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Cat. No. Product Name Target Signaling Pathways
T24850 Takeda103A

CMPD103A,Takeda-103A,Takeda-103-A,CMPD-103A,Takeda 103 A

GRK GPCR/G Protein
Takeda103A (CMPD103A) 是 GRK2抑制剂。G 蛋白偶联受体是许多生理过程的核心。Takeda103A 对研究心力衰竭具有潜在的研究价值。
T14565 BI-671800

AP-761,Cmpd A

GPR; Prostaglandin Receptor Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation
BI-671800 (AP-761) 是高特异性的前列腺素 D2 受体拮抗剂,对哮喘有研究潜力,对人和小鼠 CRTH2 转染细胞中 PGD2 结合 CRTH2 的 IC50值分别为 4.5 和 3.7 nM。
T14989 CMPD101

ROCK; GRK; PKC Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; GPCR/G Protein; Stem Cells
CMPD101 是膜透性的 GRK2/3高选择性小分子抑制剂,IC50分别为 18 nM 和 5.4 nM。它针对 GRK1、GRK5 ROCK-2 和 PKCα 的选择性较小,IC50值分别为 3.1 μM,2.3 μM,1.4 μM 和 8.1 μM,可研究心衰疾病。
T70628 Cmpd-A

Cmpd-A is a time-dependent CENP-E inhibitor with potent antitumor activity. Cmpd-A inhibits the ATPase activity of the CENP-E motor domain, acting as a time-dependent inhibitor with an ATP-competitive-like behavior. Cmpd-A causes chromosome misalignment on the metaphase plate, leading to prolonged mitotic arrest. Treatment with Cmpd-A induces antiproliferation in multiple cancer cell lines.
T14988 CMPD1

MAPK MAPK
CMPD1 是非 ATP 竞争性 p38 MAPK 介导的 MK2磷酸化选择性抑制剂(Ki:330 nM)。
T70626 MS 347a

MS 347a is a myosin light chain kinase (MLCK) inhibitor; an epoxide analog of sydowinin B (MS-347b).
T82702 CMPD167

MRK-1

CCR Immunology/Inflammation; Microbiology/Virology
CMPD167 (MRK-1)为口服活性CCR5抑制剂,体外显示出高效的抗病毒能力。
T25267 Cmpd 339509

Cmpd339509,Cmpd-339509

Cmpd 339509 is a DprE1 inhibitor. DprE1 is an epimerase required for cell wall biosynthesis.

化合物

Takeda103A
Cat.No: T24850
Synonym: CMPD103A,Takeda-103A,Takeda-103-A,CMPD-103A,Takeda 103 A
Target: GRK
BI-671800
Cat.No: T14565
Synonym: AP-761,Cmpd A
Target: GPR, Prostaglandin Receptor
CMPD101
Cat.No: T14989
Synonym:
Target: ROCK, GRK, PKC
Cmpd-A
Cat.No: T70628
Synonym:
Target:
CMPD1
Cat.No: T14988
Synonym:
Target: MAPK
MS 347a
Cat.No: T70626
Synonym:
Target:
CMPD167
Cat.No: T82702
Synonym: MRK-1
Target: CCR
Cmpd 339509
Cat.No: T25267
Synonym: Cmpd339509,Cmpd-339509
Target:
TargetMol Loading
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