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Cat. No. Product Name Target Signaling Pathways
T0116 Balofloxacin

DNA gyrase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Balofloxacin 是一种具有口服活性的氟喹诺酮类抗生素,可通过干扰 DNA 促旋酶来抑制细菌 DNA 的合成,对革兰氏阴性,革兰氏阳性和厌氧菌具有广谱抗菌活性。它可研究呼吸道,肠道和泌尿道感染。
T3117 Marbofloxacin

马波沙星,Marbofloxacine,Zeniquin,Marbocyl

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Marbofloxacin (Zeniquin) 是一种具有口服活性的氟喹诺酮类广谱抗菌剂。它可研究革兰氏阳性和革兰氏阴性细菌以及支原体引起的感染。
T9066 Merafloxacin

CI 934

SARS-CoV Microbiology/Virology
Merafloxacin (CI 934) 是一种氟喹诺酮类抗菌药物,也被确定为 SARS-CoV-2 的 1 PRF 抑制剂。它对革兰氏阳性菌和革兰氏阴性菌具有体外活性。
T6349 Sitafloxacin Hydrate

西他沙星水合物,DU-6859a,DU6859a hydrate

Antibacterial; Antibiotic Microbiology/Virology
Sitafloxacin Hydrate (DU-6859a) 是一种口服有效的氟喹诺酮类抗生素,在体外可对抗广泛的革兰氏阳性和阴性细菌有活性。Sitafloxacin 可研究呼吸道感染和尿路感染。
T7865 Danofloxacin

达氟沙星,达诺沙星,Danofloxacino,Danofloxacin free base,Danofloxacine

Others; DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Danofloxacin (Danofloxacin free base) free base 是一种具有口服活性第三代氟喹诺酮抗菌剂,对大多数革兰氏阴性和革兰氏阳性细菌,支原体和衣原体物种具有广谱的活性,并通过抑制细菌的 DNA 回转酶发挥抗菌作用。它可用于牛,猪和鸡呼吸道疾病的研究。
T6406 Besifloxacin Hydrochloride

BOL-303224-A,Besivance hydrochloride,Besifloxacin HCl,盐酸贝西沙星

Antibacterial; Antibiotic Microbiology/Virology
Besifloxacin Hydrochloride (BOL-303224-A) 是一种氟喹诺酮类抗生素。
T1620 Pazufloxacin Mesylate

Pazucross,Pazufloxacin mesilate,甲磺酸帕珠沙星,T-3762,帕珠沙星甲磺酸盐,Pazufloxacin methanesulfonate

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Pazufloxacin Mesylate (T-3762) 是一种喹诺酮类抗生素。
T1444 Lomefloxacin

洛美沙星,SC47111A

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Lomefloxacin (SC47111A) 是一种广谱喹诺酮类抗生素,具有抗菌活性。它可研究支气管炎、尿路感染、结膜炎、外耳炎和中耳炎。
T8173 Delafloxacin meglumine

ABT492 meglumine,德拉沙星葡甲胺,WQ-3034 meglumine,RX-3341 meglumine

Antibacterial; Antibiotic Microbiology/Virology
Delafloxacin meglumine (RX-3341 meglumine) 是一种广谱氟喹诺酮类抗生素。Delafloxacin 对耐药性的金黄色葡萄球菌,肺炎克雷伯菌和肺炎链球菌有活性。
T1294 Fleroxacin

AM-833,氟罗沙星,RO 23-6240

DNA gyrase; Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Fleroxacin (RO 23-6240) 是一种广谱氟喹诺酮类抗菌素。
TQ0221 Rufloxacin hydrochloride

MF-934 hydrochloride,盐酸芦氟沙星

Antibacterial Microbiology/Virology
Rufloxacin hydrochloride (MF-934 hydrochloride) 是一种氟喹诺酮类抗菌剂,可抑制拓扑异构酶。 Rufloxacin hydrochloride 抑制人单核细胞中的 B 细胞分化。
T0292 Orbifloxacin

