10
4
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T19654 |
Guanoclor
胍氯酚,VATENSOL |
Others | Others |
Guanoclor (VATENSOL) 也称为guanochlor,是一种交感神经药物。已知它与猪肾膜中的非肾上腺素能位点结合。 | |||
T13383 |
Zamicastat
BIA 5-1058 |
BCRP; Hydroxylase; P-gp | Membrane transporter/Ion channel; Metabolism; Neuroscience |
Zamicastat (BIA 5-1058) 是多巴胺 β-羟化酶 (DBH) 抑制剂,可透过血脑屏障引起中枢和周边效应,具有降血压作用。它也是一种浓度依赖性的双重 P-gp 和 BCRP 抑制剂,IC50值分别为 73.8 和 17.0 μM。 | |||
T6604 |
Nepicastat hydrochloride
Nepicastat HCl,内匹司他盐酸盐,RS-25560-197 hydrochloride,SYN-117 hydrochloride,Nepicastat (SYN-117) HCl |
Hydroxylase | Metabolism |
Nepicastat hydrochloride (RS-25560-197 hydrochloride) 是一种选择性的,有效的,口服活性的多巴胺 β 羟化酶(dopamine-beta-hydroxylase)抑制剂,对牛和人多巴胺 β 羟化酶的IC50分别为IC50=8.5 nM 和IC50=9 nM。Nepicastat HCl 可以穿过血脑屏障。 | |||
T11238L |
Etamicastat hydrochloride
BIA 5-453 hydrochloride |
Dehydrogenase | Metabolism |
Etamicastat hydrochloride (BIA 5-453 hydrochloride) 是一种外周选择性多巴胺β-羟化酶抑制剂,具有降低高血压的作用。 | |||
T50049 |
4-Methylhistamine hydrochloride
|
Others | Others |
4-Methylhistamine hydrochloride 已被证明能抑制铜依赖性酶如酪氨酸酶和多巴胺β-羟化酶的活性,还被证明可以调节参与细胞周期调节和凋亡的基因的表达。 | |||
T71936 | Phenylthiazolylthiourea | ||
Phenylthiazolylthiourea ia a dopamine-beta-hydroxylase inhibitor. | |||
T69568 |
FLA-63
|
||
FLA-63 is a dopamine-beta-hydroxylase (DBH)-inhibitor and an inhibitor of the last step of noradrenaline biosynthesis. | |||
T23848 |
Calcium Fusarate
|
||
Calcium Fumarate is an inhibitor of dopamine beta-hydroxylase. It also inhibited cell proliferation and DNA synthesis. | |||
T70209 |
Nepicastat hydrochloride monohydrate
|
||
Nepicastat hydrochloride monohydrate is an inhibitor of dopamine beta-hydroxylase, an enzyme that catalyzes the conversion of dopamine to norepinephrine. | |||
T60633 | Nepicastat | ||
Nepicastat (SYN117) 是一种选择性的,有效的,口服的多巴胺 β 羟化酶抑制剂,可穿过血脑屏障(BBB)。Nepicastat (SYN117) 对牛和人多巴胺 β 羟化酶产生浓度依赖性抑制作用,IC50值分别为8.5 nM 和 9 nM。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6S0923 |
Hypericin
Hypericine,金丝桃素,Cyclosan |
Apoptosis; Antiviral; Influenza Virus; Tyrosine Kinases; Antibacterial; PKC | Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Immunology/Inflammation; Microbiology/Virology; Tyrosine Kinase/Adaptors |
Hypericin (Cyclosan) 是贯叶连翘的提取物,有抗菌、抗病毒、抗肿瘤和抗抑郁作用。 | |||
T2S1778 |
DL-Goitrin
DL-甲状腺肿素,板蓝根,Goitrin,(R,S)-告依春 |
Others | Others |
DL-Goitrin 也称为 (R,S)-Goitrin,由 epigoitrin (R-Goitrin) 和告依春 (S-Goitrin) 两种异构体组成,是板蓝根的成分。 | |||
TN2252 |
Syrosingopine
|
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Syrosingopine 是 MCT1和 MCT4双重抑制剂,对 MCT4 的效力高 60 倍,可防止乳酸和 H+ 流出。它是可口服抗高血压药物,联合二甲双胍具有研究癌症疾病的潜力。 | |||
T25900 |
Oosponol
Lenzitin |
||
Oosponol is a dopamine beta-hydroxylase inhibitor exhibiting hypotensive effects. |