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抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T26778 Besipirdine

HP 749 free base,P-867493,P867493,HP 749,HP749,P 867493

Sodium Channel; Adrenergic Receptor GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Besipirdine (HP 749 free base)是一种非受体依赖性拟胆碱化合物,具有α-肾上腺素能活性和心血管活性。Besipirdine 抑制电压依赖性钠钾通道,抑制生物胺的摄取。Besipirdine 可减少大鼠的时间表诱导的烦渴,增强中枢神经系统中的胆碱能和肾上腺素能神经传递。
T26778L Besipirdine hydrochloride

HP 749 hydrochloride,Besipirdine hydrochloride(119257-34-0 Free base)

Adrenergic Receptor GPCR/G Protein; Neuroscience
Besipirdine hydrochloride 是一种非受体依赖性拟胆碱化合物,具有α-肾上腺素能活性和心血管活性。Besipirdine hydrochloride 抑制电压依赖性钠钾通道,抑制生物胺的摄取。Besipirdine hydrochloride 可减少大鼠的时间表诱导的烦渴,增强中枢神经系统中的胆碱能和肾上腺素能神经传递。
T68811 Trimetaphan camsilate

Trimetaphan camsilate is a drug that counteracts cholinergic transmission at the ganglion type of nicotinic receptors of the autonomic ganglia and therefore blocks both the sympathetic nervous system and the parasympathetic nervous system. It acts as a non-depolarizing competitive antagonist at the nicotinic acetylcholine receptor, is short-acting, and is given intravenously.
TP2058 Catestatin

Non-competitive nicotinic cholinergic antagonist; selectively inhibits nicotinic-stimulated catecholamine secretion from chromaffin cells and noradrenergic neurons (IC50 ~ 200 nM). Blocks nicotinic-induced cationic signaling (IC50 ~ 200 - 250 nM) and inhi

化合物

Besipirdine
Cat.No: T26778
Synonym: HP 749 free base,P-867493,P867493,HP 749,HP749,P 867493
Target: Sodium Channel, Adrenergic Receptor
Besipirdine hydrochloride
Cat.No: T26778L
Synonym: HP 749 hydrochloride,Besipirdine hydrochloride(119257-34-0 Free base)
Target: Adrenergic Receptor
Trimetaphan camsilate
Cat.No: T68811
Synonym:
Target:
Catestatin
Cat.No: TP2058
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T3026 (-)-Huperzine A

HupA,石杉碱,Huperzine A,石杉碱甲

Apoptosis; AChR; AChE; iGluR Apoptosis; Membrane transporter/Ion channel; Neuroscience
(-)-Huperzine A (HupA) 是从中国梅花苔中分离得到的一种生物碱,具有神经保护活性。它是高特异性可逆的,具有血脑屏障渗透性的一种乙酰胆碱酯酶抑制剂, 其IC50值为 82 nM。 它也是 N-甲基-D-天冬氨酸受体的非竞争性拮抗剂,可研究神经退行性疾病,如阿尔茨海默病。

天然产物

(-)-Huperzine A
Cat.No: T3026
Synonym: HupA,石杉碱,Huperzine A,石杉碱甲
Target: Apoptosis, AChR, AChE, iGluR
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