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Cat. No. | Product Name | Target | Signaling Pathways |
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T0270 |
Hydrocortisone 17-butyrate
丁酸氢化可的松,Cortisol 17-butyrate,Hydrocortisone butyrate |
Glucocorticoid Receptor; Annexin A; Adrenergic Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Hydrocortisone 17-butyrate (Cortisol 17-butyrate) 是一种肾上腺皮质激素类药物。 | |||
T1666 |
Fludrocortisone acetate
9α-Fluorcortisol acetate,9α-Fludrocortisone acetate,醋酸氟氢可的松,9α-fluorocortisol acetate |
Glucocorticoid Receptor; Autophagy | Autophagy; Endocrinology/Hormones |
Fludrocortisone acetate (9α-Fludrocortisone acetate) 是一种合成的盐皮质激素,可减少尿液中钠丢失量,也用于增加血压,有用于阿狄森氏病的研究潜力。 | |||
T1666L |
Fludrocortisone
9α-fluorocortisol,9α-Fludrocortisone,Florinef,9α-fluorohydrocortisone,氟氢可的松,Fludrocortisone acetate,Astonin,9α-Fluorcortisol |
Others | Others |
Fludrocortisone (Florinef) 是一种合成皮质类固醇,具有中等的糖皮质激素效力和更大的盐皮质激素效力。Fludrocortisone (Florinef) 可用于治疗低血压的研究。 | |||
T0276 |
Hydrocortisone Valerate
Westcort,氢化可的松戊酸酯 |
Glucocorticoid Receptor | Endocrinology/Hormones |
Hydrocortisone Valerate (Westcort) 具有抗炎、止痒和血管收缩的特性。 | |||
T4602 |
Hydrocortisone hemisuccinate
Hydrocortisone 21-he,氢化可的松琥珀酸酯,hydrocortisone 21-hemisuccinate*free acid,Hydrocortisone 21-hemisuccinate |
Glucocorticoid Receptor; Others; Interleukin | Endocrinology/Hormones; Immunology/Inflammation; Others |
Hydrocortisone hemisuccinate (hydrocortisone 21-hemisuccinate*free acid) 是糖皮质激素, 是口服有活性的甾体抗炎剂。它能够降低IL-6(IC50:6.7 μM)、IL-3(IC50:21.4 μM)的生物活性,可用于研究溃疡性结肠炎。 | |||
T32114 |
Hydrocortisone aceponate
Suniderma,Efficort,Hydrocortisone 17-propionate 21-acetate |
Glucocorticoid Receptor | Endocrinology/Hormones |
Hydrocortisone aceponate (Hydrocortisone 17-propionate 21-acetate) 是一种有效的外用糖皮质激素,以乳膏的形式用于治疗各种皮肤病。 | |||
T0270L |
Hydrocortisone sodium succinate
Cortop,Arcocort,Corlan,A-hydroCort,Buccalsone,Emi-Corlin |
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Hydrocortisone sodium succinate is a glucocorticoid which is used to alleviate allergic reactions, particularly those of the skin and gums. | |||
T13728 |
Hydrocortisone buteprate
HBP,Hydrocortisone probutate |
Others | Others |
Hydrocortisone buteprate (Hydrocortisone probutate) is a medium potent, non-halogenated double-ester of hydrocortisone with a favorable benefit/risk ratio for the treatment of inflammatory skin disorders. | |||
T29628 |
Acyclovir mixture with hydrocortisone
Xerese,ME 609,ME609,ME-609,Lipsovir |
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Acyclovir mixture with hydrocortisone is used for Herpes simplex labialis. | |||
T36927 | Hydrocortisone phosphate | ||
Hydrocortisone phosphate is the pharmaceutical term for cortisol, which is a steroid hormone, in the glucocorticoid class of hormones, increases blood sugar through gluconeogenesis, to suppress the immune system, and to aid in the metabolism of fat, protein, and carbohydrate. | |||
T63227 | Hydrocortisone phosphate sodium | ||
Hydrocortisone phosphate (sodium) (Hydrocortisone 21-phosphate (sodium)) 是一种具有较弱抗炎作用的软类固醇,作用时间短,能够用于研究几种眼部疾病和胃溃疡。 | |||
