3
1
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T13231L |
Trovafloxacin mesylate
|
Others; DNA/RNA Synthesis; Topoisomerase; Antibacterial | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others |
Trovafloxacin是一种广谱氟喹诺酮类抗生素,可阻断 DNA 促旋酶 (DNA gyrase) 和拓扑异构酶 IV (topoisomerase IV) 的活性,也是一种有效的特异性 pannexin 1 通道抑制剂 (PANX1, IC50 = 4 μM)。 | |||
T13231 | Trovafloxacin | DNA gyrase; Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Trovafloxacin 是广谱喹诺酮类抗生素,对革兰氏阳性,革兰氏阴性和厌氧菌有活性。它可阻断 DNA 促旋酶 和拓扑异构酶 IV 的活性。它也是口服活性的 Pannexin 1通道选择性抑制剂,对 PANX1内向电流的 IC50为 4 μM。 | |||
T30981 |
Clometocillin
Penicilline 356 |
||
Clometocillin is a penicillin that can active penicillin to pen-I or pen-R pneumococci. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN1407 |
Artocarpin
桂木黄素,2',4',5-三羟基-7-甲氧基-6-(3-甲基-1-丁烯基)-3-(3-甲基-2-丁烯基)黄酮 |
IL Receptor; TNF; COX | Apoptosis; Immunology/Inflammation; Neuroscience |
Artocarpin has anti- bactericidal effect, can reduce the viability of pneumococci by a factor of >1000, without obvious harm to lung epithelial cells. |