CP-104354,奥比沙星

Antibacterial; Antibiotic Microbiology/Virology
Orbifloxacin (CP-104354) 是一种可用于犬类的氟喹诺酮类合成广谱抗生素。
T1095 Sparfloxacin

AT-4140,PD 131501,Zagam,司帕沙星,CI-978

DNA gyrase; Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Sparfloxacin (CI-978) 是一种氟喹诺酮类抗菌素。
T1640 Ciprofloxacin

Ciproxan,环丙沙星,Ciprobay,Bay o 9867,Bay-09867

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Ciprofloxacin (Bay-09867) 是一种有高抗菌活性的氟喹诺酮类抗生素。
T1293 Gatifloxacin

BMS 206584-01,PD 135432,CG5501,BMS-206584,AM-1155,加替沙星

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Gatifloxacin (CG5501) 是一种具有广谱抗菌活性的氟喹诺酮类抗生素。它可抑制大肠杆菌 DNA 解旋酶 (IC50=0.109 μg/ml) 和细菌 II 型拓扑异构酶(IC50=13.8 μg/ml)。在动物模型中,它有抗细菌性结膜炎作用。
T1492 Gemifloxacin mesylate

LB-20304a,甲磺酸吉米沙星,SB-265805S,Gemifloxacin mesylate

DNA gyrase; Topoisomerase; Antibacterial DNA Damage/DNA Repair; Microbiology/Virology
Gemifloxacin mesylate (Gemifloxacin mesylate) 是一种喹诺酮类口服广谱抗菌剂,可研究轻中度肺炎和慢性支气管炎的急性细菌性发作。
T0425 Pefloxacin Mesylate

Pefloxacinium mesylate,甲磺酸培氟沙星

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Pefloxacin Mesylate (Pefloxacinium mesylate) 是一种抗菌化合物,可抑制DNA 旋转酶阻断DNA 复制。
T13231L Trovafloxacin mesylate

Others; DNA/RNA Synthesis; Topoisomerase; Antibacterial Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Trovafloxacin是一种广谱氟喹诺酮类抗生素,可阻断 DNA 促旋酶 (DNA gyrase) 和拓扑异构酶 IV (topoisomerase IV) 的活性,也是一种有效的特异性 pannexin 1 通道抑制剂 (PANX1, IC50 = 4 μM)。
T8142 Difloxacin hydrochloride

Difloxacin HCl,盐酸二氟沙星

Antibacterial; Antibiotic Microbiology/Virology
Difloxacin hydrochloride (Difloxacin HCl) 是一种广谱抗菌药物。它干扰 DNA 促旋酶和拓扑异构酶 IV 的活性,抑制细菌 DNA 促旋酶并显示出浓度依赖性的杀菌作用。
T12649 Ibafloxacine

S25930,Ibafloxacin,R835

Antifungal Microbiology/Virology
Ibafloxacine (R835) 是一种氟喹诺酮类抗生素,专门用于兽类,对巴氏杆菌显示出良好的抑菌效果。
T4063 Delafloxacin

ABT492,WQ-3034,德拉沙星,RX-3341

Antibacterial; Antibiotic Microbiology/Virology
Delafloxacin (WQ-3034) 是一种广谱氟喹诺酮类抗生素,抑制耐药性的金黄色葡萄球菌,肺炎链球菌和肺炎克雷伯菌。
T8835 Tosufloxacin hydrochloride

A-61827 hydrochloride,盐酸妥舒沙星,T-3262 hydrochloride

Antibacterial Microbiology/Virology
Tosufloxacin hydrochloride 是一种氟喹诺酮类抗菌剂,用于治疗细菌感染。 Tosufloxacin hydrochloride 也是一种细菌 Topo(DNA 促旋酶,拓扑异构酶)抑制剂。
T13346L WQ3810 TFA