T19358 | Hydrocortisone cypionate | Others | Others |
Hydrocortisone cypionate is a corticosteroid ester and synthetic glucocorticoid corticosteroid. | |||
T30375 |
Benzodrocortisone
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Benzodrocortisone is a corticosteroid. | |||
T25511 |
Hydrocortisone-21-lysinate
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Hydrocortisone-21-lysinate is a hydrocortisone prodrug that is water soluble. | |||
T16510 |
PF-915275
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Dehydrogenase | Metabolism |
PF-915275 是口服有效的人 11β-羟基类固醇脱氢酶1型选择性抑制剂,Ki 为 2.3 nM,在 HEK293 细胞中的EC50为 15 nM 。它对人和猴原代肝细胞中可的松向皮质醇的转化具有剂量依赖性,EC50分别为 20 nM 和 100 nM。 | |||
T1124 |
Flumethasone
氟米松,Flumetasone,RS-2177,NSC-54702 |
Glucocorticoid Receptor | Endocrinology/Hormones |
Flumethasone (RS-2177) 是皮质类固醇,可局部用药。它可与 Clioquinol 联合使用,研究外耳炎和耳真菌病。它作用于动物模型时,抗炎活性比 Cortisone 高 420 倍。 | |||
T61593 | 11β-HSD1-IN-6 | ||
11β-HSD1-IN-6 is a potent inhibitor of 11β hydroxysteroid dehydrogenase enzymes (11β-HSDs). These enzymes are responsible for catalyzing the conversion of the active glucocorticoids, corticosterone or cortisol, to their respective inactive forms, 11-dehydrocorticosterone (11-DHC) and cortisone. The compound 11β-HSD1-IN-6 specifically targets and inhibits 11β-HSD-1, effectively modulating the interconversion of these glucocorticoids. [1] |
Cat. No. | Product Name | Target | Signaling Pathways |
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T2884 |
Cortisone
Kendall's compound E,17-Hydroxy-11-dehydrocorticosterone,可的松 |
Glucocorticoid Receptor; Endogenous Metabolite | Endocrinology/Hormones; Metabolism |
Cortisone (17-Hydroxy-11-dehydrocorticosterone) 是 Cortisol(一种糖皮质激素)的氧化代谢产物。Cortisone 具有消炎和免疫抑制的作用。Cortisone 在高浓度下对 Glucocorticoid 与Glucocorticoid-receptor 的结合具有部分干预作用。 | |||
T0034 |
Cortisone acetate
醋酸可的松,Cortisone 21-acetate,NSC 49420 |
Glucocorticoid Receptor; Endogenous Metabolite | Endocrinology/Hormones; Metabolism |
Cortisone acetate (NSC-49420) 是 Cortisol(一种糖皮质激素)的氧化代谢产物。它在高浓度下能够部分干预 Glucocorticoid 与Glucocorticoid-receptor 的结合。它具有免疫抑制和消炎的作用。 | |||
T1614 |
Hydrocortisone
氢化可的松,Cortisol |
Glucocorticoid Receptor; Endogenous Metabolite | Endocrinology/Hormones; Metabolism |
Hydrocortisone (Cortisol) 是一种糖皮质激素,由肾上腺素皮质分泌。Hydrocortisone 激动糖皮质激素受体,可促进蛋白质分解代谢、糖异生、毛细血管壁稳定性、肾脏钙排泄,并抑制免疫和炎症反应。 | |||
T1243 |
Hydrocortisone acetate
Cortisol 21-acetate,Hydrocortisone 21-acetate,醋酸氢化可的松 |
Glucocorticoid Receptor; Annexin A; Endogenous Metabolite | Endocrinology/Hormones; GPCR/G Protein; Metabolism |
Hydrocortisone acetate (Cortisol 21-acetate) 是皮质类固醇,能够减少轻微皮肤刺激或痔疮引起的肿胀、搔痒和疼痛。 | |||
T19576 | Tetrahydrocortisone | Others | Others |
Tetrahydrocortisone, a stress-induced hormone and a urinary metabolite of Cortisone, originates from the reduction of Cortisone facilitated by 5-reductase. | |||
T40796 |
5β-Dihydrocortisone
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5β-Dihydrocortisone is a sterol metabolite of cortisone by 5β-reductase (AKR1D1) in liver. |