7
3
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0276 |
Hydrocortisone Valerate
Westcort,氢化可的松戊酸酯 |
Glucocorticoid Receptor | Endocrinology/Hormones |
Hydrocortisone Valerate (Westcort) 具有抗炎、止痒和血管收缩的特性。 | |||
T0270 |
Hydrocortisone 17-butyrate
丁酸氢化可的松,Cortisol 17-butyrate,Hydrocortisone butyrate |
Glucocorticoid Receptor; Annexin A; Adrenergic Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Hydrocortisone 17-butyrate (Cortisol 17-butyrate) 是一种肾上腺皮质激素类药物。 | |||
T4602 |
Hydrocortisone hemisuccinate
Hydrocortisone 21-he,氢化可的松琥珀酸酯,hydrocortisone 21-hemisuccinate*free acid,Hydrocortisone 21-hemisuccinate |
Glucocorticoid Receptor; Others; Interleukin | Endocrinology/Hormones; Immunology/Inflammation; Others |
Hydrocortisone hemisuccinate (hydrocortisone 21-hemisuccinate*free acid) 是糖皮质激素, 是口服有活性的甾体抗炎剂。它能够降低IL-6(IC50:6.7 μM)、IL-3(IC50:21.4 μM)的生物活性,可用于研究溃疡性结肠炎。 | |||
T32114 |
Hydrocortisone aceponate
Suniderma,Efficort,Hydrocortisone 17-propionate 21-acetate |
Glucocorticoid Receptor | Endocrinology/Hormones |
Hydrocortisone aceponate (Hydrocortisone 17-propionate 21-acetate) 是一种有效的外用糖皮质激素,以乳膏的形式用于治疗各种皮肤病。 | |||
T19358 | Hydrocortisone cypionate | Others | Others |
Hydrocortisone cypionate is a corticosteroid ester and synthetic glucocorticoid corticosteroid. | |||
T34298 |
Retene
NSC 26317,NSC-26317,NSC26317 |
||
Retene (NSC-26317) 广泛存在于近代和古代沉积物中,可从冷杉林土壤、腐殖质煤、陆相石油烃源岩和深海沉积物中提取得到化合物。Retene 是松木酸在成岩作用过程中脱氢产生的。 | |||
T16510 |
PF-915275
|
Dehydrogenase | Metabolism |
PF-915275 是口服有效的人 11β-羟基类固醇脱氢酶1型选择性抑制剂,Ki 为 2.3 nM,在 HEK293 细胞中的EC50为 15 nM 。它对人和猴原代肝细胞中可的松向皮质醇的转化具有剂量依赖性,EC50分别为 20 nM 和 100 nM。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1614 |
Hydrocortisone
氢化可的松,Cortisol |
Glucocorticoid Receptor; Endogenous Metabolite | Endocrinology/Hormones; Metabolism |
Hydrocortisone (Cortisol) 是一种糖皮质激素,由肾上腺素皮质分泌。Hydrocortisone 激动糖皮质激素受体,可促进蛋白质分解代谢、糖异生、毛细血管壁稳定性、肾脏钙排泄,并抑制免疫和炎症反应。 | |||
T1243 |
Hydrocortisone acetate
Cortisol 21-acetate,Hydrocortisone 21-acetate,醋酸氢化可的松 |
Glucocorticoid Receptor; Annexin A; Endogenous Metabolite | Endocrinology/Hormones; GPCR/G Protein; Metabolism |
Hydrocortisone acetate (Cortisol 21-acetate) 是皮质类固醇,能够减少轻微皮肤刺激或痔疮引起的肿胀、搔痒和疼痛。 | |||
T1560 |
Prednisolone
氢化泼尼松,Predonine,Hydroretrocortine,泼尼松龙,Metacortandralone |
Glucocorticoid Receptor; Endogenous Metabolite | Endocrinology/Hormones; Metabolism |
Prednisolone (Hydroretrocortine) 是有口服活性的皮质类固醇和糖皮质激素。它的抗炎特性约为氢化可的松的四倍,同时减少了水和盐的保留。它能够用于眼部抗炎研究。 |