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7

抑制剂 & 化合物

9

天然产物

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Cat. No. Product Name Target Signaling Pathways
T64511 Sodium cholate

Sodium cholate 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64511。
T6993 Tauroursodeoxycholate sodium

牛磺熊脱氧胆酸钠,Sodium tauroursodeoxycholate,Tauroursodeoxycholic acid sodium salt,TUDC,牛磺熊去氧胆酸钠,Sodium Tauroursodeoxycholate (TUDC)

Apoptosis; ERK; Caspase Apoptosis; MAPK; Proteases/Proteasome
Tauroursodeoxycholate sodium (TUDC) 是一种内质网应激抑制剂。Tauroursodeoxycholate sodium (TUDC) 抑制ERK,显著降低凋亡分子表达,如caspase-3和caspase-12。
T9154 Sodium taurodeoxycholate hydrate

牛磺去氧胆酸钠,Taurodeoxycholic acid sodium salt monohydrate

Others Others
Sodium taurodeoxycholate hydrate (Taurodeoxycholic acid sodium salt monohydrate) 已用于一项研究,以评估亚胶束浓度的胆汁盐对脂质双层膜的影响。
T67974 Berberine ursodeoxycholate

HTD1801,BUDCA

Berberine ursodeoxycholate (HTD1801) 是一种口服有效的降血脂剂 ,是 Berberine 和 Ursodeoxycholic acid 的一种离子盐。Berberine ursodeoxycholate 具有广泛的代谢活性,可显著降低肝脏脂肪含量。Berberine ursodeoxycholate 可用于研究高脂血症、非酒精性脂肪性肝炎 (NASH) 和糖尿病。
T16998 Tauroursodeoxycholate dihydrate

牛磺熊去氧胆酸二水合物,Taurolite dihydrate,TUDCA dihydrate,UR 906 dihydrate

ERK; Caspase Apoptosis; MAPK; Proteases/Proteasome
Tauroursodeoxycholate dihydrate is an endoplasmic reticulum stress inhibitor. Tauroursodeoxycholate also inhibits ERK. Tauroursodeoxycholate significantly decreases the expression of apoptosis molecules, such as caspase-3 and caspase-12.
T66376 Sodium glycocholate hydrate

Sodium glycocholate hydrate 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66376,CAS号为 338950-81-5。
T30270 Azidobenzamidotaurocholate

Azido Benzamido Taurocholate is a bile acid transporter.

化合物

Sodium cholate
Cat.No: T64511
Synonym:
Target:
Tauroursodeoxycholate sodium
Cat.No: T6993
Synonym: 牛磺熊脱氧胆酸钠,Sodium tauroursodeoxycholate,Tauroursodeoxycholic acid sodium salt,TUDC,牛磺熊去氧胆酸钠,Sodium Tauroursodeoxycholate (TUDC)
Target: Apoptosis, ERK, Caspase
Sodium taurodeoxycholate hydrate
Cat.No: T9154
Synonym: 牛磺去氧胆酸钠,Taurodeoxycholic acid sodium salt monohydrate
Target: Others
Berberine ursodeoxycholate
Cat.No: T67974
Synonym: HTD1801,BUDCA
Target:
Tauroursodeoxycholate dihydrate
Cat.No: T16998
Synonym: 牛磺熊去氧胆酸二水合物,Taurolite dihydrate,TUDCA dihydrate,UR 906 dihydrate
Target: ERK, Caspase
Sodium glycocholate hydrate
Cat.No: T66376
Synonym:
Target:
Azidobenzamidotaurocholate
Cat.No: T30270
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T2744 Methyl Cholate

胆酸甲酯,Cholic acid methyl ester

Others Others
Methyl Cholate (Cholic acid methyl ester) 是胆酸的甲酯形式。其中胆酸是一种由肝脏产生的主要胆汁酸,由胆固醇合成。
T2963 Cholic Acid

Cholanic acid,胆汁酸,Cholate,Colalin

Endogenous Metabolite Metabolism
Cholic Acid (Cholate) 是肝脏产生的主要胆汁酸,与牛磺酸或甘氨酸缀合,有助于脂肪吸收和胆固醇排泄。
TN2349 Taurodeoxycholate sodium salt

Sodium taurodeoxylate,牛磺脱氧胆酸钠

Endogenous Metabolite Metabolism
Taurodeoxycholate sodium salt (Sodium taurodeoxylate) 是胆盐相关的阴离子洗涤剂,用于分离膜蛋白,包括线粒体内膜蛋白。它还可以抑制各种炎症反应。
TWA2417 Sodium taurocholate

牛黄胆酸钠(牛胆酸钠,牛胆酸钠盐,牛磺膽酸鈉,牛磺胆酸钠,牛磺胆酸钠盐,牛胆酸钠水合物,水合牛磺胆酸钠,牛胆酸钠(混合物),牛黄胆酸钠(水合),牛磺胆酸钠(标准品)),Taurocholate Sodium

