2
1
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T63115 |
Perphenazine dihydrochloride
|
Apoptosis; Dopamine Receptor; 5-HT Receptor; Histamine Receptor | Apoptosis; GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Perphenazine dihydrochloride 是一种具有口服活性和高效性的多巴胺受体和组胺-1 受体拮抗剂,抑制 D2、D3 和 5-HT2A。Perphenazine dihydrochloride 抑制癌细胞增殖,并诱导细胞凋亡,可用于研究精神分裂和宫内膜癌。 | |||
T1090 |
Perphenazine
Perphenazin,Etaperazine,Trilafon,奋乃静 |
CaMK; Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Perphenazine (Trilafon) 是吩噻嗪衍生物和多巴胺拮抗剂,具有止吐和抗精神病特性。它能够抑制5-HT2A 受体,α1A 肾上腺素能受体,多巴胺D2、D3、D2L 受体,以及组胺H1受体,对应的Ki 值分别为5.6、10、0.765、0.13、3.4 和 8 nM。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T12411 |
Perphenazine D8 Dihydrochloride
|
Others | Others |
Perphenazine D8 Dihydrochloride is the deuterium labeled Perphenazine, which is an antipsychotic drug. |