WQ3810 TFA(888032-58-4 Free base),KPI-10 TFA

Antifungal Microbiology/Virology
WQ3810 TFA 是一种可口服的氟喹诺酮,具有抗菌活性,对结核分枝杆菌有抑制作用,抑制氧氟沙星耐药麻风分枝杆菌的 DNA 旋转酶活性。
T1283 Clinafloxacin

克林沙星,PD 127391,CI-960,AM-1091

Antibacterial; Antibiotic Microbiology/Virology
Clinafloxacin (CI-960) 是一种高效广谱氟喹诺酮类抗生素,抑制革兰氏阳性、革兰氏阴性和厌氧病原体。它对金黄色葡萄球菌的 DNA 促旋酶和拓扑异构酶 IV 有抑制作用,IC50值分别为 0.92 µg/ml 和 1.62 µg/ml。
T0902 Ofloxacin

DL8280,菲宁达,Hoe-280,氧氟沙星,Floxin,Tarivid,Oxaldin

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Ofloxacin (Oxaldin) 是可抑制细菌DNA 旋转酶的一种氟喹诺酮类抗生素。
T5394 Prulifloxacin

AF 3012,Pruvel,NM441,普卢利沙星

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Prulifloxacin (NM441) 是一种口服有效的氟喹诺酮抗生素 ,对革兰氏阳性和阴性细菌具有广泛活性。它是噻唑喹啉羧酸衍生物 Ulifloxacin 的前药。它有潜力用于下尿路感染和慢性支气管炎。
T0331L Moxifloxacin

Avelox,Moxeza,莫西沙星

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Moxifloxacin (Avelox) 是一种8-甲氧基喹诺酮类口服有效抗菌药物,用于急性细菌性鼻窦炎,慢性支气管炎的急性细菌性加重和感染性肺炎的研究。
T1625 Lomefloxacin hydrochloride

Lomefloxacin HCl,盐酸洛美沙星,Okacyn,Maxaquin

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Lomefloxacin hydrochloride (Okacyn) 是一种广谱喹诺酮类抗生素,具有抗菌活性。它可研究支气管炎、尿路感染、结膜炎、外耳炎和中耳炎。
T1451 Levofloxacin hydrate

左氧氟沙星半水合物,Levaquin hydrate,Cravit hydrate,Quixin hydrate,Levofloxacin Hemihydrate,Tavanic hydrate,Iquix hydrate

DNA gyrase; Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Levofloxacin hydrate (Cravit hydrate) 是抗生素化合物,抑制细菌DNA 旋转酶活性。
T0331 Moxifloxacin hydrochloride

盐酸莫西沙星,莫西沙星盐酸盐,BAY-128039,Moxifloxacin HCl,BAY12-8039 HCl

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Moxifloxacin hydrochloride (BAY12-8039 HCl) 是一种口服有效的 8-甲氧基喹诺酮类抗菌药物,可研究感染性肺炎,急性细菌性鼻窦炎和慢性支气管炎的急性细菌性加重。
T8747 Levofloxacin hydrochloride

DNA gyrase; Topoisomerase DNA Damage/DNA Repair
Levofloxacin hydrochloride 是一种广谱的第三代氟喹诺酮类抗生素,是氧氟沙星的光学活性 L-异构体,具有抗菌活性。左氧氟沙星通过细菌细胞壁扩散并通过抑制 DNA 促旋酶(细菌拓扑异构酶 II)起作用,这是一种 DNA 复制、RNA 转录和细菌 DNA 修复所需的酶。 DNA 促旋酶活性的抑制导致细菌细胞生长受阻。
T16703 Quarfloxin

CX-3543

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Quarfloxin (CX-3543) 是一种氟喹诺酮衍生物,具有抗肿瘤活性,可靶向抑制RNA pol I 的活性,在神经母细胞瘤细胞中的 IC50 值在纳摩尔范围内。它破坏核糖体 DNA 模板中核仁蛋白和 G-四链体 DNA 结构之间的相互作用。
T13346 WQ3810

KPI-10 free base

Others Others
WQ3810 is an orally active fluoroquinolone, has potent antibacterial activities.
T22265 Balofloxacin Dihydrate

