8
3
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11785 |
KT203
|
MAGL | Metabolism |
KT203 是一种具有选择性和高效性的 α/β 水解酶结构域 6 (ABHD6) 抑制剂,具有潜在的抗病毒和抗炎活性,可用于研究肺炎。 | |||
T0372 |
Gabexate mesylate
甲磺酸加贝酯,FOY |
Factor Xa; Serine Protease; Proteasome | Metabolism; Proteases/Proteasome; Ubiquitination |
Gabexate mesylate (FOY) 是一种非抗原的类胰蛋白酶丝氨酸蛋白酶抑制剂。 | |||
T33731 |
N-Phthaloylglutamic acid
alpha-N-Phthaloylglutamic acid,N,N-Phthaloyl-L-glutamic acid,PhGA |
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N-Phthaloylglutamic acid is a hydrolytic metabolite of thalidomide. | |||
T24615 |
PF04677490
PF-04677490,PF 04677490 |
||
PF04677490 is an effective PDE1 inhibitor. PF04677490 efficaciously inhibits cAMP- and cGMP-hydrolytic activity in preparations from human myocardium at concentrations selective for PDE1. | |||
T35788 |
Orlistat Degradation Product (sodium salt)
|
||
Orlistat degradation product is a degradation product of the digestive lipase inhibitor orlistat . It is formed via hydrolytic and thermal degradation as well as digestion by human carboxyl ester lipase. | |||
T62861 |
ERAP2-IN-1
|
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ERAP2-IN-1 (compound 61) 是一种 ERAP2 的非竞争性抑制剂。ERAP2-IN-1 特异性抑制 ERAP2 肽水解活性,抑制 Arg-AMC 水解作用 (IC50: 27 μM) 和模型肽的水解活性 (IC50: 44 μM)。 | |||
T83932 |
Phenyl-glutarimide 4'-piperazine
|
||
Phenyl-glutarimide 4'-piperazine是一种具有piperazine功能化的cereblon配体,可用于PROTACDegrader的开发。该化合物可用于开发PG-PROTACs,与使用IMiD(immunomodulatory imide drug)类似物合成的PROTACs相比,展示出改善的水解稳定性和效力。 | |||
T83928 |
DA ZP1
|
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DA ZP1(diacetylated Zinpyr1)是一种荧光性的Zn(II)传感器(KdZn2+= 0.6 nM),可用于体外成像和分离胰腺β细胞及类似β细胞,并用于纯化源自干细胞的活体类似β细胞。该传感器亦可用于体内成像移植的岛细胞移植物和内源性小鼠岛细胞。在没有Zn(II)离子存在时,DA ZP1不发光,但其与Zn(II)的结合促进乙酰基的水解裂解,产生强烈的荧光信号。其激发和发射最大波长(λ)分别为490 nm和522 nm。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T41044 |
Naringinase
|
Glucosidase | Metabolism |
Naringinase 是一种在自然界中广泛存在的水解酶复合物,具有 α-L-鼠李糖苷酶和 β-D-葡萄糖苷酶的活性,主要用于糖苷的水解。 | |||
T2S1840 |
Rebaudioside D
莱苞迪苷D,瑞鲍迪甙D |
Others | Others |
Rebaudioside D 是一种苷类化合物,存在于甜菊叶中,可用作甜味剂。 | |||
T1591 |
Ancitabine hydrochloride
NSC 145668 HCl,盐酸环胞苷,Cyclocytidine hydrochloride,Cyclo-CMP hydrochloride,Cyclocytidine HCl,Cyclo-C |
Others; DNA/RNA Synthesis; Autophagy | Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Others |
Ancitabine hydrochloride (NSC 145668 HCl) 是一种天然的抗白血病药物。 |