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Cat. No. | Product Name | Target | Signaling Pathways |
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T24843 |
Syk-IN-1
SykIN11,Syk-IN-11,Syk IN 11,Syk inhibitor-11,Syk inhibitor 11,Syk-inhibitor-11 |
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Syk-IN-11 is a selective Syk inhibitor. | |||
T63086 |
SYK/JAK-IN-1
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SYK/JAK-IN-1 是一种 SYK/JAK 双重抑制剂,对 SYK 和 JAK2 的 IC50 值均小于 5 nM。 | |||
T9543 |
Syk Inhibitor II hydrochloride
|
Others | Others |
Syk Inhibitor II hydrochloride 信号传导的影响在狼疮中可能很突出。 | |||
T3211 |
Midostaurin
米哚妥林,N-Benzoylstaurosporine,PKC412,CGP41231,CGP 41251,苯甲酰基十字孢碱 |
Others; PKC | Chromatin/Epigenetic; Cytoskeletal Signaling; Others |
Midostaurin (PKC412) 是一种多靶点蛋白激酶抑制剂,有抗肿瘤活性,对 PKCα/β/γ、Syk、Flk-1、Akt、PKA、c-Kit、c-Fgr、c-Src、FLT3、PDFRβ和VEGFR1/2的IC50值范围为 22 到500 nM 之间。 | |||
T78943 |
Syk-IN-7
|
Syk | Angiogenesis; Tyrosine Kinase/Adaptors |
Syk-IN-7(化合物17)是一类特定的酪氨酸激酶(SYK)抑制剂。 | |||
T37077 |
Syk-IN-4
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Syk-IN-4 is a potent, selective, and orally bioavailable inhibitor of SYK, demonstrating an IC50 of 0.31 nM. It targets SYK, which has been identified as a potential therapeutic target for autoimmunity and hematological cancers[1]. | |||
T79443 |
Syk-IN-8
|
Syk | Angiogenesis; Tyrosine Kinase/Adaptors |
Syk-IN-8(compound 19q)是一款Syk抑制剂,有效抗血液肿瘤细胞增殖。该化合物能够阻断PLCγ2的磷酸化过程,常用于血癌的科学研究。 | |||
T61527 |
GSK2646264
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GSK2646264 (Compound 44) is a highly effective and specific inhibitor of spleen tyrosine kinase (SYK) with a pIC50 of 7.1. In addition to targeting SYK, GSK2646264 also inhibits several other kinases, including LCK, LRRK2, GSK3β, JAK2, VEGFR2, Aurora B, and Aurora A, with pIC50 values of 5.4, 5.4, 5.3, 5, 4.5, <4.6 and <4.3, respectively. Notably, GSK2646264 demonstrates skin penetrability, reaching both the epidermis and dermis [1]. |
Cat. No. | Product Name | Target | Signaling Pathways |
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T4S0498 |
Glaucocalyxin A
蓝萼甲素,Wangzaozin B,Leukamenin F |
Apoptosis; Akt; Caspase; PI3K | Apoptosis; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Proteases/Proteasome |
Glaucocalyxin A (Leukamenin F) 是来自日本黑纹病菌的一种对映型月桂基二萜,具有抗肿瘤作用。它通过调节PI3K/Akt 信号通路抑制 GLI1 的核易位,诱导骨肉瘤凋亡。 |