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10

抑制剂 & 化合物

5

天然产物

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Cat. No. Product Name Target Signaling Pathways
T0510 Sulfaguanidine

Sulfaguine,Guanicil,磺胺脒

Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology
Sulfaguanidine (Guanicil) 是一种具有口服活性的磺胺类抗菌剂和抗生素。它可用于肠道感染,例如细菌性痢疾的研究。
T1647 Ronidazole

洛硝哒唑,Ronidazol,罗硝唑,Ridzol

Antibacterial; Antibiotic; Parasite Microbiology/Virology
Ronidazole (Ronidazol) 是一种口服有效的抗原虫和抗菌试剂。它在猫模型中对胎儿三毛滴虫有效,还可研究组织口癣和猪痢疾。
T0512 Phthalylsulfathiazole

酞磺胺噻唑,Sulfathalidine,N4-Phthalylsulfathiazole

Antibacterial; Antibiotic Microbiology/Virology
Phthalylsulfathiazole (N4-Phthalylsulfathiazole) 是磺胺类抗菌药。
T9049 Difurazon hydrochloride

Others Others
Difurazon hydrochloride 是一种致突变药物。它可能已用于治疗细菌性痢疾。它是动物饲料中的抗菌促生长剂。
T0770 Carbadox

Getroxel,卡巴多,Mecadox

Antibacterial; Antibiotic Microbiology/Virology
Carbadox (Mecadox) 是一种喹喔啉二氧化氮抗生素,用于育龄期的猪,治疗猪痢疾和肠炎,促进成长。
T9549 Chiniofon

Loretin,Ferron,8-hydroxy-7-iodo-5-quinolinesulfonate,quiniophen,喹碘方

Others Others
Chiniofon (Ferron) 是一种卤代 8-羟基喹啉,用作抗阿米巴药物。该类抗阿米巴药物通过抑制肠道共生菌发挥抗阿米巴作用,影响阿米巴痢疾,但对肠外阿米巴寄生虫无作用。
T24777 Sedecamycin

T-2636A,T-2636,Ro 23-0731/000,NSC 145117

Sedecamycin is a 17-membered macrolide antibiotic. It is used for treating swine dysentery.
T40573 Hydroxymetronidazole

Hydroxymetronidazole,Metronidazole-OH

Hydroxymetronidazole (Metronidazole-OH) is a nitroimidazole compound that functions as a metabolite of Metronidazole. It is commonly employed in poultry research to investigate bacterial and protozoal diseases, as well as in the study of swine dysentery and genital trichomoniasis in cattle.
T24277 Hydroxy ipronidazole

L-12407,Ipronidazole-OH,L12407,L 12407

L 12407 is an antiprotozoal drug of the nitroimidazole class. It is used for the treatment of histomoniasis in turkeys and for swine dysentery.
T31006 Conessine hydrobromide

Neriine dihydrobromide,Konessin dihydrobromide,Conessine HCl

Conessine hydrobromide is a naturally occurring steroid alkaloid and has been used in traditional herbal medicine as a treatment for amoebic dysentery.

化合物

Sulfaguanidine
Cat.No: T0510
Synonym: Sulfaguine,Guanicil,磺胺脒
Target: Antibacterial, Antibiotic, Autophagy
Ronidazole
Cat.No: T1647
Synonym: 洛硝哒唑,Ronidazol,罗硝唑,Ridzol
Target: Antibacterial, Antibiotic, Parasite
Phthalylsulfathiazole
Cat.No: T0512
Synonym: 酞磺胺噻唑,Sulfathalidine,N4-Phthalylsulfathiazole
Target: Antibacterial, Antibiotic
Difurazon hydrochloride
Cat.No: T9049
Synonym:
Target: Others
Carbadox
Cat.No: T0770
Synonym: Getroxel,卡巴多,Mecadox
Target: Antibacterial, Antibiotic
Chiniofon
Cat.No: T9549
Synonym: Loretin,Ferron,8-hydroxy-7-iodo-5-quinolinesulfonate,quiniophen,喹碘方
Target: Others
Sedecamycin
Cat.No: T24777
Synonym: T-2636A,T-2636,Ro 23-0731/000,NSC 145117
Target:
Hydroxymetronidazole
Cat.No: T40573
Synonym: Hydroxymetronidazole,Metronidazole-OH
Target:
Hydroxy ipronidazole
Cat.No: T24277
Synonym: L-12407,Ipronidazole-OH,L12407,L 12407
Target:
Conessine hydrobromide
Cat.No: T31006
Synonym: Neriine dihydrobromide,Konessin dihydrobromide,Conessine HCl
Target:
Cat. No. Product Name Target Signaling Pathways
T8065 Tiamulin

