Powder: -20°C for 3 years | In solvent: -80°C for 1 year
JTE-907 是一种具有高度选择性和口服活性的 CB2 受体反向激动剂。JTE-907在体内展现出抗炎活性。
规格 | 价格/CNY | 货期 | 数量 | |
---|---|---|---|---|
1 mg | ¥ 673 | 现货 | ||
5 mg | ¥ 1,730 | 现货 | ||
10 mg | ¥ 2,770 | 现货 | ||
25 mg | ¥ 4,620 | 现货 | ||
50 mg | ¥ 6,580 | 现货 | ||
100 mg | ¥ 8,890 | 现货 | ||
500 mg | ¥ 17,800 | 6-8周 | ||
1 mL * 10 mM (in DMSO) | ¥ 2,080 | 现货 |
产品描述 | JTE-907 is a CB2 receptor inverse agonist with high selectivity and oral activity.JTE-907 exhibits anti-inflammatory activity in vivo. |
体外活性 | JTE 907 acts as a Gq-coupled agonist in islets to stimulate insulin secretion and maintain β-cell mass in a GPR55-independent fashion. JTE 907 (10 μM) significantly stimulated insulin secretion from islets isolated from human donors and islets from Gpr55+/+ and Gpr55-/- mice. These stimulatory effects were accompanied by significant elevations of IP1 and [Ca2+]i, but there were no changes in cAMP generation. JTE 907 also significantly reduced cytokine-induced apoptosis in human and mouse islets and promoted human β-cell proliferation.[4] |
别名 | JTE 907 |
分子量 | 438.47 |
分子式 | C24H26N2O6 |
CAS No. | 282089-49-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 112.5 mg/mL (256.6 mM), Sonication is recommended.
可选溶剂 | 浓度 体积 质量 | 1 mg | 5 mg | 10 mg | 25 mg |
DMSO | 1 mM | 2.2807 mL | 11.4033 mL | 22.8066 mL | 57.0164 mL |
5 mM | 0.4561 mL | 2.2807 mL | 4.5613 mL | 11.4033 mL | |
10 mM | 0.2281 mL | 1.1403 mL | 2.2807 mL | 5.7016 mL | |
20 mM | 0.114 mL | 0.5702 mL | 1.1403 mL | 2.8508 mL | |
50 mM | 0.0456 mL | 0.2281 mL | 0.4561 mL | 1.1403 mL | |
100 mM | 0.0228 mL | 0.114 mL | 0.2281 mL | 0.5702 mL |
对于不同动物的给药剂量换算,您也可以参考 更多...
请在以下方框中输入您的动物实验信息后点击计算,可以得到母液配置方法和体内配方的制备方法: 比如您的给药剂量是10 mg/kg,每只动物体重20 g,给药体积100 μL,一共给药动物10 只,您使用的配方为5% DMSO+30% PEG300+5% Tween 80+60% ddH2O。那么您的工作液浓度为2 mg/mL。
母液配置方法:2 mg 药物溶于 50 μL DMSO (母液浓度为 40 mg/mL), 如您需要配置的浓度超过该产品的溶解度,请先与我们联系。
体内配方的制备方法:取 50 μL DMSO 主液,加入 300 μL PEG300, 混匀澄清,再加 50 μL Tween 80,混匀澄清,再加 600 μL ddH2O, 混匀澄清。
您可能有的问题的答案可以在抑制剂处理说明中找到,包括如何准备库存溶液,如何存储产品,以及基于细胞的分析和动物实验需要特别注意的问题。
JTE-907 282089-49-0 GPCR/G Protein Cannabinoid Receptor JTE907 JTE 907 Inhibitor inhibitor inhibit