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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TP1935L1 |
RAGE antagonist peptide acetate
|
Beta Amyloid | Neuroscience |
RAGE antagonist peptide acetate 是一种高级的糖基化终产物 (RAGE) 拮抗剂。 它具有抗肿瘤和抗炎活性。 它可防止 RAGE 与其几个重要的配体结合,包括 HMGB-1、S100P 和 S100A4。 | |||
T24167 |
Inflachromene
ICM |
Others | Others |
Inflachromene(ICM) 是一种 HMGB1 和 HMGB 表达抑制剂,具有抗炎活性。Inflachromene 通过抑制 HMGB1 易位来减轻小鼠癫痫模型的癫痫发作严重程度,通过 HMGB1/2 调节的 TLR4-NF-κB 通路抑制内膜增生,通过调节 Beclin 1 活性来抑制自噬。Inflachromene 可用于研究癫痫。 | |||
TP1935 |
RAGE antagonist peptide
|
||
Receptor for advanced glycation end products (RAGE) antagonist. Blocks S100P, S100A4 and HMGB-1 mediated RAGE activation in vitro and in vivo. Inhibits growth and metastasis of rat glioma tumors. Reduces cell growth and RAGE-mediated NF-κB activity in hum |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5S1632 |
Barlerin
8-O-乙酰山栀苷甲酯,8-O-Acetylshanzhiside methyl ester,ND01 |
VEGFR; TNF; NF-κB; Akt; Caspase | Angiogenesis; Apoptosis; Cytoskeletal Signaling; NF-κB; PI3K/Akt/mTOR signaling; Proteases/Proteasome; Tyrosine Kinase/Adaptors |
Barlerin (8-O-Acetylshanzhiside methyl ester) 是一种环孢菌素葡萄糖苷,从中国西藏民间药用植物中分离得到,能够抑制NF-κB 活性。 |