Others Others
Sodium taurocholate (Taurocholate Sodium) hydrate 具有显著的生物学效应,例如通过上调 VEGF-A 的表达抑制肝动脉结扎所致的胆道损伤。对免疫系统具有一定的调节作用。
T0516 Dehydrocholate sodium

去氢胆酸钠,Sodium dehydrocholate

Endogenous Metabolite; Lipid Metabolism
Dehydrocholate sodium 是胆液排泄增多剂,能够提高胆汁输出,清除提高的胆汁酸负载。
T5254 Glycodeoxycholate Sodium

Sodium glycyldeoxycholate,Sodium glycodeoxycholate,Glycodeoxycholic acid sodium salt,脱氧甘胆酸钠

Others; Endogenous Metabolite Metabolism; Others
Glycodeoxycholate Sodium (Glycodeoxycholic acid sodium salt) 诱导肝细胞凋亡的机制与内切酶的DNA裂解有关。它是一种次级胆汁酸,由结肠环境中微生物菌群中存在的酶的作用产生。
T2532 Tauroursodeoxycholate

Taurolite,牛磺熊去氧胆酸,Tauroursodeoxycholic Acid,UR 906,Ursodeoxycholyltaurine,TUDCA

Apoptosis; ERK; P450; Caspase; Endogenous Metabolite Apoptosis; MAPK; Metabolism; Proteases/Proteasome
Tauroursodeoxycholate (UR 906),又称 ursodoxicoltaurine,是一种高度亲水性的三级胆汁酸,在人体内以低浓度产生。Tauroursodeoxycholate 是 ursodeoxycholic acid 更亲水的形式,而 ursodeoxycholic acid 是人类体内自然产生的更丰富的胆汁酸。Tauroursodeoxycholate 正在研究用于几种疾病,如原发性胆汁性肝硬化(PBC)、胰岛素抵抗、淀粉样变性、囊性纤维化、胆汁淤滞和肌萎缩性侧索硬化症。
T13916 Taurochenodeoxycholate-3-sulfate

Others Others
Taurochenodeoxycholate-3-sulfate is a bile salt found in urine.
T2965 Deoxycholic acid

Cholorebic,去氧胆酸,脱氧胆酸,Deoxycholate,Desoxycholic acid,Cholanoic Acid,Cholerebic

Endogenous Metabolite; GPCR19 GPCR/G Protein; Metabolism
Deoxycholic acid (Cholanoic Acid) 是 G 蛋白偶联胆汁酸受体 TGR5的激活剂。

天然产物

Methyl Cholate
Cat.No: T2744
Synonym: 胆酸甲酯,Cholic acid methyl ester
Target: Others
Cholic Acid
Cat.No: T2963
Synonym: Cholanic acid,胆汁酸,Cholate,Colalin
Target: Endogenous Metabolite
Taurodeoxycholate sodium salt
Cat.No: TN2349
Synonym: Sodium taurodeoxylate,牛磺脱氧胆酸钠
Target: Endogenous Metabolite
Sodium taurocholate
Cat.No: TWA2417
Synonym: 牛黄胆酸钠(牛胆酸钠,牛胆酸钠盐,牛磺膽酸鈉,牛磺胆酸钠,牛磺胆酸钠盐,牛胆酸钠水合物,水合牛磺胆酸钠,牛胆酸钠(混合物),牛黄胆酸钠(水合),牛磺胆酸钠(标准品)),Taurocholate Sodium
Target: Others
Dehydrocholate sodium
Cat.No: T0516
Synonym: 去氢胆酸钠,Sodium dehydrocholate
Target: Endogenous Metabolite, Lipid
Glycodeoxycholate Sodium
Cat.No: T5254
Synonym: Sodium glycyldeoxycholate,Sodium glycodeoxycholate,Glycodeoxycholic acid sodium salt,脱氧甘胆酸钠
Target: Others, Endogenous Metabolite
Tauroursodeoxycholate
Cat.No: T2532
Synonym: Taurolite,牛磺熊去氧胆酸,Tauroursodeoxycholic Acid,UR 906,Ursodeoxycholyltaurine,TUDCA
Target: Apoptosis, ERK, P450, Caspase, Endogenous Metabolite
Taurochenodeoxycholate-3-sulfate
Cat.No: T13916
Synonym:
Target: Others
Deoxycholic acid
Cat.No: T2965
Synonym: Cholorebic,去氧胆酸,脱氧胆酸,Deoxycholate,Desoxycholic acid,Cholanoic Acid,Cholerebic
Target: Endogenous Metabolite, GPCR19
TargetMol Loading
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