin 7-sulfate, derived from the marine plant Phyllospadix iwatensis Makino, suppresses TYR gene expression by intervening in a signaling pathway involving the cAMP-responsive element binding protein (CREB) and microphthalmia-associated transcription factor (MITF). This inhibition ultimately leads to a decrease in melanin synthesis. |