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Search Results for " pneumococci "

3

抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T13231L Trovafloxacin mesylate

Others; DNA/RNA Synthesis; Topoisomerase; Antibacterial Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Trovafloxacin是一种广谱氟喹诺酮类抗生素,可阻断 DNA 促旋酶 (DNA gyrase) 和拓扑异构酶 IV (topoisomerase IV) 的活性,也是一种有效的特异性 pannexin 1 通道抑制剂 (PANX1, IC50 = 4 μM)。
T13231 Trovafloxacin

DNA gyrase; Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Trovafloxacin 是广谱喹诺酮类抗生素,对革兰氏阳性,革兰氏阴性和厌氧菌有活性。它可阻断 DNA 促旋酶 和拓扑异构酶 IV 的活性。它也是口服活性的 Pannexin 1通道选择性抑制剂,对 PANX1内向电流的 IC50为 4 μM。
T30981 Clometocillin

Penicilline 356

Clometocillin is a penicillin that can active penicillin to pen-I or pen-R pneumococci.

化合物

Trovafloxacin mesylate
Cat.No: T13231L
Synonym:
Target: Others, DNA/RNA Synthesis, Topoisomerase, Antibacterial
Trovafloxacin
Cat.No: T13231
Synonym:
Target: DNA gyrase, Topoisomerase, Antibacterial, Antibiotic
Clometocillin
Cat.No: T30981
Synonym: Penicilline 356
Target:
Cat. No. Product Name Target Signaling Pathways
TN1407 Artocarpin

桂木黄素,2',4',5-三羟基-7-甲氧基-6-(3-甲基-1-丁烯基)-3-(3-甲基-2-丁烯基)黄酮

IL Receptor; TNF; COX Apoptosis; Immunology/Inflammation; Neuroscience
Artocarpin has anti- bactericidal effect, can reduce the viability of pneumococci by a factor of >1000, without obvious harm to lung epithelial cells.

天然产物

Artocarpin
Cat.No: TN1407
Synonym: 桂木黄素,2',4',5-三羟基-7-甲氧基-6-(3-甲基-1-丁烯基)-3-(3-甲基-2-丁烯基)黄酮
Target: IL Receptor, TNF, COX
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