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Cat. No. Product Name Target Signaling Pathways
T23861 CAY10526

CAY-10526,BTH,CAY 10526

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
CAY10526 (BTH) 是 mPGES-1 的选择性抑制剂,可抑制 NF-κB 信号通路。
T16856 SB228357

5-HT Receptor GPCR/G Protein; Neuroscience
SB228357 是一种有效且的选择性 5-HT 受体拮抗剂,对 5-HT2A、5-HT2B 和 5-HT2C 的 pKis 分别为 6.9、8.0 和 9.0。
T1955 SB225002

CXCR Autophagy; GPCR/G Protein; Immunology/Inflammation
SB225002 是一种有效的选择性 CXCR2 拮抗剂,抑制白介素 IL-8 与 CXCR2 的结合,IC50为 22 nM。
T12851 SB290157 trifluoroacetate

Complement System Immunology/Inflammation
SB290157 trifluoroacetate 是一种选择性 C3a 受体拮抗剂,IC50值为200 nM。
T6657 SB273005

Integrin Cytoskeletal Signaling
SB273005 是一种有效的整合素抑制剂,对 αvβ3 受体和 αvβ5 受体的 Ki 分别为 1.2 nM 和 0.3 nM。
T4674 SB297006

SB 297006

CCR Immunology/Inflammation; Microbiology/Virology
SB297006 是一种CCR3拮抗剂,IC50为39 nM。它能够显著抑制 CCL11 处理的神经祖细胞的增殖和神经球形成。
T75013 SB26019

SB26019 是一种有效的抗神经炎症剂。SB26019 通过诱导单体 α-微管蛋白 (α-tubulin) 形成来调节 NF-κB 激活。SB26019 诱导的 α-微管蛋白单体抑制 p65 易位。
T28683 SB234551

SB 234551,SB-234551

SB234551 is a selective antagonist of endothelin ETA receptor.
T28688 SB2602

SB-2602,SB 2602

SB2602 selectively inhibits mTOR.
T16857 SB269652

Others Others
SB269652 is the first drug-like allosteric modulator of the dopamine D2 receptor.
T28685 SB236057

SB-236057,SB 236057

SB236057 is a potent and selective inverse agonist for the 5-HT receptor, acting especially at 5-HT autoreceptors on nerve terminals. It produces a rapid increase in 5-HT levels in the brain. SB236057 also acts as a potent teratogen, producing severe musc
T28687 SB251023

SB-251023,SB 251023

SB251023 is an agonist of β3-adrenoceptor.
T82961 ASB20123

ASB20123 是一款融合了CNP/ghrelin序列的嵌合肽,具有促进骨骼生长的效能,适用于研究生长障碍和侏儒症。
T28681 SB220025

SB-220025,SB 220025

SB220025, a specific and potent inhibitor of human p38 mitogen-activated protein kinase, reduces the production of tumor necrosis factor induced by lipopolysaccharide.

化合物

CAY10526
Cat.No: T23861
Synonym: CAY-10526,BTH,CAY 10526
Target: Prostaglandin Receptor
SB228357
Cat.No: T16856
Synonym:
Target: 5-HT Receptor
SB225002
Cat.No: T1955
Synonym:
Target: CXCR
SB290157 trifluoroacetate
Cat.No: T12851
Synonym:
Target: Complement System
SB273005
Cat.No: T6657
Synonym:
Target: Integrin
SB297006
Cat.No: T4674
Synonym: SB 297006
Target: CCR
SB26019
Cat.No: T75013
Synonym:
Target:
SB234551
Cat.No: T28683
Synonym: SB 234551,SB-234551
Target:
SB2602
Cat.No: T28688
Synonym: SB-2602,SB 2602
Target:
SB269652
Cat.No: T16857
Synonym:
Target: Others
SB236057
Cat.No: T28685
Synonym: SB-236057,SB 236057
Target:
SB251023
Cat.No: T28687
Synonym: SB-251023,SB 251023
Target:
ASB20123
Cat.No: T82961
Synonym:
Target:
SB220025
Cat.No: T28681
Synonym: SB-220025,SB 220025
Target:
TargetMol Loading
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