7
2
Cat. No. | Product Name | Target | Signaling Pathways |
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TP1956L |
PKC ζ pseudosubstrate acetate
PKC ζ pseudosubstrate acetate (799764-07-1 free base) |
PKC | Chromatin/Epigenetic; Cytoskeletal Signaling |
PKC ζ pseudosubstrate acetate 是蛋白激酶 C (PKC) ζ 的抑制剂;附着于细胞通透性触角足结构域载体肽。由 PKC ζ 假底物结构域的氨基酸 113-129 组成,通过二硫键连接到触角足结构域载体肽。 Antennapedia 肽在 4 或 37°C 时被完整细胞积极吸收,确保快速有效地吸收抑制肽。一旦进入细胞,二硫键在细胞质中被还原,导致抑制肽的释放。通过 PKC ζ 非依赖性途径诱导肥大细胞脱粒。 | |||
T35407 |
Ζ-Stat
|
PKC | Chromatin/Epigenetic; Cytoskeletal Signaling |
ζ-Stat 是非典型的、特异性的PKC-ζ抑制剂,IC50为 5 μM。ζ-Stat 能够减少黑色素瘤细胞系的增殖并诱导细胞凋亡,在体外显示除抗肿瘤活性。 | |||
TP1956 |
PKC ζ pseudosubstrate
|
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Inhibitor of protein kinase C (PKC) ζ; attached to cell permeabilisation Antennapedia domain vector peptide. Consists of amino acids 113 - 129 of PKC ζ pseudosubstrate domain linked by a disulphide bridge to the Antennapedia domain vector peptide. The Antennapedia peptide is actively taken up by intact cells, at 4 or 37°C, ensuring rapid and effective uptake of the inhibitor peptide. Once inside the cell, the disulphide bonds are subjected to reduction in the cytoplasm leading to release of the ... | |||
T81449 |
PKC-ε translocation inhibitor peptide
|
PKC | Chromatin/Epigenetic; Cytoskeletal Signaling |
PKC-ε translocation inhibitor peptide,作为一种特定的PKC-ε易位抑制剂,能够特异性地调控FcγR介导的调理珠内化速率,而对FcαR运输不产生影响。 | |||
T3689 |
Ruboxistaurin hydrochloride
Ruboxistaurin,LY333531 HCl,LY 333531 hydrochloride,芦布妥林 |
PKC | Chromatin/Epigenetic; Cytoskeletal Signaling |
Ruboxistaurin hydrochloride (LY 333531 hydrochloride) 是蛋白激酶 C(PKC) 的同工酶选择性抑制剂,竞争性且可逆地抑制 PKCβI 和 PKCβII,IC50 值分别为 4.7 和 5.9 nM。 | |||
T40395 |
ζ-Stat trisodium
NSC37044 trisodium,ζ-Stat trisodium |
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ζ-Stat trisodium (NSC37044 trisodium) is a potent and selective inhibitor of protein kinase C-ζ (PKC-ζ), exhibiting an IC50 of 5 μM. It effectively suppresses the proliferation of melanoma cell lines and promotes apoptosis. Moreover, ζ-Stat trisodium demonstrates notable antitumor activity in vitro. | |||
T75937 |
Pep2m, myristoylated TFA
|
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Pep2m, myristoylated TFA (Myr-Pep2m TFA)为具备细胞渗透性的肽。该化合物通过破坏PKMζ与其下游靶点NSF/GluR2的相互作用而发挥作用,其中PKMζ为具有自主活性的PKC同工酶。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5239 |
Cholesteryl sulfate sodium
Cholesterol 3-Sulfate Sodium Salt,胆固醇硫酸酯钠盐,Sodium Cholesteryl Sulfate |
Endogenous Metabolite; PKC | Chromatin/Epigenetic; Cytoskeletal Signaling; Metabolism |
Cholesteryl sulfate sodium (Sodium Cholesteryl Sulfate) 是内源性代谢产物的一种。 | |||
T16791 |
Rottlerin
Mallotoxin,NSC 56346,粗糠柴苦素,NSC 94525 |
CaMK; Apoptosis; Others; HIV Protease; PKA; PKC; Autophagy | Apoptosis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology; Neuroscience; Others; Proteases/Proteasome; Tyrosine Kinase/Adaptors |
Rottlerin (NSC-56346) 是一种从Mallotus Philippinensis 中得到的天然产物, 是 PKC 的特异性抑制剂,抑制HIV-1整合和狂犬病病毒感染。它通过活化 caspase 3 诱导细胞凋亡. |