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19

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T9793 Methyl Ergoline Acid

Others Others
Methyl Ergoline Acid 是一种麦角碱衍生物,可用作趋化因子受体配体。
T31663 Lysergamide, N-cycloheptyl-, maleate

Ergoline-8-beta-carboxamide, N-cycloheptyl-9,10-didehydro-6-methyl-, maleate

Lysergamide, N-cycloheptyl-, maleate 可用于生命科学领域的相关研究。其产品编号为 T31663,CAS号为 103070-86-6。
T31664 Lysergamide, N-cyclopropyl-, maleate

Ergoline-8-beta-carboxamide, N-cyclopropyl-9,10-didehydro-6-methyl-, maleate

Ergoline-8-beta-carboxamide, N-cyclopropyl-9,10-didehydro-6-methyl-, maleate is a bioactive chemical.
T2226 Pergolide mesylate

甲磺酸培高利特,Pergolide mesylate salt,LY127809,Pergolide methanesulfonate

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor GPCR/G Protein; Neuroscience
Pergolide mesylate salt(LY127809) 是一种有效的,具有口服活性的多巴胺 D1和 D2受体激动剂,是一种 Ergoline 衍生物,可用于帕金森氏病和高泌乳素血症的研究。
T1132 Nicergoline

尼麦角林,Nicergolinum,Nimergoline

Adrenergic Receptor GPCR/G Protein; Neuroscience
Nicergoline (Nicergolinum) 是一种有效的,选择性的、具有口服活性的α1A-肾上腺素能受体拮抗剂,是一种溴烟碱酸的麦角林衍生物。它具有血管舒张作用,可以改善阿尔茨海默症小鼠的认知功能。
T4008 Metergoline

甲麦角林,Methergoline,Liserdol

Dopamine Receptor; 5-HT Receptor; Sodium Channel GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Metergoline (Methergoline) 是多巴胺激动剂和血清素拮抗剂。它是 h5-HT7受体的高亲和力配体,Ki 为 16 nM。它还是可逆神经 Na+通道抑制剂,用于研究季节性情绪障碍、催乳激素调节。
T71707L Romergoline 2HCl

Romergoline 2HCl(107052-56-2 Free base),FCE 23884 2HCl

Dopamine Receptor GPCR/G Protein; Neuroscience
Romergoline 2HCl 是一种 D1 激动剂和 D2 拮抗剂,可用于研究帕金森病。
T71707 Romergoline

Romergoline 是一种新合成的麦角碱衍生物,具有独特的药理作用,在正常动物中表现出完全的多巴胺(DA)拮抗作用,而在“去神经”动物模型中表现出完全的DA 拮抗作用。
T68551 Cabergoline diphosphate

Cabergoline diphosphate is a dopamine D2 receptor agonist used for prolactinoma treatment. Cabergoline permits rapid and effective hormonal and tumor control by normalizing prolactin-producing pituitary adenomas levels.
T1132L Nicergoline tartrate

Adavin

Nicergoline tartrate is a bioactive chemical.
T25247 Cianergoline

Cianergolinum

Cianergoline is a dopaminergic agonist.
T11011 Dexpramipexole dihydrochloride

普拉克索杂质D,KNS-760704 dihydrochloride,R-(+)-Pramipexole dihydrochloride,右旋普拉克索二盐酸盐,(R)-Pramipexole dihydrochloride

Dopamine Receptor GPCR/G Protein; Neuroscience
Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) 是一种神经保护剂,是一种弱的非麦角类多巴胺受体激动剂。
T25671L Lergotrile mesylate

LY83636,LY-83636,LY 83636

Lergotrile mesylate, an ergoline derivative, suppresses prolactin in vivo and in vitro.
T34432 RU 28306

RU-28306,RU28306

RU 28306 is a racemic partial ergoline.
TQ0175 Dexpramipexole

右旋普拉克索,R-(+)-Pramipexole,(R)-Pramipexole,KNS-760704

Dopamine Receptor GPCR/G Protein; Neuroscience
Dexpramipexole (KNS-760704, R-(+)-Pramipexole) is a neuroprotective agent and weak non-ergoline dopamine agonist.
T25657 LEK 8841

