Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T34189 |
PTZ-256
phenothiazine derivative,PTZ256 |
||
PTZ-256 is a phenothiazine derivative with chemical name: 3-(10H-phenothiazin-10-yl)propane-1-amine. PTZ-256 has molecule weight 256, therefore, we call it as PTZ-256. | |||
T1090 |
Perphenazine
Perphenazin,Etaperazine,Trilafon,奋乃静 |
CaMK; Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Perphenazine (Trilafon) 是吩噻嗪衍生物和多巴胺拮抗剂,具有止吐和抗精神病特性。它能够抑制5-HT2A 受体,α1A 肾上腺素能受体,多巴胺D2、D3、D2L 受体,以及组胺H1受体,对应的Ki 值分别为5.6、10、0.765、0.13、3.4 和 8 nM。 | |||
T23843L |
Butaperazine maleate
Tyrylen,Repoise maleate |
||
Butaperazine maleate, a phenothiazine derivative, is an antipsychotic. | |||
T40854 |
Imiclopazine
|
||
Imiclopazine is a phenothiazine derivative with good sedative, analgesic, antiaggressive and antiemetic effects. | |||
T23949 |
Dacemazine hydrochloride
Ahistan HCl,Dacemazine HCl,Histantine HCl,UNII-DK78VKA001 |
||
Dacemazine is a phenothiazine derivative that acts as a histamine antagonist at the H1 subtype. It was also assessed as a possible anticancer drug. | |||
T28282 |
Oxypertine
Win-18501,Forit,Win18501,Win 18501 |
||
Oxypertine is an indole-derivative antipsychotic with general properties similar to those of the chlorpromazine and phenothiazine. Oxypertine is used as a treatment for various psychoses including mania, schizophrenia, disturbed behaviour, and severe anx | |||
TMIH-0454 |
Prochlorperazine-d8
|
||
Prochlorperazine-d8 是 Prochlorperazine 的氘代化合物。Prochlorperazine 的 CAS 号为 58-38-8。Prochlorperazine 是一种抗精神病药phenothiazine衍生物。 | |||
T68133 |
quisultazine
|
||
Quisultazine 是一种非中枢作用的吩噻嗪衍生物,可归类为非抗H2抗分泌剂。 | |||
T61915 |
Thiethylperazine
|
||
Thiethylperazine 是一种吩噻嗪衍生物。Thiethylperazine 是具有口服活性的组胺H1受体和多巴胺D2受体拮抗剂。Thiethylperazine 也是选择性的ABCC1激活剂,可减少小鼠中的淀粉样 β (Aβ) 负荷。Thiethylperazine 具有抗精神病,止吐和抗菌作用。 |