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33

抑制剂 & 化合物

6

天然产物

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Cat. No. Product Name Target Signaling Pathways
T3563 Lvguidingan

Others Others
Lvguidingan 是一种抗惊厥药。
T0992 Carbenoxolone disodium

Biogastrone,Duogastrone,甘珀酸钠,Bioral

Gap Junction Protein Cytoskeletal Signaling
Carbenoxolone disodium (Duogastrone) 是甘草酸的活性代谢物和人11β-HSD 和细菌3α, 20β-HSD 的抑制剂。它是一种缝隙连接的解耦剂,可抑制牛痘病毒生长,用于消化性、食道和口腔溃疡和炎症的相关研究。
T0370 Pheniramine maleate

Daneral,Inhiston,Trimetose,马来酸非尼拉敏

5-HT Receptor; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Pheniramine maleate (Trimetose) 是一种具有抗组胺和血管扩张特性的烷基胺衍生物,可与组胺 H1 受体结合,从而抑制磷脂酶 A2 和内皮源性松弛因子一氧化氮的产生。
T30248 AZD 3043

AZD-3043,THRX 918661,AZD3043

AZD 3043 is a propofol derivative which acts as a sedative-hypnotic agent.
T0227 Bromisoval

2-Bromo-N-carbamoyl-3-methylbutanamide,Isobromyl,溴米那,BRN 1773255,Bromovalerylurea,溴米索伐,Bromaral

Others Others
Bromisoval (Isobromyl) 具有抗炎活性。
T31724 Etoxybamide

Others Others
Etoxybamide 是镇静剂(催眠药)的候选药物。
T14314 Apronal

Apronalide,Allylisopropylacetylurea,丙戊酰脲

Others Others
Apronal (Apronalide) 具有催眠和镇静作用,可用于神经精神疾病的相关研究。
T24451 Mepyramine

NSC-13136,NSC13136,NSC 13136

Mepyramine is a histamine H1 antagonist. It has mild hypnotic properties and some local anesthetic action and is used for allergies both parenterally and locally.
T19991 N-desmethylmirtazapine

米氮平杂质D,N-Demethylmirtazapine,Normirtazapine,ORG3838,ORG 3838,J1.061.658A,ORG-3838

Others Others
N-desmethylmirtazapine (J1.061.658A) 是mirtazapine 的代谢物。它也常用作抗焦虑药、催眠药、止吐药和食欲兴奋剂。
T10002 (E)-Crotylbarbital

Kalypnon

Others Others
(E)-Crotylbarbital (Kalypnon) 是Crotylbarbital 的异构体,是一种巴比妥酸衍生物,具有镇静、催眠和抗惊厥的作用。(E)-Crotylbarbital 可用于促进精神安定和睡眠的研究。
T3282 Alimemazine hemitartrate

Alimemazine Tartrate,Methylpromazine Tartrate,酒石酸异丁嗪,Trimeprazine tartrate,Trimeprazine hemitartrate

Others Others
Alimemazine hemitartrate (Trimeprazine hemitartrate) 是血凝素 (HA)-受体的拮抗剂,也是一种吩噻嗪衍生物,常用作止痒剂。
TQ0023 Lorediplon

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Lorediplon 是一种新型催眠药物,作为 GABAA 受体调节剂,在 α1 亚基上具有差异活性,与促进睡眠有关。
T1232 Mepyramine maleate

马来酸吡纳明,Pyrilamine maleate,吡拉明马来酸盐

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Mepyramine maleate (Pyrilamine maleate) 是一种组胺 H1 拮抗剂,对 H1、H2 和 H3 受体的 Kd 值分别为 0.8、5200 和大于 3000 nM,对 H1 受体的 pKd 值为 9.4。它是感冒药的常见成分,具有温和的催眠特性和局部麻醉作用,可用于胃肠外和局部过敏。
T21428 Mianserin

Lantanon,Lumin,Norval,Lerivon,Depnon

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Mianserin 是H1受体反向激动剂,是四环抗抑郁药(TeCA)治疗家族中的一种精神活性化合物,具有抗抑郁、抗焦虑、止吐、促氧、催眠和抗组胺作用,可作为去甲肾上腺素和特定的血清素联合用药能治疗抑郁症。
T0901 Chlorobutanol

Chlortran,Chloretone,YM-57158,三氯叔丁醇,Chlorbutol,Chloreton

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Chlorobutanol (Chlortran) 是一种药物防腐剂,对多种革兰氏阳性和革兰氏阴性细菌以及几种霉菌孢子和真菌具有抗性。它广泛用于食品和化妆品工业,有促进安定、睡眠的作用。
T26948 Capuride

NSC-27178,NSC27178,NSC-27690,NSC 27178,NSC27690

Capuride is a sedative with hypnotic properties and possible anticonvulsant activity.
T19318 Ethyl dirazepate

Others Others
Ethyl dirazepate has anxiolytic and hypnotic and possibly other characteristic benzodiazepine properties,is a drug which is a benzodiazepine derivative.
T26061 Reposal

