Cat. No. | Product Name | CAS No. | Purity | Chemical Structure |
---|---|---|---|---|
T11044 | Dihydromunduletone
化合物Dihydromunduletone
|
674786-20-0 | 99.96% |
|
Dihydromunduletone (DHM) 是一种粘附 G 蛋白偶联受体 (aGPCR)拮抗剂,可做一种化学探针,对具有相似拴系激动剂的 GPR56 和 GPR114/ADGRG5 有抑制作用。 | ||||
T62858 | HGPR91 antagonist 3
hGPR91拮抗剂3
|
1314796-31-0 | 98.82% |
|
hGPR91 antagonist 3 是一种具有口服活性、有效性和选择性的 hGPR91 拮抗剂。hGPR91 antagonist 3 可用于研究高血压、自身免疫性疾病和视网膜血管生成方面的疾病。 | ||||
T4689 | Palosuran hydrochloride 540769-28-6(free base)
化合物Palosuran hydrochloride
|
T4689 |
|
|
Palosuran hydrochloride 540769-28-6(free base) (ACT-058362 hydrochloride) 是一种新型强效特异性人 UT 受体拮抗剂,IC50 为 3.6±0.2 nM。 | ||||
TQ0241 | TUG-770
化合物TUG-770
|
1402601-82-4 | 98% |
|
TUG-770 is a highly potent agonist of free fatty acid receptor 1 (FFA1/GPR40, EC50: 6 nM for hFFA1). | ||||
T10507 | GPR40 Agonist 2
化合物 T10507
|
1147729-48-3 | 98% |
|
GPR40 Agonist 2 is a GPR40 agonist. It can be used in the research of diabetes. | ||||
T15283 | Firuglipel
化合物 T15283
|
1371591-51-3 | 98% |
|
Firuglipel is an orally available and selective agonist of GPR119. | ||||
T14200 | AM-1638
化合物 T14200
|
1142214-62-7 | 98% |
|
AM-1638 is a full agonist of GPR40/FFA1 (EC50: 0.16 μM). | ||||
T14202 | AM-4668
化合物 T14202
|
1011531-27-3 | 98% |
|
AM-4668 is a type 2 diabetes GPR40 agonist. For GPR40, in A9 cells (GPR40 IP3 assay) and CHO cells (GPR40 aequorin assay), the EC50s are 3.6 nM and 36 nM, respec... | ||||
T37264 | 15(R)-15-methyl Prostaglandin D2
化合物 T37264
|
210978-26-0 | 98% |
|
15(R)-15-methyl Prostaglandin D2 (15(R)15methyl PGD2) 是一种 PGD2 合成类似物,也是一种具有选择性和强效性的 CRTH2/DP2 受体激动剂,可调节嗜酸性粒细胞 CD11b 表达、肌动蛋白聚合和趋化。 | ||||
T15448 | GW-1100
化合物 T15448
|
306974-70-9 | 98% |
|
GW-1100 is a selective antagonist of GPR40 (pIC50: 6.9). GW1100 also plays the role of a GPR40 inverse agonist. | ||||
T2351L | TAK-875 Hemihydrate
化合物TAK-875 Hemihydrate
|
1374598-80-7 | 98% |
|
TAK-875 Hemihydrate (Fasiglifam) 是一种选择性 GPR40 激动剂,EC50 为 14 nM,比油酸强 400 倍。 | ||||
T11452 | GPR120 Agonist 1
化合物 T11452
|
1628448-77-0 | 98% |
|
GPR120 Agonist 1 is a selective GPR120 agonist. In GPR120 transfected HEK293 cells, GPR120 Agonist 1 displays good EC50 of 42 nM and 77 nM for human and mouse GP... | ||||
T11460 | GPR4 antagonist 1
化合物 T11460
|
1197879-16-5 | 98% |
|
GPR4 antagonist 1 is a GPR4 antagonist (IC50: 189 nM). | ||||
TP2166 | Urotensin II, mouse TFA (9047-55-6 free base)
化合物 TP2166
|
TP2166 | 98% |
|
Urotensin II, mouse TFA is an endogenous ligand for the orphan GPR14 or SENR. It is a potent vasoconstrictor. | ||||
T12778L | RTI-13951-33
化合物 T12778L
|
2244884-08-8 | 98% |
|
RTI-13951-33 is an effective and brain-penetrant GPR88 agonist (EC50: 25 nM, in GPR88 cAMP functional assay). | ||||
TQ0051 | MK-7246
化合物MK-7246
|
1218918-62-7 | 98% |
|
MK-7246 is a potent and specific CRTH2 antagonist (Ki: 2.5 nM). | ||||
T11462 | GPR84 antagonist 8
化合物 T11462
|
1445846-30-9 | 98% |
|
GPR84 antagonist 8 is a selective GPR84 antagonist. | ||||
T21623 | AS1269574
化合物AS 1269574
|
330981-72-1 | 99.98% |
|
AS1269574 是口服有效的GPR119激动剂,在表达人 GPR119 的 HEK293 细胞中EC50为 2.5 μM。它激活 TRPA1 阳离子通道,刺激胰高血糖素样肽-1分泌。它仅在高糖条件下特异性诱导胰腺 β 细胞分泌葡萄糖依赖性胰岛素。它在 2 型糖尿病的研究中具有价值。 | ||||
T2088 | APD668
化合物APD 668
|
832714-46-2 | 99.97% |
|
APD668 是选择性的,口服有效的GPR119激动剂,对hGPR119和rGPR119的EC50分别为 2.7 nM 和 33 nM。它对除CYP2C9(Ki=0.1 μM) 以外的五种主要 CYP 亚型均无明显抑制作用。它可用于脂肪性肝炎和糖尿病的研究。 | ||||
T2396 | Ramatroban
雷马曲班
|
116649-85-5 | 99.96% |
|
Ramatroban (BAY u3405) 是一种血栓素 A(2) (TxA(2)) 拮抗剂,IC50为 14 nM。它还通过抑制PGD2结合从而拮抗CRTH2,IC50为113 nM。它用于治疗过敏性鼻炎,可用于治疗哮喘的研究。 |