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Cat. No. | Product Name | Target | Signaling Pathways |
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T9793 | Methyl Ergoline Acid | Others | Others |
Methyl Ergoline Acid 是一种麦角碱衍生物,可用作趋化因子受体配体。 | |||
T31663 |
Lysergamide, N-cycloheptyl-, maleate
Ergoline-8-beta-carboxamide, N-cycloheptyl-9,10-didehydro-6-methyl-, maleate |
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Lysergamide, N-cycloheptyl-, maleate 可用于生命科学领域的相关研究。其产品编号为 T31663,CAS号为 103070-86-6。 | |||
T31664 |
Lysergamide, N-cyclopropyl-, maleate
Ergoline-8-beta-carboxamide, N-cyclopropyl-9,10-didehydro-6-methyl-, maleate |
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Ergoline-8-beta-carboxamide, N-cyclopropyl-9,10-didehydro-6-methyl-, maleate is a bioactive chemical. | |||
T2226 |
Pergolide mesylate
甲磺酸培高利特,Pergolide mesylate salt,LY127809,Pergolide methanesulfonate |
Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Pergolide mesylate salt(LY127809) 是一种有效的,具有口服活性的多巴胺 D1和 D2受体激动剂,是一种 Ergoline 衍生物,可用于帕金森氏病和高泌乳素血症的研究。 | |||
T1132 |
Nicergoline
尼麦角林,Nicergolinum,Nimergoline |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Nicergoline (Nicergolinum) 是一种有效的,选择性的、具有口服活性的α1A-肾上腺素能受体拮抗剂,是一种溴烟碱酸的麦角林衍生物。它具有血管舒张作用,可以改善阿尔茨海默症小鼠的认知功能。 | |||
T4008 |
Metergoline
甲麦角林,Methergoline,Liserdol |
Dopamine Receptor; 5-HT Receptor; Sodium Channel | GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience |
Metergoline (Methergoline) 是多巴胺激动剂和血清素拮抗剂。它是 h5-HT7受体的高亲和力配体,Ki 为 16 nM。它还是可逆神经 Na+通道抑制剂,用于研究季节性情绪障碍、催乳激素调节。 | |||
T71707L |
Romergoline 2HCl
Romergoline 2HCl(107052-56-2 Free base),FCE 23884 2HCl |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Romergoline 2HCl 是一种 D1 激动剂和 D2 拮抗剂,可用于研究帕金森病。 | |||
T71707 |
Romergoline
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Romergoline 是一种新合成的麦角碱衍生物,具有独特的药理作用,在正常动物中表现出完全的多巴胺(DA)拮抗作用,而在“去神经”动物模型中表现出完全的DA 拮抗作用。 | |||
T68551 |
Cabergoline diphosphate
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Cabergoline diphosphate is a dopamine D2 receptor agonist used for prolactinoma treatment. Cabergoline permits rapid and effective hormonal and tumor control by normalizing prolactin-producing pituitary adenomas levels. | |||
T1132L |
Nicergoline tartrate
Adavin |
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Nicergoline tartrate is a bioactive chemical. | |||
T25247 |
Cianergoline
Cianergolinum |
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Cianergoline is a dopaminergic agonist. | |||
T11011 |
Dexpramipexole dihydrochloride
普拉克索杂质D,KNS-760704 dihydrochloride,R-(+)-Pramipexole dihydrochloride,右旋普拉克索二盐酸盐,(R)-Pramipexole dihydrochloride |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) 是一种神经保护剂,是一种弱的非麦角类多巴胺受体激动剂。 | |||
T25671L |
Lergotrile mesylate
LY83636,LY-83636,LY 83636 |
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Lergotrile mesylate, an ergoline derivative, suppresses prolactin in vivo and in vitro. | |||
T34432 |
RU 28306
RU-28306,RU28306 |
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RU 28306 is a racemic partial ergoline. | |||
TQ0175 |
Dexpramipexole
右旋普拉克索,R-(+)-Pramipexole,(R)-Pramipexole,KNS-760704 |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Dexpramipexole (KNS-760704, R-(+)-Pramipexole) is a neuroprotective agent and weak non-ergoline dopamine agonist. | |||
T25657 |
LEK 8841
LEK-8841,LEK8841 |
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LEK 8841 is an ergoline derivative that is a potential antipsychotic. | |||
T24003 |
Disulergine
CM 29717,CH 29717,CH 29-717 |
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Disulergine is a dopamine receptor agonist. It also prolactin release-inhibiting 8 alpha-amino-ergoline. | |||
T21340 | Pergolide | ||
Pergolide, an ergoline-based dopamine receptor agonist, is used for the treatment of Parkinson's disease, which is associated with low levels of the neurotransmitter dopamine in the brain. | |||
T68440 |
Epicriptine
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Epicriptine or beta-dihydroergocryptine is a dopamine agonist of the ergoline class. It constitutes one third of the mixture known as dihydroergocryptine, the other two thirds consisting of alpha-dihydroergocryptine. The alpha differs from the beta form only in the position of a single methyl group, which is a consequence of the biosynthesis in which the proteinogenic amino acid isoleucine is replaced by leucine. |
Cat. No. | Product Name | Target | Signaling Pathways |
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T14853 |
Cabergoline
FCE-21336,卡麦角林 |
Dopamine Receptor; 5-HT Receptor; Autophagy | Autophagy; GPCR/G Protein; Neuroscience |
Cabergoline (FCE-21336) 是一种麦角衍生的多巴胺 D2亚类受体激动剂,高亲和力作用于D2、D3和5-HT2B 受体,Ki 分别为 0.7、1.5 和 1.2。 |