WT-161,Reposamal,Reposal novo,WT161,WT 161

Reposal is a barbiturate derivative invented in the 1960s in Denmark. It has hypnotic, sedative, and anticonvulsant properties, and was used primarily for the therapy of insomnia.
T24138 Hexapropymate

Lunamin,Esapropimato,L-2103,L2103,L 2103

Hexapropymate is a hypnotic drug.
T13682 Epipregnanolone

Others Others
Epipregnanolone is an endogenous neurosteroid with hypnotic and sedative effects.
T29546 Acecarbromal

Paxerel,Absin,Darilonl,Adityl

Acecarbromal is a central nervous system drug with potential hypnotic effects.
T34771 Taglutimide

Taglutimide is a sedative-hypnotic derivative of glutarimide.
T27007 Chlormethiazole edisylate

Clomethiazole ethanedisulfonate,Clomethiazole edisylate,Heminevrin,Hemithiamine,Distraneurin

Chlormethiazole edisylate is a positive allosteric modulator of the GABAA receptor. Chlormethiazole edisylate is a sedative and hypnotic.
T27543 HIE-124

HIE-124 is a central cervous system active anticonvulsant and ultra-short acting hypnotic.
T24201 JM-1232

JM 1232,MR 04A3,MR-04A3,MR04A3

JM-1232 is a sedative and hypnotic drug being researched as a potential anesthetic.
T28378 PF-0713

PF 0713,PF713

PF 0713, a GABAA receptor agonist, is used as an intravenous sedative-hypnotic for general anaesthesia, ICU sedation, procedural sedation, chemotherapy.
T30945 Cinolazepam

Gerodorm,OX-373

Cinolazepam is a benzodiazepine derivative drug.It has a powerful sedative effect, so it is mainly used as a hypnotic.
T40205 Posovolone

Co 134444

Posovolone (Co 134444), an orally active neuroactive steroid with sedative-hypnotic properties, exhibits anticonvulsant and anxiolytic-like activities, alongside ataxic effects.
T23604 Acebrochol

Acebrochol is a neuroactive steroid. It may act as a sedative and hypnotic, by the mechanism of altering ligand-gated ion channels and cell surface receptors.
T68933 Gaboxadol hydrobromide

Gaboxadol hydrobromide is a GABA agonist. It is an inhibitor of GABA uptake systems. Gaboxadol can also be a non-opioid analgesic and a novel type of hypnotic.
T68111 nabitan

Nabitan 是δ -9-四氢大麻酚的类似物,根据其在动物中的镇静、催眠和镇痛特性而被选择。
T69434 Methapyrilene fumarate

Methapyrilene fumarate is a histamine H1 antagonist with sedative action used as a hypnotic and in allergies. It is a hepatocarcinogen in sufficiently high doses, inducing mutations through an indirect genotoxic mechanism; e.g., via an oxidative mechanism or interaction with chromosomal proteins.
T78111 NCS-382 sodium

GABA Receptor Membrane transporter/Ion channel; Neuroscience
NCS-382 (sodium) 为一种高效GABA受体拮抗剂,具备抗镇静及抗催眠特性,适用于神经系统疾病研究。