Neuroquinoron,巴洛沙星/1-环丙基-7-(3-甲氨基-1-哌啶基)-8-甲氧基-6-氟-1,4-二氢-4-氧代-3-喹啉羧酸

Others Others
Balofloxacin is a fluoroquinolone antibiotic with oral activity.
T27818 Levonadifloxacin Arginine Salt

WCK 771,WCK-771A,WCK 771A,WCK-771,WCK771A,WCK771

Levonadifloxacin, a broad-spectrum fluoroquinolone antibiotic, is used potentially for the treatment of staphylococci.
T26449 A 80556

A-80556,A80556

A 80556, a fluoroquinolone antibiotic, has potent antibacterial activity against gram-positive, gram-negative, and anaerobic organisms.
T30684 Cadrofloxacin

CS-940,CS 940,Cadrofloxacin hydrochloride,Caderofloxacin,CS940

Cadrofloxacin (Caderofloxacin, CS-940) is a novel fluoroquinolone antimicrobial agent.
T33899 PD 131628

PD131628,PD-131628

PD 131628 is a novel fluoroquinolone that is a bioactive form of PD 131112 or CI-990 for use against anaerobic bacteria.
T25461 Grepafloxacin, (S)-

L-Grepafloxacin

Grepafloxacin, (S)- is an oral broad-spectrum fluoroquinolone antibacterial used for the treatment of bacterial infections.
T23622 Acorafloxacin HCl

JNJ-32729463,JNJ-Q2 hydrochloride,Acorafloxacin hydrochloride,JNJ 32729463,JNJ-Q2 HCl

Acorafloxacin is a broad-spectrum fluoroquinolone antibacterial drug being developed for the treatment of acute bacterial skin and skin structure infections and community-acquired pneumonia.
T10420 Avarofloxacin

JNJ-Q2

Others Others
Avarofloxacin (JNJ-Q2) is a broad-spectrum fluoroquinolone antibacterial drug being developed for the treatment of acute bacterial skin and community-acquired pneumonia and skin structure infections.
T81412 Pradofloxacin

Pradofloxacin是一种第三代的氟喹诺酮类抗菌化合物。
T1466L Difloxacin HCl

Difloxacin 是第二代合成的氟喹诺酮抗菌抗生素。
T36031 Desmethyl Ofloxacin (hydrochloride)

Desmethyl ofloxacin is a metabolite of the fluoroquinolone antibiotic ofloxacin .1 1.Sudo, K., Okazaki, O., Tsumura, M., et al.Isolation and identification of metabolites of ofloxacin in rats, dogs and monkeysXenobiotica16(8)725-732(1986)
T71982 Ofloxacin HCl

Ofloxacin HCl is a synthetic fluoroquinolone ( FLUOROQUINOLONES) antibacterial agent that inhibits the supercoiling activity of bacterial DNA GYRASE, halting DNA REPLICATION.
T38586 Grepafloxacin

dl-Grepafloxacin,OPC-17116

Grepafloxacin (OPC-17116) is a fluoroquinolone antibiotic that is administered orally. It possesses strong efficacy against community-acquired respiratory pathogens, notably Streptococcus pneumonia. Grepafloxacin exhibits excellent tissue penetration and demonstrates a promising pharmacodynamic profile.
T26368 Tosufloxacin tosylate

Tosufloxacin,T-3262,T3262,T 3262

Tosufloxacin is a fluoroquinolone antibiotic used to treat susceptible infections.
T31031 CP 74667

UNII-D66A707X1B,CP74667,CP-74667

CP 74667 is a new fluoroquinolone that has good activity against several gram-positive and gram-negative pathogens.
T3522 Tosufloxacin tosilate

Others Others
Tosufloxacin tosilate 是一种氟喹诺酮类抗生素。
T22797 Gatifloxacin mesylate

Others Others
Gatifloxacin (mesylate) is an antibiotic of the fourth-generation fluoroquinolone family. It also inhibits the bacterial enzymes DNA gyrase and topoisomerase IV.

