Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2841 |
Plumbagin
Plumbagone,Plumbagine,白花丹素,Plumbaein,2-Methyljuglone |
ROS | Immunology/Inflammation |
Plumbagin (Plumbaein) 是一种萘醌类物质,从Plumbago zeylanica L 中获得,具有抗肿瘤、抗增殖作用。 | |||
TN1552 |
7,8-Dimethoxycoumarin
7,8-dimethoxychromen-2-one,Daphnetin dimethyl ether |
Others | Others |
7,8-Dimethoxycoumarin 是一种从 Artemisia caruifolia 和 Wikstroemia indica 中分离出来的天然产物。 | |||
T20189 |
Benzoylphenylalanine
L-BPA,NSC118532,N-Benzoyl-L-phenylalanine,LBPA,NSC-118532,L BPA,N-苯甲酰-L-苯丙氨酸,NSC 118532 |
Others | Others |
Benzoylphenylalanine (LBPA) 可用作光亲和肽灭活剂。 | |||
T3S2390 |
Caftaric acid
trans-Caftaric acid,单咖啡酰洒石酸 |
Others | Others |
Caftaric acid (trans-Caftaric acid) 是一种具有抗氧化和抗炎作用的天然产物,具有抗致突变性,也是Src 家族激酶介导的蛋白质-蛋白质相互作用的抑制剂。 | |||
T7050 |
alpha-Tocopherolquinone
托可醌,Metarene |
Antioxidant | oxidation-reduction |
alpha-Tocopherolquinone (Metarene) 会下调线粒体的呼吸活动。在还原为生育酚氢醌后,它还显示出抗氧化活性。在大鼠缺氧期间,已发现它的水平升高。 | |||
TL0006 |
Cichoric Acid
菊苣酸,Dicaffeoyltartaric acid,Chicoric Acid |
Reactive Oxygen Species; HIV Protease | Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome |
Cichoric Acid (Dicaffeoyltartaric acid) 是一种天然化合物,具有抗氧化作用。 | |||
TN4368 |
Kaempferol-3,7-di-O-β-glucoside
Kaempferol 3,7-di-O-glucoside |
Glucosidase; Amylase | Metabolism |
Kaempferol-3,7-di-O-β-glucoside (Kaempferol 3,7-diglucoside) 是一种来自 Morettia philaena 的黄酮醇,对 α-淀粉酶 (α-amylase)、α-葡萄糖苷酶 (α-glucosidase) 和乙酰胆碱酯酶 (Acetylcholinesterase) 具有抑制作用。Kaempferol-3,7-di-O-β-glucoside 具有神经保护活性,可减缓分化神经元细胞 SH-SY5Y 免受 Amyloid β 肽诱导的损伤。Kaempferol-3,7-di-O-β-glucoside 可用于研究阿尔茨海默氏症类的神经系统疾病。 | |||
T6S1294 |
Nicotiflorin
Nictoflorin,Kaempferol-3-O-Rutinoside,山奈酚-3-O-芸香糖苷,Nicotifloroside |
Others | Others |
Nicotiflorin (Kaempferol-3-O-Rutinoside) 是一种黄酮苷,从传统中药Flos Carthami 中提取得到。它有抗糖化活性和神经保护作用。 | |||
T3863 |
Chikusetsusaponin IVa
竹节参皂苷IVa,Calenduloside F,竹节人参皂苷 IVA |
AMPK | Chromatin/Epigenetic; PI3K/Akt/mTOR signaling |
Chikusetsusaponin IVa (Calenduloside F) 是一种三萜皂苷中主要的活性成分,是一种蛋白激酶的激活剂,对血栓及一些代谢性疾病具有抵抗作用。 | |||
TN3233 |
7-Hydroxy-5-methylflavon
|
Others | Others |
7-Hydroxy-5-methylflavon 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3233,CAS号为 15235-99-1。 | |||
TN6861 | Euphorbetin | ||
Euphorbetin is a natural product. | |||
TN6501 | Isololiolide | ||
Isololiolide has phytotoxicity, it inhibited seedling growth of cress and barnyard grass. It also showed in vitro activity against both trypomastigote and intracellular amastigotes of Trypanosoma cruzi, with IC50 values of 32 μM and 40 μM, respectively. I | |||
TN4270 |
Isocarlinoside
|
||
Isocarlinoside,是一种二-C-糖基黄酮,可从Lespedeza capitate中分离得到。 | |||
TN1394 |
Apigenin6-C-α-L-arabinopyranosyl-8-C-β-D-xylopyranoside
Apigenin 6-C-alpha-L-arabinopyranosyl-8-C-beta-D-xylopyranoside,芹菜素-6-C-Α-L-吡喃阿拉伯糖-8-C-Β-D-吡喃木糖苷,apigenin6-c-alpha-l-arabinopyranosyl-8-c-beta-d-xylopyranoside |
Others | Others |
Apigenin 6-C-alpha-L-arabinopyranosyl-8-C-beta-D-xylopyranoside is a natural product from Viola yedoensis. | |||
TN5065 |
Stigmasta-4,25-dien-3-one
|
Others | Others |
Stigmasta-4,25-dien-3-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5065,CAS号为 848669-08-9。 | |||
TN5174 | Trichosanatine | MMP; LDL; p38 MAPK; Lipoxygenase; ROS | Immunology/Inflammation; MAPK; Metabolism; Proteases/Proteasome |
Trichosanatine and squamosamide, as potential candidates as lead compounds for further study in drug development process with the PP2A- α protein. Trichosanatine can alleviate oxidized low-density lipoprotein induced endothelial cells injury via inhibiting the LOX-1/p38 MAPK pathway. | |||
TN6974 |
(-)-Isobicyclogermacrenal
|
||
(-)-Isobicyclogermacrenal is a natural product. | |||
TN6942 |
Chlorophyll a
|
||
Chlorophyll a is a natural product. | |||
TN3523 |
Blumenol B
|
Others | Others |
Blumenol B是一种天然产物,属于蔷薇科蔷薇属,其产品编号为 TN3523,CAS号为 36151-01-6。Blumenol B可用作对照参考。 | |||
TN6981 | daphneticin | ||
daphneticin is a natural product. | |||
TN4236 |
Hydrangetin
7-Hydroxy-8-methoxycoumarin |
Others | Others |
Hydrangetin (7-Hydroxy-8-methoxycoumarin) 是一种来自 Daphne papyracea var 的小分子化合物,可抑制血小板聚集。 | |||
TN4613 |
(-)-N-methylcoclaurine
N-Methylcoclaurine |
Others | Others |
N-Methylcoclaurine shows binding affinities for the ĸ opioid receptor with the equilibrium dissociation constant (Ki) value of 0.9 ± 0.1 uM. N-methylcoclaurine also shows promising butyrylcholinesterase inhibition activities, with the IC50 value of 1 | |||
TN2928 |
Pygenic acid A
3-Epicorosolic acid,脓毒酸A |
||
3-Epicorosolic acid has a potent inhibitory effect on Epstein-Barr virus early antigen (EBV-EA) induction, it has potential anti-inflammatory activities as well as cancer chemopreventive activity.3-Epicorosolic acid shows both potent α-glucosidase and pro |