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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T0946 Mepivacaine hydrochloride

Mepivacaine HCl,盐酸甲哌卡因

Sodium Channel Membrane transporter/Ion channel
Mepivacaine hydrochloride (Mepivacaine HCl) 是具有局部麻醉特性的酰胺衍生物。Mepivacaine hydrochloride 与神经元细胞膜上特定的电压门控钠离子通道结合,抑制钠离子内流和膜去极化。
T11318 Dopexamine hydrochloride

盐酸多培沙明,FPL60278AR

Adrenergic Receptor GPCR/G Protein; Neuroscience
Dopexamine hydrochloride (FPL60278AR) 是β2肾上腺素能受体激动剂。
T0914 Metacetamol

酰胺苯酚,3-Acetamidophenol

Others Others
Metacetamol (3-Acetamidophenol) 是对乙酰氨基酚的衍生物,为其无毒区域异构体,是一种非处方镇痛剂和解热剂,也可用作有机合成中间体。
T0372 Gabexate mesylate

甲磺酸加贝酯,FOY

Factor Xa; Serine Protease; Proteasome Metabolism; Proteases/Proteasome; Ubiquitination
Gabexate mesylate (FOY) 是一种非抗原的类胰蛋白酶丝氨酸蛋白酶抑制剂。
T27351 Fostedil

KB-944,KB944,A 53986,KB 944,A-53986,BRN 3626546

Fostedil is a calcium channel antagonist. KB-944 increased regional segment function in normal and ischemic regions and maintained distal coronary artery perfusion pressure, coronary flow and transmural regional myocardial blood flow during partial corona
TP1488 Proadrenomedullin (45-92), human

Proadrenomedullin (45-92), human, a mid-regional fragment of proadrenomedullin (MR-proADM), comprises amino acids 45–92 of pre-proADM.
T78458 IR 813 tosylate

IR 813 tosylate, 一近红外(NIR)荧光染料(λex=815 nm,λem=840 nm),适用于小鼠局部淋巴结的可视化。
T35858 Adrenomedullin (22-52) (human) (trifluoroacetate salt)

Adrenomedullin (22-52) is a C-terminal fragment of adrenomedullin (1-52) . In vitro, adrenomedullin (22-52) reduces basal corticosterone production in a mixture of rat adrenocortical and adrenomedulllary cells. It also reverses increases in ACTH-stimulated corticosterone production induced by adrenomedullin (1-52). Adrenomedulin (22-52) (0.5 and 5 μg/kg/min) has no effect on basal regional cerebral blood flow but reverses increases in regional cerebral blood flow induced by rat adrenomedullin in...
T62509 Antitumor agent-74

Antitumor agent-74 是一种喹唑啉衍生物,是一种抗肿瘤剂。Antitumor agent-74 与区域同分异构体 Antitumor agent-75 (compound 14 da) (mriBIQ 13da/14da) 联合使用表现出更强的肿瘤抑制效果。其中 mriBIQ 13da/14da 能够抑制 DNA 合成,将细胞周期阻滞在 S 期,并诱导线粒体凋亡。
T81400 Pritumumab

Pritumumab是一种自然源的人类IgG1kappa单克隆抗体,其最初源于一位宫颈癌患者的区域淋巴结分离得到。该单抗特异性地识别波形蛋白,该蛋白在多种恶性肿瘤细胞表面展现。Pritumumab在胶质母细胞瘤的科研应用中具有潜在价值。
T29922 Aluminum phthalocyanine disulfonate disodium

AlPcS2,AlPcS(2a),Disulfonated aluminum phthalocyanine,ClAlPcS2. Clalpcs,AlS2Pc

Aluminum phthalocyanine disulfonate sodium, also known as AlPcS2 disodium or AlS2Pc or AlPcS(2a), is a potent photosensitizer, and is potentially useful in cancer sonodynamic therapy and cancer photodynamic therapy. Aluminum phthalocyanine disulfonate is
T29890 AlPcS4

Aluminum phthalocyanine tetrasulfonate tetrasodium,Chloroaluminum tetrasulfophthalocyanine

AlPcS4 , also known as aluminum phthalocyanine tetrasulfonate Chloroaluminum tetrasulfophthalocyanine; or AlS4Pc, AlPcS4(a), is a potent photosensitizer, and is potentially useful in cancer sonodynamic therapy and cancer photodynamic therapy. Aluminum pht

化合物

Mepivacaine hydrochloride
Cat.No: T0946
Synonym: Mepivacaine HCl,盐酸甲哌卡因
Target: Sodium Channel
Dopexamine hydrochloride
Cat.No: T11318
Synonym: 盐酸多培沙明,FPL60278AR
Target: Adrenergic Receptor
Metacetamol
Cat.No: T0914
Synonym: 酰胺苯酚,3-Acetamidophenol
Target: Others
Gabexate mesylate
Cat.No: T0372
Synonym: 甲磺酸加贝酯,FOY
Target: Factor Xa, Serine Protease, Proteasome
Fostedil
Cat.No: T27351
Synonym: KB-944,KB944,A 53986,KB 944,A-53986,BRN 3626546
Target:
Proadrenomedullin (45-92), human
Cat.No: TP1488
Synonym:
Target:
IR 813 tosylate
Cat.No: T78458
Synonym:
Target:
Adrenomedullin (22-52) (human) (trifluoroacetate salt)
Cat.No: T35858
Synonym:
Target:
Antitumor agent-74
Cat.No: T62509
Synonym:
Target:
Pritumumab
Cat.No: T81400
Synonym:
Target:
Aluminum phthalocyanine disulfonate disodium
Cat.No: T29922
Synonym: AlPcS2,AlPcS(2a),Disulfonated aluminum phthalocyanine,ClAlPcS2. Clalpcs,AlS2Pc
Target:
AlPcS4
Cat.No: T29890
Synonym: Aluminum phthalocyanine tetrasulfonate tetrasodium,Chloroaluminum tetrasulfophthalocyanine
Target:
Cat. No. Product Name Target Signaling Pathways
T6S2227 Spinosin

斯皮诺素,Flavoayamenin

Others Others
Spinosin (Flavoayamenin) 是一种具有神经保护作用的 C-糖苷类黄酮,从 Zizyphus jujube 种子分离得到,能够激活 Nrf2/HO-1 通路,并抑制 Aβ1-42的产生和聚合。

天然产物

Spinosin
Cat.No: T6S2227
Synonym: 斯皮诺素,Flavoayamenin
Target: Others
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