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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T60054 EJMC-1

N-(3-chloro-4-hydroxyphenyl)-2-oxo-1,2-dihydrobenzo[cd]indole-6-sulfonamide

TNF Apoptosis
EJMC-1 是一种 TNF-α 抑制剂,IC50 值为 42 μM,可用于自身炎症性疾病的研究。
T9210 CD73-IN-4

CD73 Immunology/Inflammation
CD73-IN-4 是高选择性的亚甲基膦酸 CD73抑制剂,对人 CD73 作用的 IC50值为 2.6 nM,在癌症免疫学中具有研究潜力。
T4371 CD437

AHPN,O-Desmethyl Adapalene,6-[3-(1-金刚烷基)-4-羟基苯基]-2-萘甲酸,Apoptosis Activator VI

Retinoid Receptor; Autophagy Autophagy; Metabolism
CD437 (AHPN) 是一种特异性视黄酸受体激动剂。
T71094 CD4 (81-92)

CD4 (81-92) is a peptide that was previously found to inhibit gp120 binding, HIV-1 infectivity, and syncytium formation.
T4698 8-Fluoro-1,3,4,5-tetrahydro-6H-azepino[5,4,3-cd]indol-6-one

8-氟-1,3,4,5-四氢-2-[4-[(甲基氨基)甲基]苯基]-6H-吡咯并[4,3,2-EF][2]苯并氮杂-6-酮

Others Others
8-Fluoro-1,3,4,5-tetrahydro-6H-azepino[5,4,3-cd]indol-6-one 用作医药中间体。
T35388 Anti-mouse CD4-InVivo

Anti-mouse CD4-InVivo

gp120/CD4 Immunology/Inflammation
Anti-mouse CD4-InVivo 一种抗小鼠 CD4 抗体抑制剂,可用于生命科学领域的相关研究,其产品编号为 T35388。
T38100 Betamethasone 21-phosphate (sodium salt hydrate)

Betamethasone 21-phosphate is a synthetic glucocorticoid.1It prevents increases in macrophage and eosinophil numbers in bronchoalveolar lavage fluid (BALF) and decreases in blood leukocyte numbers in a guinea pig model of parainfluenza-3 viral infection when administered at a dose of 8 mg/kg but does not prevent airway hyperresponsiveness after infection.2Betamethasone 21-phosphate inhibits cell infiltration into the aqueous humor in a rat model of endotoxin-induced uveitis when administered top...

化合物

EJMC-1
Cat.No: T60054
Synonym: N-(3-chloro-4-hydroxyphenyl)-2-oxo-1,2-dihydrobenzo[cd]indole-6-sulfonamide
Target: TNF
CD73-IN-4
Cat.No: T9210
Synonym:
Target: CD73
CD437
Cat.No: T4371
Synonym: AHPN,O-Desmethyl Adapalene,6-[3-(1-金刚烷基)-4-羟基苯基]-2-萘甲酸,Apoptosis Activator VI
Target: Retinoid Receptor, Autophagy
CD4 (81-92)
Cat.No: T71094
Synonym:
Target:
8-Fluoro-1,3,4,5-tetrahydro-6H-azepino[5,4,3-cd]indol-6-one
Cat.No: T4698
Synonym: 8-氟-1,3,4,5-四氢-2-[4-[(甲基氨基)甲基]苯基]-6H-吡咯并[4,3,2-EF][2]苯并氮杂-6-酮
Target: Others
Anti-mouse CD4-InVivo
Cat.No: T35388
Synonym: Anti-mouse CD4-InVivo
Target: gp120/CD4
Betamethasone 21-phosphate (sodium salt hydrate)
Cat.No: T38100
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T4S0498 Glaucocalyxin A

蓝萼甲素,Wangzaozin B,Leukamenin F

Apoptosis; Akt; Caspase; PI3K Apoptosis; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Glaucocalyxin A (Leukamenin F) 是来自日本黑纹病菌的一种对映型月桂基二萜,具有抗肿瘤作用。它通过调节PI3K/Akt 信号通路抑制 GLI1 的核易位,诱导骨肉瘤凋亡。

天然产物

Glaucocalyxin A
Cat.No: T4S0498
Synonym: 蓝萼甲素,Wangzaozin B,Leukamenin F
Target: Apoptosis, Akt, Caspase, PI3K
TargetMol Loading
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