LEK-8841,LEK8841

LEK 8841 is an ergoline derivative that is a potential antipsychotic.
T24003 Disulergine

CM 29717,CH 29717,CH 29-717

Disulergine is a dopamine receptor agonist. It also prolactin release-inhibiting 8 alpha-amino-ergoline.
T21340 Pergolide

Pergolide, an ergoline-based dopamine receptor agonist, is used for the treatment of Parkinson's disease, which is associated with low levels of the neurotransmitter dopamine in the brain.
T68440 Epicriptine

Epicriptine or beta-dihydroergocryptine is a dopamine agonist of the ergoline class. It constitutes one third of the mixture known as dihydroergocryptine, the other two thirds consisting of alpha-dihydroergocryptine. The alpha differs from the beta form only in the position of a single methyl group, which is a consequence of the biosynthesis in which the proteinogenic amino acid isoleucine is replaced by leucine.

化合物

Methyl Ergoline Acid
Cat.No: T9793
Synonym:
Target: Others
Lysergamide, N-cycloheptyl-, maleate
Cat.No: T31663
Synonym: Ergoline-8-beta-carboxamide, N-cycloheptyl-9,10-didehydro-6-methyl-, maleate
Target:
Lysergamide, N-cyclopropyl-, maleate
Cat.No: T31664
Synonym: Ergoline-8-beta-carboxamide, N-cyclopropyl-9,10-didehydro-6-methyl-, maleate
Target:
Pergolide mesylate
Cat.No: T2226
Synonym: 甲磺酸培高利特,Pergolide mesylate salt,LY127809,Pergolide methanesulfonate
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor
Nicergoline
Cat.No: T1132
Synonym: 尼麦角林,Nicergolinum,Nimergoline
Target: Adrenergic Receptor
Metergoline
Cat.No: T4008
Synonym: 甲麦角林,Methergoline,Liserdol
Target: Dopamine Receptor, 5-HT Receptor, Sodium Channel
Romergoline 2HCl
Cat.No: T71707L
Synonym: Romergoline 2HCl(107052-56-2 Free base),FCE 23884 2HCl
Target: Dopamine Receptor
Romergoline
Cat.No: T71707
Synonym:
Target:
Cabergoline diphosphate
Cat.No: T68551
Synonym:
Target:
Nicergoline tartrate
Cat.No: T1132L
Synonym: Adavin
Target:
Cianergoline
Cat.No: T25247
Synonym: Cianergolinum
Target:
Dexpramipexole dihydrochloride
Cat.No: T11011
Synonym: 普拉克索杂质D,KNS-760704 dihydrochloride,R-(+)-Pramipexole dihydrochloride,右旋普拉克索二盐酸盐,(R)-Pramipexole dihydrochloride
Target: Dopamine Receptor
Lergotrile mesylate
Cat.No: T25671L
Synonym: LY83636,LY-83636,LY 83636
Target:
RU 28306
Cat.No: T34432
Synonym: RU-28306,RU28306
Target:
Dexpramipexole
Cat.No: TQ0175
Synonym: 右旋普拉克索,R-(+)-Pramipexole,(R)-Pramipexole,KNS-760704
Target: Dopamine Receptor
LEK 8841
Cat.No: T25657
Synonym: LEK-8841,LEK8841
Target:
Disulergine
Cat.No: T24003
Synonym: CM 29717,CH 29717,CH 29-717
Target:
Pergolide
Cat.No: T21340
Synonym:
Target:
Epicriptine
Cat.No: T68440
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T14853 Cabergoline

FCE-21336,卡麦角林

Dopamine Receptor; 5-HT Receptor; Autophagy Autophagy; GPCR/G Protein; Neuroscience
Cabergoline (FCE-21336) 是一种麦角衍生的多巴胺 D2亚类受体激动剂,高亲和力作用于D2、D3和5-HT2B 受体,Ki 分别为 0.7、1.5 和 1.2。

天然产物

Cabergoline
Cat.No: T14853
Synonym: FCE-21336,卡麦角林
Target: Dopamine Receptor, 5-HT Receptor, Autophagy
TargetMol Loading
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