首页 工具
登录
购物车

搜索结果

Search Results for " new compound 3 "

8

抑制剂 & 化合物

5

天然产物

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T50028 6-fluoro-3-(4-1,2,5,6-tetrahydropyridyl)indole

6-氟-3-(1,2,3,6-四氢吡啶-4-基)-1H-吲哚,6-fluoro-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole

Others Others
6-fluoro-3-(4-1,2,5,6-tetrahydropyridyl)indole (6-fluoro-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) 是一种吲哚衍生物,具有潜在抗癌活性,是开发新药的潜在先导化合物。
T3465L Vesnarinone HCl

Synonym 2,OPC-8212 HCl,Vesnarinone HCl(81840-15-5 Free base)

Potassium Channel; Calcium Channel; PDE Membrane transporter/Ion channel; Metabolism
Vesnarinone HCl (OPC-8212 HCl) 是一种具有口服活性的 phosphodiesterase 3 (PDE3) 抑制剂。Vesnarinone HCl 可对钙离子和钾离子进行调节, 增加钙通量,减少钾通量。Vesnarinone HCl 是一种新的正性肌力化合物,可增强心肌收缩力,可用于心力衰竭的研究。
T3295 1-Methyl-1H-pyrazol-3-amine

Others Others
1-Methyl-1H-pyrazol-3-amine 是一种吡唑类化合物。它已被用于合成各种化合物,如药物、染料和聚合物。它也是合成某些药物的重要中间体。它还被用于新药的开发,以及酶抑制剂和受体调节剂的研究。
T8826 3-AMINO-1,2,4-TRIAZINE

Others Others
3-AMINO-1,2,4-TRIAZINE 是一种芳香族生物活性化合物,已用于合成各种药物,包括抗真菌药物氟康唑、抗炎药物布洛芬和抗癌药物紫杉醇;也被用于设计新药,如抗艾滋病药物齐多夫定和抗疟疾药物青蒿素;以及用于合成各种其他化合物,如抗糖尿病药物二甲双胍和抗高血压药物赖诺普利。
T14296 Antitumor agent-3

Others Others
Antitumor agent-3 is a potent compound. It comprises a new imidazopyridine having excellent antitumor activity as an active ingredient.
T60925 TRβ agonist 3

TRβ agonist 3 (Compound 3) 是TRβ的有效激动剂,它是一种新的潜在 TRβ 选择性拟甲状腺素。在体外研究中,TRβ agonist 3 可减少 HepG2 中的脂质积累并促进脂肪分解。
T60282 Metallo-β-lactamase-IN-3

Metallo-β-lactamase-IN-3 (compound 35) 是一种有效的金属 -β- 内酰胺酶 (MBL) 抑制剂,具有恢复现有 β-内酰胺类抗生素活性的潜力并为新抗生素的发现提供正交策略。Metallo-β-lactamase-IN-3 对 VIM-1和 NDM-1的活性较高,其 IC50值分别为 0.6 和 1.0 μM。Metallo-β-lactamase-IN-3 对 IMP-7 无抑制作用。
T71230 VMY-1-103

VMY-1-103 is a potent CDK inhibitor, is also a novel dansylated analog of purvalanol B, was shown to inhibit cell cycle progression and proliferation in prostate and breast cancer cells more effectively than purvalanol B. VMY-1-103 , but not purvalanol B, significantly decreased the proportion of cells in S phase and increased the proportion of cells in G(2)/M. VMY-1-103 increased the sub G(1) fraction of apoptotic cells, induced PARP and caspase-3 cleavage and increased the levels of the Death ...

化合物

6-fluoro-3-(4-1,2,5,6-tetrahydropyridyl)indole
Cat.No: T50028
Synonym: 6-氟-3-(1,2,3,6-四氢吡啶-4-基)-1H-吲哚,6-fluoro-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole
Target: Others
Vesnarinone HCl
Cat.No: T3465L
Synonym: Synonym 2,OPC-8212 HCl,Vesnarinone HCl(81840-15-5 Free base)
Target: Potassium Channel, Calcium Channel, PDE
1-Methyl-1H-pyrazol-3-amine
Cat.No: T3295
Synonym:
Target: Others
3-AMINO-1,2,4-TRIAZINE
Cat.No: T8826
Synonym:
Target: Others
Antitumor agent-3
Cat.No: T14296
Synonym:
Target: Others
TRβ agonist 3
Cat.No: T60925
Synonym:
Target:
Metallo-β-lactamase-IN-3
Cat.No: T60282
Synonym:
Target:
VMY-1-103
Cat.No: T71230
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN6410 New compound 3

New compound 3 可用于生命科学领域的相关研究,其产品编号为 TN6410。
T5S1988 Isorhamnetin-3-O-glucoside

Isorhamnetin-3-O-beta-D-Glucoside,异鼠李素-3-O-葡萄糖苷

Others Others
Isorhamnetin-3-O-glucoside (Isorhamnetin-3-O-beta-D-Glucoside) 是一种天然化合物,广泛存在于蔬菜和水稻中,经消化后可在肠道菌群中代谢。
T4S21320 ISOGINKGETIN

异银杏素,4',4'''-Dimethylamentoflavone,异银杏双黄酮

MMP; Others Others; Proteases/Proteasome
ISOGINKGETIN (4',4'''-Dimethylamentoflavone) 是一种MMP9抑制剂,也是一种Pre-mRNA Splicing 抑制剂。
TN3218 7-(4-Hydroxyphenyl)-1-phenyl-4-hepten-3-one

Beta Amyloid; PI3K; mTOR Neuroscience; PI3K/Akt/mTOR signaling
7-(4-Hydroxyphenyl)-1-phenyl-4-hepten-3-one as a beneficial compound to ameliorate the deleterious effects of Aβ on dendrite integrity and cell survival, and may provide new insights on drug discovery of Alzheimer's disease (AD).
T37690 Phenylpyropene A

Phenylpyropene A is a fungal metabolite originally isolated from P. griseofulvum that has enzyme inhibitory and insecticidal activities.1,2,3 It inhibits acyl-coenzyme A:cholesterol acyltransferase (ACAT; IC50 = 0.8 μM).1 Phenylpyropene A inhibits diacylglycerol acyltransferase (DGAT) in rat liver microsomes (IC50 = 78.7 μM). It induces mortality in 100% of M. persicae when used at a concentration of 5 ppm.3 |1. Kwon, O.E., Rho, M.C., Song, H.Y., et al. Phenylpyropene A and B, new inhibitors of ...

天然产物

New compound 3
Cat.No: TN6410
Synonym:
Target:
Isorhamnetin-3-O-glucoside
Cat.No: T5S1988
Synonym: Isorhamnetin-3-O-beta-D-Glucoside,异鼠李素-3-O-葡萄糖苷
Target: Others
ISOGINKGETIN
Cat.No: T4S21320
Synonym: 异银杏素,4',4'''-Dimethylamentoflavone,异银杏双黄酮
Target: MMP, Others
7-(4-Hydroxyphenyl)-1-phenyl-4-hepten-3-one
Cat.No: TN3218
Synonym:
Target: Beta Amyloid, PI3K, mTOR
Phenylpyropene A
Cat.No: T37690
Synonym:
Target:
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