9
2
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T20720 |
Norethisterone enanthate
NSC 9564,Norethindrone enanthate,LG-202,LG202,NSC9564,LG 202,炔诺酮庚酸酯,NSC-9564 |
Estrogen/progestogen Receptor | Endocrinology/Hormones |
Norethisterone enanthate (NSC-9564) 是一种口服有效的长效的孕激素。 | |||
T1490 |
Gestodene
SHB 331,WL 70,孕二烯酮 |
Estrogen/progestogen Receptor; Progesterone Receptor | Endocrinology/Hormones; Others |
Gestodene (WL 70) 是一种孕激素类避孕药。 | |||
T3036 |
Dydrogesterone
|
Progesterone Receptor | Others |
Dydrogesterone 是一种口服有效的孕激素,可作用于孕酮缺乏相关疾病。 | |||
T0870 |
Altrenogest
R2267,RU2267,Allyltrenbolone,A35957,烯丙孕素 |
Estrogen/progestogen Receptor; Progesterone Receptor | Endocrinology/Hormones; Others |
Altrenogest (Allyltrenbolone) 是一种结构与trenbolone 相关的孕激素,能作用于孕激素受体。 | |||
T2577 |
Dienogest
地诺孕素,STS 557 |
Apoptosis; Estrogen/progestogen Receptor; Progesterone Receptor; Autophagy | Apoptosis; Autophagy; Endocrinology/Hormones; Others |
Dienogest (STS 557) 是一种孕酮受体激动剂,作用于子宫内膜异位,有口服的子宫内膜活性。 | |||
T0272 |
Nilutamide
尼鲁米特,RU23908 |
Androgen Receptor | Endocrinology/Hormones |
Nilutamide (RU23908) 是一种非甾体抗雄激素药物,有用于转移性前列腺癌的潜力。 | |||
T20755 |
Trimegestone
RU27987,RU-27987,RU 27987 |
||
Trimegestone, a highly effective oral progestogen, is used for endometrial protection, all doses inducing secretory endometrial transformation. | |||
T25429 |
Flumedroxone acetate
WG 537,NSC 52412,NSC-52412,NSC52412,Leomigran |
||
Flumedroxone acetate is a progestogen medication which is or has been used as an antimigraine. | |||
T25304 |
Demegestone
R-2453,Lutionex,R 2453,RU 2453,R2453 |
||
Demegestone is a progestin, or a synthetic progestogen, and hence is a progesterone receptor agonist, the biological target of progestogens like progesterone. It has no androgenic activity. Previously used to treat luteal insufficiency. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0301 |
Ethisterone
炔孕酮,17α-Ethynyltestosterone,Pregneninolone |
Estrogen Receptor/ERR; Estrogen/progestogen Receptor | Endocrinology/Hormones |
Ethisterone (17α-Ethynyltestosterone) 是一种口服活性类固醇避孕药,是一种合成类固醇雌激素。据报道,它具有雄激素活性,用于妇科疾病的研究。 | |||
T1284 |
Megestrol acetate
SC10363,醋酸甲地孕酮,BDH1298 |
Glucocorticoid Receptor; Estrogen/progestogen Receptor; Progesterone Receptor; HIV Protease; Autophagy | Autophagy; Endocrinology/Hormones; Microbiology/Virology; Others; Proteases/Proteasome |
Megestrol acetate (BDH1298) 是具有口服活性的合成孕激素。它还具有抗雄激素特性,可用于治疗厌食症和恶病质。 |