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Cat. No. Product Name Target Signaling Pathways
T7544 Fucoidan

岩藻多糖

Others Others
Fucoidan 是一种 α-淀粉酶和 α-葡萄糖苷酶的有效抑制剂,是一种生物特性多糖。 它具有抗凝血,抗肿瘤,抗氧化和抗脂肪特性。
TN1990 Norathyriol

芒果苷元

Akt; DNA/RNA Synthesis; AMPK; PPAR Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; Metabolism; PI3K/Akt/mTOR signaling
Norathyriol 是来自芒果的芒果苷代谢物,具有抗氧化、抗癌、抗菌和抗炎活性。它以非竞争性方式抑制 α-葡萄糖苷酶,IC50为 3.12 μM。它还抑制PPARα、PPARβ和PPARγ,IC50分别为 92.8、102.4 和 153.5 µM。
T2S1158 4,5-Dicaffeoylquinic acid

3,4-Dicaffeoylquinic acid,异绿原酸C(4,5),Isochlorogenic acid C

Others; HBV; Endogenous Metabolite Metabolism; Microbiology/Virology; Others
4,5-Dicaffeoylquinic acid (Isochlorogenic acid C) 是一种天然产物,有抗病毒、抗肝毒性活性。
T6S1371 Isovitexin

Homovitexin,Saponaretin,Apigenin-6-C-Glucoside,异牡荆黄素

NF-κB; JNK; Glucosidase MAPK; Metabolism; NF-κB
Isovitexin (Apigenin-6-C-Glucoside) 是从亚洲水稻种得到的一种黄酮,具有抗氧化和抗炎活性。它的作用与JNK1/2的抑制剂类似,抑制NF-κB 的活化。
T6S1369 Vitexin

牡荆素,Apigenin-8-C-glucoside

Antioxidant oxidation-reduction
Vitexin 是一种存在于多种药用植物(如榕树、螺旋藻)中的 c-糖基化的黄酮。 它具有广泛的药理作用,包括抗氧化,抗癌,抗炎,抗痛觉过敏和神经保护作用。
T3851 Vicenin 2

Vicenin -2,维采宁 2,新西兰牡荆苷

RAAS Endocrinology/Hormones
Vicenin 2 来源于广金钱草 (Desmodium styracifolium) 的地上部分。Vicenin 2 是一种血管紧张素转换酶 (ACE) 抑制剂,IC50=43.83 μM。
TMA1890 Icariside F2

淫羊藿次苷F2

NF-κB NF-κB
Icariside F2 shows modest α-glucosidase inhibitory (4.60±1.74% to 11.97±3.30%) and antioxidant activities. It also displays potent NF-κB inhibitory effects, with the IC50 value of 16.25 ± 2.19 uM.
TN5192 Tuberosin

NOS; Glucokinase Immunology/Inflammation; Metabolism
Tuberosin shows anti-inflammatory and antioxidant activities.It demonstrated a significantly potent inhibition on yeast α-glucosidase in a dose dependent manner.
TN1820 cis-Tiliroside

Kaempferol-3-O-(6''-O-cis-coumaryl)glucoside,山奈酚-3-O-(6''-O-顺-香豆酰基)葡萄糖苷,顺式银椴苷

Others Others
Kaempferol-3-O-α2-D-(6''-O-coumaryl) glycoside has antioxidant activity and α±-glucosidase inhibitory effects, it could potentially be used for food additives and the development of useful natural compounds.
T79980 Flaccidoside III

Glucosidase Metabolism
Flaccidoside III, 分离自黑种草(N. sativa)地上部分的一种类黄酮和三萜类化合物,具有抑制α-Glucosidase(IC50:256.7 μM)的活性,表现出潜在的抗氧化和抗糖尿病效应。
TN5090 Tachioside

Glucokinase Metabolism
Tachioside has antiobesity, antioxidant and α-glucosidase inhibitory activities, it decreases lipid content in 3T3-L1 adipocytes by inhibiting lipogenesis, shows antiobesity activities. Tachioside can inhibit nitric oxide production in lipopolysaccharides-stimulated RAW 264.7 cells with IC50 value of 12.14 μM.
TWS0787 Oroxin A

木蝴蝶苷A,Baicalin-7-glucoside

PPAR; Glucosidase DNA Damage/DNA Repair; Metabolism
Oroxin A (Baicalin-7-glucoside) 是一种部分 PPARγ 激动剂,可在体外和体内激活 PPARγ 转录激活。 Oroxin A 还表现出对 α-葡萄糖苷酶的抑制活性和抗氧化能力。
T73402 Flavipin

Flavipin 是一种芳香烃受体(Ahr)激动剂,可诱导小鼠 CD4+T 细胞和 CD11b+巨噬细胞表达 Ahr 下游基因。Flavipin 抑制 Arid5a 在 Il23a3'UTR 上的稳定功能,这是一种新发现的靶 mRNA。Flavipin 具有清除 DPPH 自由基的能力,IC50值为7.2 μM,对α-葡萄糖苷酶具有较强的抑制作用,IC50值为 33.8 μM。

天然产物

Fucoidan
Cat.No: T7544
Synonym: 岩藻多糖
Target: Others
Norathyriol
Cat.No: TN1990
Synonym: 芒果苷元
Target: Akt, DNA/RNA Synthesis, AMPK, PPAR
4,5-Dicaffeoylquinic acid
Cat.No: T2S1158
Synonym: 3,4-Dicaffeoylquinic acid,异绿原酸C(4,5),Isochlorogenic acid C
Target: Others, HBV, Endogenous Metabolite
Isovitexin
Cat.No: T6S1371
Synonym: Homovitexin,Saponaretin,Apigenin-6-C-Glucoside,异牡荆黄素
Target: NF-κB, JNK, Glucosidase
Vitexin
Cat.No: T6S1369
Synonym: 牡荆素,Apigenin-8-C-glucoside
Target: Antioxidant
Vicenin 2
Cat.No: T3851
Synonym: Vicenin -2,维采宁 2,新西兰牡荆苷
Target: RAAS
Icariside F2
Cat.No: TMA1890
Synonym: 淫羊藿次苷F2
Target: NF-κB
Tuberosin
Cat.No: TN5192
Synonym:
Target: NOS, Glucokinase
cis-Tiliroside
Cat.No: TN1820
Synonym: Kaempferol-3-O-(6''-O-cis-coumaryl)glucoside,山奈酚-3-O-(6''-O-顺-香豆酰基)葡萄糖苷,顺式银椴苷
Target: Others
Flaccidoside III
Cat.No: T79980
Synonym:
Target: Glucosidase
Tachioside
Cat.No: TN5090
Synonym:
Target: Glucokinase
Oroxin A
Cat.No: TWS0787
Synonym: 木蝴蝶苷A,Baicalin-7-glucoside
Target: PPAR, Glucosidase
Flavipin
Cat.No: T73402
Synonym:
Target:
TargetMol Loading
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