化合物

Balofloxacin
Cat.No: T0116
Synonym:
Target: DNA gyrase, Antibacterial, Antibiotic
Marbofloxacin
Cat.No: T3117
Synonym: 马波沙星,Marbofloxacine,Zeniquin,Marbocyl
Target: Topoisomerase, Antibacterial, Antibiotic
Merafloxacin
Cat.No: T9066
Synonym: CI 934
Target: SARS-CoV
Sitafloxacin Hydrate
Cat.No: T6349
Synonym: 西他沙星水合物,DU-6859a,DU6859a hydrate
Target: Antibacterial, Antibiotic
Danofloxacin
Cat.No: T7865
Synonym: 达氟沙星,达诺沙星,Danofloxacino,Danofloxacin free base,Danofloxacine
Target: Others, DNA/RNA Synthesis, Antibacterial, Antibiotic
Besifloxacin Hydrochloride
Cat.No: T6406
Synonym: BOL-303224-A,Besivance hydrochloride,Besifloxacin HCl,盐酸贝西沙星
Target: Antibacterial, Antibiotic
Pazufloxacin Mesylate
Cat.No: T1620
Synonym: Pazucross,Pazufloxacin mesilate,甲磺酸帕珠沙星,T-3762,帕珠沙星甲磺酸盐,Pazufloxacin methanesulfonate
Target: Topoisomerase, Antibacterial, Antibiotic
Lomefloxacin
Cat.No: T1444
Synonym: 洛美沙星,SC47111A
Target: Topoisomerase, Antibacterial, Antibiotic
Delafloxacin meglumine
Cat.No: T8173
Synonym: ABT492 meglumine,德拉沙星葡甲胺,WQ-3034 meglumine,RX-3341 meglumine
Target: Antibacterial, Antibiotic
Fleroxacin
Cat.No: T1294
Synonym: AM-833,氟罗沙星,RO 23-6240
Target: DNA gyrase, Topoisomerase, Antibacterial, Antibiotic
Rufloxacin hydrochloride
Cat.No: TQ0221
Synonym: MF-934 hydrochloride,盐酸芦氟沙星
Target: Antibacterial
Orbifloxacin
Cat.No: T0292
Synonym: CP-104354,奥比沙星
Target: Antibacterial, Antibiotic
Sparfloxacin
Cat.No: T1095
Synonym: AT-4140,PD 131501,Zagam,司帕沙星,CI-978
Target: DNA gyrase, Topoisomerase, Antibacterial, Antibiotic
Ciprofloxacin
Cat.No: T1640
Synonym: Ciproxan,环丙沙星,Ciprobay,Bay o 9867,Bay-09867
Target: Topoisomerase, Antibacterial, Antibiotic
Gatifloxacin
Cat.No: T1293
Synonym: BMS 206584-01,PD 135432,CG5501,BMS-206584,AM-1155,加替沙星
Target: Topoisomerase, Antibacterial, Antibiotic
Gemifloxacin mesylate
Cat.No: T1492
Synonym: LB-20304a,甲磺酸吉米沙星,SB-265805S,Gemifloxacin mesylate
Target: DNA gyrase, Topoisomerase, Antibacterial
Pefloxacin Mesylate
Cat.No: T0425
Synonym: Pefloxacinium mesylate,甲磺酸培氟沙星
Target: Topoisomerase, Antibacterial, Antibiotic
Trovafloxacin mesylate
Cat.No: T13231L
Synonym:
Target: Others, DNA/RNA Synthesis, Topoisomerase, Antibacterial
Difloxacin hydrochloride
Cat.No: T8142
Synonym: Difloxacin HCl,盐酸二氟沙星
Target: Antibacterial, Antibiotic
Ibafloxacine
Cat.No: T12649
Synonym: S25930,Ibafloxacin,R835
Target: Antifungal
Delafloxacin
Cat.No: T4063
Synonym: ABT492,WQ-3034,德拉沙星,RX-3341
Target: Antibacterial, Antibiotic
Tosufloxacin hydrochloride
Cat.No: T8835
Synonym: A-61827 hydrochloride,盐酸妥舒沙星,T-3262 hydrochloride
Target: Antibacterial
WQ3810 TFA