Thiamutilin,泰妙菌素

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Tiamulin (Thiamutilin) 是一类二萜,广泛用于控制猪的传染疾病,包括猪痢疾和地方性肺炎等。
T0861 Tylosin tartrate

酒石酸泰洛星,酒石酸泰乐菌素

Antibacterial; Antibiotic Microbiology/Virology
Tylosin tartrate 是一种大环内酯类抗生素,是 Streptomyces fradiae 的产物。它对革兰氏阳性菌具有高效的抗菌活性。它作为饲料添加剂可促进动物生长。它被用于治疗家禽、猪和牛的细菌性痢疾和呼吸道疾病。
T1003 Tylosin

Fradizine,Tylosin A,泰乐菌素,Tylosine,Tylocine

Antibacterial; Antibiotic Microbiology/Virology
Tylosin (Tylosine) 是一种兽医用大环内酯类抗生素,是 Streptomyces fradiae 的产物。它对革兰氏阳性菌具有高抗菌活性。它是饲料添加剂用于促进动物生长。它被用于治疗家禽、猪和牛的细菌性痢疾和呼吸道疾病。
T5S0802 Palmatine

巴马汀,Berbericinine,Burasaine

Indoleamine 2,3-Dioxygenase (IDO); AChR; AChE; Aurora Kinase Cell Cycle/Checkpoint; Chromatin/Epigenetic; Metabolism; Neuroscience
Palmatine (Burasaine) 是口服具有活力的、不可逆IDO-1抑制剂。它可以减轻结肠损伤,预防肠道菌群失调和调节色氨酸分解代谢,从而改善DSS (Dextran Sulphate Sodium Salt) 诱发的结肠炎。它有用于结肠炎的研究潜力。
T4S1469 Cucurbitacin IIb

葫芦素IIB,雪胆素乙

Apoptosis; Others Apoptosis; Others
Cucurbitacin IIb 是一种雪胆中的活性成分。它阻碍 STAT3,JNK 和 Erk1/2 的磷酸化,提高 IκB 和 NF-κB (p65) 的磷酸化水平,抑制 NF-κB (p65) 的核转位,降低 IκBα 和 TNF-α 的 mRNA 水平。它能够诱导细胞凋亡,具有抗炎作用。

天然产物

Tiamulin
Cat.No: T8065
Synonym: Thiamutilin,泰妙菌素
Target: Others, Antibacterial, Antibiotic
Tylosin tartrate
Cat.No: T0861
Synonym: 酒石酸泰洛星,酒石酸泰乐菌素
Target: Antibacterial, Antibiotic
Tylosin
Cat.No: T1003
Synonym: Fradizine,Tylosin A,泰乐菌素,Tylosine,Tylocine
Target: Antibacterial, Antibiotic
Palmatine
Cat.No: T5S0802
Synonym: 巴马汀,Berbericinine,Burasaine
Target: Indoleamine 2,3-Dioxygenase (IDO), AChR, AChE, Aurora Kinase
Cucurbitacin IIb
Cat.No: T4S1469
Synonym: 葫芦素IIB,雪胆素乙
Target: Apoptosis, Others
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