化合物

Lvguidingan
Cat.No: T3563
Synonym:
Target: Others
Carbenoxolone disodium
Cat.No: T0992
Synonym: Biogastrone,Duogastrone,甘珀酸钠,Bioral
Target: Gap Junction Protein
Pheniramine maleate
Cat.No: T0370
Synonym: Daneral,Inhiston,Trimetose,马来酸非尼拉敏
Target: 5-HT Receptor, Histamine Receptor
AZD 3043
Cat.No: T30248
Synonym: AZD-3043,THRX 918661,AZD3043
Target:
Bromisoval
Cat.No: T0227
Synonym: 2-Bromo-N-carbamoyl-3-methylbutanamide,Isobromyl,溴米那,BRN 1773255,Bromovalerylurea,溴米索伐,Bromaral
Target: Others
Etoxybamide
Cat.No: T31724
Synonym:
Target: Others
Apronal
Cat.No: T14314
Synonym: Apronalide,Allylisopropylacetylurea,丙戊酰脲
Target: Others
Mepyramine
Cat.No: T24451
Synonym: NSC-13136,NSC13136,NSC 13136
Target:
N-desmethylmirtazapine
Cat.No: T19991
Synonym: 米氮平杂质D,N-Demethylmirtazapine,Normirtazapine,ORG3838,ORG 3838,J1.061.658A,ORG-3838
Target: Others
(E)-Crotylbarbital
Cat.No: T10002
Synonym: Kalypnon
Target: Others
Alimemazine hemitartrate
Cat.No: T3282
Synonym: Alimemazine Tartrate,Methylpromazine Tartrate,酒石酸异丁嗪,Trimeprazine tartrate,Trimeprazine hemitartrate
Target: Others
Lorediplon
Cat.No: TQ0023
Synonym:
Target: GABA Receptor
Mepyramine maleate
Cat.No: T1232
Synonym: 马来酸吡纳明,Pyrilamine maleate,吡拉明马来酸盐
Target: Histamine Receptor
Mianserin
Cat.No: T21428
Synonym: Lantanon,Lumin,Norval,Lerivon,Depnon
Target: Histamine Receptor
Chlorobutanol
Cat.No: T0901
Synonym: Chlortran,Chloretone,YM-57158,三氯叔丁醇,Chlorbutol,Chloreton
Target: Antibacterial, Antibiotic, Antifungal
Capuride
Cat.No: T26948
Synonym: NSC-27178,NSC27178,NSC-27690,NSC 27178,NSC27690
Target:
Ethyl dirazepate
Cat.No: T19318
Synonym:
Target: Others
Reposal
Cat.No: T26061
Synonym: WT-161,Reposamal,Reposal novo,WT161,WT 161
Target:
Hexapropymate
Cat.No: T24138
Synonym: Lunamin,Esapropimato,L-2103,L2103,L 2103
Target:
Epipregnanolone
Cat.No: T13682
Synonym:
Target: Others
Acecarbromal
Cat.No: T29546
Synonym: Paxerel,Absin,Darilonl,Adityl
Target:
Taglutimide
Cat.No: T34771
Synonym:
Target:
Chlormethiazole edisylate
Cat.No: T27007
Synonym: Clomethiazole ethanedisulfonate,Clomethiazole edisylate,Heminevrin,Hemithiamine,Distraneurin
Target:
HIE-124
Cat.No: T27543
Synonym:
Target:
JM-1232
Cat.No: T24201
Synonym: JM 1232,MR 04A3,MR-04A3,MR04A3
Target:
PF-0713
Cat.No: T28378
Synonym: PF 0713,PF713
Target:
Cinolazepam
Cat.No: T30945
Synonym: Gerodorm,OX-373
Target:
Posovolone
Cat.No: T40205
Synonym: Co 134444
Target:
Acebrochol
Cat.No: T23604
Synonym:
Target:
Gaboxadol hydrobromide
Cat.No: T68933
Synonym:
Target:
nabitan
Cat.No: T68111
Synonym:
Target:
Methapyrilene fumarate
Cat.No: T69434
Synonym:
Target:
NCS-382 sodium
Cat.No: T78111
Synonym:
Target: GABA Receptor
Cat. No. Product Name Target Signaling Pathways
T37709 2,2,2-Trichloroethanol

Potassium Channel; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism
2,2,2-Trichloroethanol 是非经典的 K2P 通道 TREK-1和 TRAAK 的激动剂。
T4S0675 Polygalasaponin V

瓜子金皂苷V,瓜子金皂苷 V

Others Others
Polygalasaponin V 是一种三萜皂苷,分离自Polygala japonica 的地上部分。其中Polygala japonica 是民间的药用植物,在中国南方用作祛痰、抗菌、抗炎、抗抑郁药。
T7646 Alloepipregnanolone

Endogenous Metabolite Metabolism
Alloepipregnanolone 是具有促进安定和睡眠的孕酮,可干扰乙醇抗焦虑作用的快速耐受。
T8297 Gomisin N

Apoptosis Apoptosis
Gomisin N 是从五味子中分离得到的一种天然产物,有镇静和催眠生物活性。它具有用于治疗过敏和抑制癌症增殖和诱导细胞凋亡的潜力。
T0330 Diphenhydramine hydrochloride

盐酸苯海拉明,Diphenhydramine HCl,DPH

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Diphenhydramine hydrochloride (DPH) 是一种组胺 H1 拮抗剂,用作镇咳药和止吐药。它还用于治疗瘙痒和皮肤病、过敏反应、抗帕金森病、催眠药和普通感冒制剂的成分。
TN1812 Jujuboside B1

酸枣仁皂苷 B1

5-HT Receptor GPCR/G Protein; Neuroscience
Jujubosides have hypnotic effect on normal rats, may be influenced by circadian rhythm and the serotonergic system may involve in the hypnotic effect of jujubosides, jujubosides may be good source of lead compounds for novel hypnotics.

天然产物

2,2,2-Trichloroethanol
Cat.No: T37709
Synonym:
Target: Potassium Channel, Endogenous Metabolite
Polygalasaponin V
Cat.No: T4S0675
Synonym: 瓜子金皂苷V,瓜子金皂苷 V
Target: Others
Alloepipregnanolone
Cat.No: T7646
Synonym:
Target: Endogenous Metabolite
Gomisin N
Cat.No: T8297
Synonym:
Target: Apoptosis
Diphenhydramine hydrochloride
Cat.No: T0330
Synonym: 盐酸苯海拉明,Diphenhydramine HCl,DPH
Target: Histamine Receptor
Jujuboside B1
Cat.No: TN1812
Synonym: 酸枣仁皂苷 B1
Target: 5-HT Receptor
TargetMol Loading
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