Cat.No: T13346L
Synonym: WQ3810 TFA(888032-58-4 Free base),KPI-10 TFA
Target: Antifungal
Clinafloxacin
Cat.No: T1283
Synonym: 克林沙星,PD 127391,CI-960,AM-1091
Target: Antibacterial, Antibiotic
Ofloxacin
Cat.No: T0902
Synonym: DL8280,菲宁达,Hoe-280,氧氟沙星,Floxin,Tarivid,Oxaldin
Target: Topoisomerase, Antibacterial, Antibiotic
Prulifloxacin
Cat.No: T5394
Synonym: AF 3012,Pruvel,NM441,普卢利沙星
Target: Topoisomerase, Antibacterial, Antibiotic
Moxifloxacin
Cat.No: T0331L
Synonym: Avelox,Moxeza,莫西沙星
Target: Others, Antibacterial, Antibiotic
Lomefloxacin hydrochloride
Cat.No: T1625
Synonym: Lomefloxacin HCl,盐酸洛美沙星,Okacyn,Maxaquin
Target: Topoisomerase, Antibacterial, Antibiotic
Levofloxacin hydrate
Cat.No: T1451
Synonym: 左氧氟沙星半水合物,Levaquin hydrate,Cravit hydrate,Quixin hydrate,Levofloxacin Hemihydrate,Tavanic hydrate,Iquix hydrate
Target: DNA gyrase, Topoisomerase, Antibacterial, Antibiotic
Moxifloxacin hydrochloride
Cat.No: T0331
Synonym: 盐酸莫西沙星,莫西沙星盐酸盐,BAY-128039,Moxifloxacin HCl,BAY12-8039 HCl
Target: Topoisomerase, Antibacterial, Antibiotic
Levofloxacin hydrochloride
Cat.No: T8747
Synonym:
Target: DNA gyrase, Topoisomerase
Quarfloxin
Cat.No: T16703
Synonym: CX-3543
Target: DNA/RNA Synthesis
WQ3810
Cat.No: T13346
Synonym: KPI-10 free base
Target: Others
Balofloxacin Dihydrate
Cat.No: T22265
Synonym: Neuroquinoron,巴洛沙星/1-环丙基-7-(3-甲氨基-1-哌啶基)-8-甲氧基-6-氟-1,4-二氢-4-氧代-3-喹啉羧酸
Target: Others
Levonadifloxacin Arginine Salt
Cat.No: T27818
Synonym: WCK 771,WCK-771A,WCK 771A,WCK-771,WCK771A,WCK771
Target:
A 80556
Cat.No: T26449
Synonym: A-80556,A80556
Target:
Cadrofloxacin
Cat.No: T30684
Synonym: CS-940,CS 940,Cadrofloxacin hydrochloride,Caderofloxacin,CS940
Target:
PD 131628
Cat.No: T33899
Synonym: PD131628,PD-131628
Target:
Grepafloxacin, (S)-
Cat.No: T25461
Synonym: L-Grepafloxacin
Target:
Acorafloxacin HCl
Cat.No: T23622
Synonym: JNJ-32729463,JNJ-Q2 hydrochloride,Acorafloxacin hydrochloride,JNJ 32729463,JNJ-Q2 HCl
Target:
Avarofloxacin
Cat.No: T10420
Synonym: JNJ-Q2
Target: Others
Pradofloxacin
Cat.No: T81412
Synonym:
Target:
Difloxacin HCl
Cat.No: T1466L
Synonym:
Target:
Desmethyl Ofloxacin (hydrochloride)
Cat.No: T36031
Synonym:
Target:
Ofloxacin HCl
Cat.No: T71982
Synonym:
Target:
Grepafloxacin
Cat.No: T38586
Synonym: dl-Grepafloxacin,OPC-17116
Target:
Tosufloxacin tosylate
Cat.No: T26368
Synonym: Tosufloxacin,T-3262,T3262,T 3262
Target:
CP 74667
Cat.No: T31031
Synonym: UNII-D66A707X1B,CP74667,CP-74667
Target:
Tosufloxacin tosilate
Cat.No: T3522
Synonym:
Target: Others
Gatifloxacin mesylate
Cat.No: T22797
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T6567 Levofloxacin

