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Cat. No. Product Name Target Signaling Pathways
T29956 Amchem R 14

R14,Polyurethane Y-195,R-14

Others Others
Amchem R 14 is a biochemical.
T7667 R1487

p38 MAPK MAPK
R1487 是一种口服生物可利用的高选择性 p38α 丝裂原活化蛋白激酶抑制剂。
T79745 IDH2R140Q-IN-2

Dehydrogenase Metabolism
IDH2R140Q-IN-2 是一种具有口服活性和高效性的 IDH2R140Q 抑制剂,IC50为29 nM。IDH2R140Q-IN-2 具有潜在的抗肿瘤活性,能减少携带IDH2R140Q突变的TF-1细胞系中D2HG的生成(IC50为10 nM),抑制肿瘤组织中D2HG的水平。IDH2R140Q-IN-2适用于研究急性髓系白血病(AML)。
T15416 GR148672X

4,4,4-三氟-1-(2-噻吩基)-1,2,3-丁三酮 2-[(3-甲基苯基)腙]

Others Others
GR148672X 是三酰甘油水解酶抑制剂(IC50:4 nM)。
T9316 JR14a

5-(Bis(4-chlorophenyl)methyl)-3-methylthiophene-2-carbonyl)-l-arginine hydrochloride

Complement System Immunology/Inflammation
JR14a (5-(Bis(4-chlorophenyl)methyl)-3-methylthiophene-2-carbonyl)-l-arginine hydrochloride) 是补体C3a 受体噻吩拮抗剂,可抑制 C3aR 介导的炎症,对人 C3a 受体的选择性高于 C5a 受体。
T16928 SR144528

Cannabinoid Receptor GPCR/G Protein
SR144528 是 CB2 受体的拮抗剂 (Ki = 0.6 nM) 并抑制微粒体 ACAT 活性 (IC50 = 3.6 μM)。
TP1312L [SER140]-PLP(139-151) acetate

[SER140]-PLP(139-151) acetate (122018-58-0 Free base)

Others Others
[SER140]-PLP(139-151) acetate 是来自髓鞘蛋白脂蛋白 (PLP) 的肽片段。
T80897 UniPR1447

Ephrin Receptor Tyrosine Kinase/Adaptors
UniPR1447 是一种双重EphA2和EphB2拮抗剂,其对EphA2−ephrin-A1结合的IC50为6.6 μM。
T7162 R1487 Hydrochloride

R1487 (Hydrochloride)

p38 MAPK; Autophagy Autophagy; MAPK
R1487 Hydrochloride (R1487(Hydrochloride)) 是一种可口服的高选择性 p38α 抑制剂,对 p38α 和 p38β 的Kd 值分别为 0.2 nM 和 29 nM。
T28845 SR142948A HCl

SR142948A,SR 142948A,SR-142948A,SR142948A hydrochloride

Others Others
SR 142948A is a non-peptide antagonist of neurotensin receptor. SR 142948A affects the expression of c-Fos and has properties of antipsychotic agent. SR 142948A blocks hypothermia and analgesia induced by neurotensin. It blocks the increase in the concent
T81039 TAS2R14 agonist-2

Others Others
TAS2R14 agonist-2 (compound 28.1) 作为选择性TAS2R14抑制剂,其EC50为72 nM。
T24699 R1498

R-1498,R 1498

Others Others
R1498 is an inhibitor of cyclin-dependent kinase 2. It also acts by targeting angiogenesis and mitosis pathways. It is well-tolerated and orally active for hepatocellular carcinoma and gastric cancer treatment.
TP1312 [SER140]-PLP(139-151)

[SER140]-PLP(139-151) is a polypeptide fragment of the lipid protein of myelin.
T80896 UniPR1449

Ephrin Receptor Tyrosine Kinase/Adaptors
UniPR1449为EphA2受体拮抗剂,具有KD值约为3.8±2.4 μM,对癌症具有关键影响。
T69340 R140309

Others Others
R140309 is an UCHL3 inhibitor.
T81040 TAS2R14 agonist-1

Others Others
TAS2R14 agonist为一种TAS2R14受体的部分激活分子,其EC50值确定为116.6±23.6 nM。
T24828 SR14150

SR-14150,SR 14150

Others Others
SR14150 is a partial agonist of high-affinity NOP receptor.
TP1402 [SER140]-PLP(139-151) TFA (122018-58-0 free base)

[SER140]-PLP(139-151) TFA

[SER140]-PLP(139-151) (TFA) is a polypeptide fragment of the myelin lipid protein.
T63193 IDH2R140Q-IN-1

Others Others
IDH2R140Q-IN-1 是IDH2R140Q 有效的抑制剂(IC50: 6.1 nM),能够用于急性髓细胞白血病的研究。

化合物

Amchem R 14
Cat.No: T29956
Synonym: R14,Polyurethane Y-195,R-14
Target: Others
R1487
Cat.No: T7667
Synonym:
Target: p38 MAPK
IDH2R140Q-IN-2
Cat.No: T79745
Synonym:
Target: Dehydrogenase
GR148672X
Cat.No: T15416
Synonym: 4,4,4-三氟-1-(2-噻吩基)-1,2,3-丁三酮 2-[(3-甲基苯基)腙]
Target: Others
JR14a
Cat.No: T9316
Synonym: 5-(Bis(4-chlorophenyl)methyl)-3-methylthiophene-2-carbonyl)-l-arginine hydrochloride
Target: Complement System
SR144528
Cat.No: T16928
Synonym:
Target: Cannabinoid Receptor
[SER140]-PLP(139-151) acetate
Cat.No: TP1312L
Synonym: [SER140]-PLP(139-151) acetate (122018-58-0 Free base)
Target: Others
UniPR1447
Cat.No: T80897
Synonym:
Target: Ephrin Receptor
R1487 Hydrochloride
Cat.No: T7162
Synonym: R1487 (Hydrochloride)
Target: p38 MAPK, Autophagy
SR142948A HCl
Cat.No: T28845
Synonym: SR142948A,SR 142948A,SR-142948A,SR142948A hydrochloride
Target: Others
TAS2R14 agonist-2
Cat.No: T81039
Synonym:
Target: Others
R1498
Cat.No: T24699
Synonym: R-1498,R 1498
Target: Others
[SER140]-PLP(139-151)
Cat.No: TP1312
Synonym:
Target:
UniPR1449
Cat.No: T80896
Synonym:
Target: Ephrin Receptor
R140309
Cat.No: T69340
Synonym:
Target: Others
TAS2R14 agonist-1
Cat.No: T81040
Synonym:
Target: Others
SR14150
Cat.No: T24828
Synonym: SR-14150,SR 14150
Target: Others
[SER140]-PLP(139-151) TFA (122018-58-0 free base)
Cat.No: TP1402
Synonym: [SER140]-PLP(139-151) TFA
Target:
IDH2R140Q-IN-1
Cat.No: T63193
Synonym:
Target: Others
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