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20

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T8133 SulfadiMethoxine sodium

Anti-infection; Antibacterial; Antibiotic Microbiology/Virology
SulfadiMethoxine sodium 是一种磺胺类抗生素,可研究由多种感染引起的疾病。
T1078 Sulfadimethoxine

Sulphadimethoxine,磺胺二甲氧嗪

Antibacterial; Antibiotic Microbiology/Virology
Sulfadimethoxine (Sulphadimethoxine) 是一种磺胺类抗生素,用于多种感染引起的疾病的研究。
T0116 Balofloxacin

DNA gyrase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Balofloxacin 是一种具有口服活性的氟喹诺酮类抗生素,可通过干扰 DNA 促旋酶来抑制细菌 DNA 的合成,对革兰氏阴性,革兰氏阳性和厌氧菌具有广谱抗菌活性。它可研究呼吸道,肠道和泌尿道感染。
T1495 Cefaclor monohydrate

Cefaclor,头孢克洛一水物,头孢克洛一水合物,Cefaclorum,Cefachlor

Antibacterial; Antibiotic Microbiology/Virology
Cefaclor monohydrate (Cefaclorum) 是一种抗生素,可特异性地结合青霉素结合蛋白。
T6436 Cefaclor

Panoral,Kefral,Cefaclorum,头孢克洛

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Cefaclor (Panoral) 是一种可特异性结合青霉素结合蛋白的抗生素。
T0284 Sulfogaiacol

guaiacolsulfonate,愈创木酚磺酸钾

Others; Antibacterial Microbiology/Virology; Others
Sulfogaiacol (guaiacolsulfonate) 是一种镇咳剂,可研究急性呼吸道感染。
T19794 Temafloxacin

替马沙星,Omniflox

Antibiotic Microbiology/Virology
Temafloxacin (Omniflox) 是一种喹诺酮类广谱抗菌剂,对革兰氏阳性菌、革兰氏阴性菌和厌氧菌均有效。
T8134 Cefathiamidine

Antibacterial; Antibiotic Microbiology/Virology
Cefathiamidine 是一种头孢菌素抗菌剂,可研究由易感细菌引起的感染,还可用于呼吸道、肝脏、五官感觉、尿路感染以及心内膜炎和败血症的研究。
T26974 Cefetamet Hydrochloride

Cefetamet HCl,Cefetamet

Cefetamet is a potent antibiotic to treat respiratory and urinary tract infections.
T68999 Cefonicid (free base)

Cefonicid (free base) is a second-generation cephalosporin administered intravenously or intramuscularly. Its bactericidal action results from inhibition of cell wall synthesis. It is used for urinary tract infections, lower respiratory tract infections, and soft tissue and bone infections.
T68817 Cefonicid monosodium

Cefonicid monosodium is the salt form of Cefonicid (free base), a second-generation cephalosporin administered intravenously or intramuscularly. Its bactericidal action results from inhibition of cell wall synthesis. It is used for urinary tract infections, lower respiratory tract infections, and soft tissue and bone infections.
T72093 Thiamphenicol glycinate hydrochloride

甲砜霉素甘氨酸酯盐酸盐

Thiamphenicol glycinate hydrochloride 是一种广谱抗菌剂,可用于呼吸道感染的研究。
T75274 Cefetamet

Cefetamet 是一种头孢类抗生素。Cefetamet 具有研究上、下社区获得性呼吸道感染的潜力。
T63214 Lomefloxacin (aspartate)

Lomefloxacin (SC47111A) aspartate 是广谱的喹诺酮类抗菌剂,能够用于呼吸道感染、胃肠道感染、泌尿生殖系统感染、耳鼻喉感染等疾病的研究。
T40971 Dehydroandrographolide succinate potassium sodium salt

Dehydroandrographolide succinate (potassium sodium salt), derived from the herbal medicine Andrographis paniculata (Burm f) Nees, is a versatile compound highly utilized for the treatment of viral pneumonia and viral upper respiratory tract infections due to its potent immunostimulatory, anti-infective, and anti-inflammatory properties.
T11819 Lascufloxacin

拉库沙星,KRP-AM1977X

Others Others
Lascufloxacin () 是一种有效的、具有口服活性的氟喹诺酮类抗菌剂。Lascufloxacin 有效抑制由多种病原体 (包括对喹诺酮类耐药的菌株) 引起的感染。Lascufloxacin 可用于多种传染病的研究,包括下呼吸道感染。
T75286 Sitafloxacin hydrochloride

Sitafloxacin (DU6859a) hydrochloride 是一款有效的口服活性氟喹诺酮类抗生素,它对广泛的革兰氏阳性细菌、革兰氏阴性细菌(包括厌氧菌)及非典型病原体都显示出抗菌活性。该化合物主要用于研究呼吸道感染和尿路感染。
T38458 Faropenem

Faropenem, a highly efficacious and orally bioavailable beta-lactam antibiotic, exhibits an extensive range of in vitro antimicrobial activity against diverse gram-positive and -negative aerobes and anaerobes. Notably, Faropenem possesses inherent resistance to hydrolysis by virtually all beta-lactamases, including extended-spectrum beta-lactamases and AmpC beta-lactamases. Moreover, Faropenem has been developed as an oral prodrug, namely faropenem medoxomil, for the investigation of respiratory...
T75287 Sitafloxacin monohydrate