Levaquin,Cravit,Tavanic,Fluoroquinolone,左氧氟沙星,(-)-Ofloxacin

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Levofloxacin (Fluoroquinolone) 是合成的氟喹诺酮类抗生素,有抑制细菌DNA 旋转酶的超螺旋活性的作用,能阻止DNA 复制。
T8046 Tosufloxacin tosylate hydrate

Tosufloxacin p-Toluenesulfonate Hydrate,A-61827 tosylate hydrate,对甲苯磺酸妥舒沙星水合物,T-3262 Tosylate Hydrate

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Tosufloxacin tosylate hydrate (A-61827 tosylate hydrate) 是一个氟喹诺酮类抗菌剂。
T8130 Ciprofloxacin hydrochloride monohydrate

Oftacilox,Ciprofloxacin hydrochloride hydrate,Bay-09867 hydrochloride monohydrate,环丙沙星盐酸盐一水合物,Ceprimax,盐酸环丙沙星(一水物),Ciloxan

Antibacterial; Antibiotic Microbiology/Virology
Ciprofloxacin hydrochloride monohydrate (Bay-09867 hydrochloride monohydrate) 是一种具有高效抗菌活性的氟喹诺酮类抗生素。
T1276 Danofloxacin mesylate

甲磺酸达氟沙星,CP 76136-27

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Danofloxacin mesylate (CP 76136-27) 是一种兽医用氟喹诺酮类抗菌素。
T8384 Gatifloxacin hydrochloride

AM-1155 (hydrochloride),BMS-206584 (hydrochloride),PD135432 (hydrochloride),加替沙星盐酸盐

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Gatifloxacin hydrochloride (AM-1155 hydrochloride) 是一种氟喹诺酮类抗生素,有广谱抗菌活性。它可抑制大肠杆菌 DNA 解旋酶 (IC50=0.109 μg/ml)和细菌 II 型拓扑异构酶(IC50=13.8 μg/ml) 。它在动物模型中,可研究细菌性结膜炎。

天然产物

Levofloxacin
Cat.No: T6567
Synonym: Levaquin,Cravit,Tavanic,Fluoroquinolone,左氧氟沙星,(-)-Ofloxacin
Target: Topoisomerase, Antibacterial, Antibiotic
Tosufloxacin tosylate hydrate
Cat.No: T8046
Synonym: Tosufloxacin p-Toluenesulfonate Hydrate,A-61827 tosylate hydrate,对甲苯磺酸妥舒沙星水合物,T-3262 Tosylate Hydrate
Target: Others, Antibacterial, Antibiotic
Ciprofloxacin hydrochloride monohydrate
Cat.No: T8130
Synonym: Oftacilox,Ciprofloxacin hydrochloride hydrate,Bay-09867 hydrochloride monohydrate,环丙沙星盐酸盐一水合物,Ceprimax,盐酸环丙沙星(一水物),Ciloxan
Target: Antibacterial, Antibiotic
Danofloxacin mesylate
Cat.No: T1276
Synonym: 甲磺酸达氟沙星,CP 76136-27
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Gatifloxacin hydrochloride
Cat.No: T8384
Synonym: AM-1155 (hydrochloride),BMS-206584 (hydrochloride),PD135432 (hydrochloride),加替沙星盐酸盐
Target: Topoisomerase, Antibacterial, Antibiotic
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