Sitafloxacin monohydrate (DU6859a) 是一种具有广谱的抗菌活性,并对多种革兰氏阳性和革兰氏阴性细菌(包括厌氧菌)以及非典型病原体有效的口服活性氟喹诺酮类抗生素。它主要用于研究呼吸道感染和尿路感染。
T60417 Fenspiride

Fenspiride 是 H1-组胺受体的拮抗剂。 Fenspiride 是一种具有口服活性的非甾体类抗炎药,可用于治疗呼吸道感染和中耳炎。 Fenspiride 抑制磷酸二酯酶 4 和磷酸二酯酶 3 的活性,-logIC50 值分别为 4.16+/-0.09 和 3.44+/-0.12。 磷酸二酯酶 5 活性也受到抑制,-logIC50 值约为 3.8。

化合物

SulfadiMethoxine sodium
Cat.No: T8133
Synonym:
Target: Anti-infection, Antibacterial, Antibiotic
Sulfadimethoxine
Cat.No: T1078
Synonym: Sulphadimethoxine,磺胺二甲氧嗪
Target: Antibacterial, Antibiotic
Balofloxacin
Cat.No: T0116
Synonym:
Target: DNA gyrase, Antibacterial, Antibiotic
Cefaclor monohydrate
Cat.No: T1495
Synonym: Cefaclor,头孢克洛一水物,头孢克洛一水合物,Cefaclorum,Cefachlor
Target: Antibacterial, Antibiotic
Cefaclor
Cat.No: T6436
Synonym: Panoral,Kefral,Cefaclorum,头孢克洛
Target: Others, Antibacterial, Antibiotic
Sulfogaiacol
Cat.No: T0284
Synonym: guaiacolsulfonate,愈创木酚磺酸钾
Target: Others, Antibacterial
Temafloxacin
Cat.No: T19794
Synonym: 替马沙星,Omniflox
Target: Antibiotic
Cefathiamidine
Cat.No: T8134
Synonym:
Target: Antibacterial, Antibiotic
Cefetamet Hydrochloride
Cat.No: T26974
Synonym: Cefetamet HCl,Cefetamet
Target:
Cefonicid (free base)
Cat.No: T68999
Synonym:
Target:
Cefonicid monosodium
Cat.No: T68817
Synonym:
Target:
Thiamphenicol glycinate hydrochloride
Cat.No: T72093
Synonym: 甲砜霉素甘氨酸酯盐酸盐
Target:
Cefetamet
Cat.No: T75274
Synonym:
Target:
Lomefloxacin (aspartate)
Cat.No: T63214
Synonym:
Target:
Dehydroandrographolide succinate potassium sodium salt
Cat.No: T40971
Synonym:
Target:
Lascufloxacin
Cat.No: T11819
Synonym: 拉库沙星,KRP-AM1977X
Target: Others
Sitafloxacin hydrochloride
Cat.No: T75286
Synonym:
Target:
Faropenem
Cat.No: T38458
Synonym:
Target:
Sitafloxacin monohydrate
Cat.No: T75287
Synonym:
Target:
Fenspiride
Cat.No: T60417
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T1134 Clofoctol

叔辛酚氯,氯福克酚

Antibacterial; Antibiotic Microbiology/Virology
Clofoctol 是一种抗生素,,可研究革兰氏阳性菌感染。它仅对革兰氏阳性菌起作用, 可渗透入人类肺组织。
T6567 Levofloxacin

Levaquin,Cravit,Tavanic,Fluoroquinolone,左氧氟沙星,(-)-Ofloxacin

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Levofloxacin (Fluoroquinolone) 是合成的氟喹诺酮类抗生素,有抑制细菌DNA 旋转酶的超螺旋活性的作用,能阻止DNA 复制。
TN5284 Sodium Houttuyfonate

Houttuynin sodium bisulfite,新鱼腥草素钠

NF-κB; Antibacterial; Antifungal Microbiology/Virology; NF-κB
Sodium Houttuyfonate (Houttuynin sodium bisulfite) 是亚硫酸氢钠与鱼腥草结合而成的活性化合物,具有抗真菌、抗菌、抗炎和心血管保护活性,主要用于治疗化脓性皮肤感染、呼吸道感染,包括老年患者的肺炎和慢性支气管炎。

天然产物

Clofoctol
Cat.No: T1134
Synonym: 叔辛酚氯,氯福克酚
Target: Antibacterial, Antibiotic
Levofloxacin
Cat.No: T6567
Synonym: Levaquin,Cravit,Tavanic,Fluoroquinolone,左氧氟沙星,(-)-Ofloxacin
Target: Topoisomerase, Antibacterial, Antibiotic
Sodium Houttuyfonate
Cat.No: TN5284
Synonym: Houttuynin sodium bisulfite,新鱼腥草素钠
Target: NF-κB, Antibacterial, Antifungal
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