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11

抑制剂 & 化合物

10

天然产物

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Cat. No. Product Name Target Signaling Pathways
T0001 Iron(II) fumarate

Ferrous fumarate,Iron Fumarate,富马酸铁 (II),富马酸亚铁

Others Others
Iron(II) fumarate (Ferrous fumarate) 是一种口服活性膳食补充剂,是一种富马酸的铁 (II) 盐,可用于研究缺铁性贫血。
T22484 (±)-Propionylcarnitine chloride

Propionyl-DL-carnitine chloride

Endogenous Metabolite Metabolism
(±)-Propionylcarnitine chloride (Propionyl-DL-carnitine chloride) 是一种短链酰基肉碱的混合物,可用作膳食补充剂,可用于研究慢性糖尿病。
T26551 Acetyl-L-carnitine

RO 447190,L-Acetylcarnitine,LAC,L-O-Acetylcarnitine,ALCAR,Acetyl L carnitine

Endogenous Metabolite Metabolism
Acetyl-L-carnitine(RO 447190) 是一种可透过血脑屏障的氨基酸左旋肉碱,常作为膳食补充剂,对神经炎症有益。Acetyl-L-carnitine 具有神经保护作用,可用以研究像阿尔茨海默病类的神经疾病。
T20062 Thiamine disulfide

二硫化硫胺,TDS,Daiomin,Algoneurina

HIV Protease; Endogenous Metabolite Metabolism; Microbiology/Virology; Proteases/Proteasome
Thiamine disulfide (Algoneurina) 是一种存在于食物中的维生素,可作为膳食补充剂和药物生产。 它还充当许多中枢代谢酶的辅助因子。
T13730 Hydroxocobalamin acetate

Others Others
Hydroxocobalamin acetate 是可注射的天然维生素 B12,其不良反应特征良好,可用于研究维生素 B12 缺乏症 (包括恶性贫血) 。
T36126 TMP-153

Acyl-CoA:cholesterol acyltransferase (ACAT) catalyses the esterification of excess cellular cholesterol with fatty acids and is important for intestinal cholesterol absorption, hepatic lipoprotein secretion, and cholesterol accumulation in vascular tissues. ACAT inhibitors improve plasma lipid profile and ameliorate proteinuria in nephrotic animals. TMP-153 is a quinolyl derivative that inhibits ACAT with IC50 values of 5-10 nM in various animals. At 0.5-1.5 mg/kg, TMP-153 dose-dependently reduc...
T19528 Propionylcarnitine

Propionyl carnitine

Others Others
Propionylcarnitine (Propionyl carnitine) 是一种被广泛使用的膳食补充剂,有青光眼和难道破裂有关。
T1129 Benfotiamine

Benzoylthiamine monophosphate,S-Benzoylthiamine O-monophosphate,苯磷硫胺

Others Others
Benfotiamine (S-Benzoylthiamine O-monophosphate) 是维生素 B1 的类似物,其吸收率和生物利用度比维生素B1高,具有直接抗氧化能力,可防止DNA 损伤。它常用作糖尿病并发症的食品补充剂。
T75328 Hydroxocobalamin hydrochloride

Hydroxocobalamin hydrochloride 是天然维生素B12的可注射形式,因其优良的安全性质,被用于研究维生素B12缺乏症(包括恶性贫血)相关治疗。
T37532 Docosahexaenoyl Glycine

The ω-3 polyunsaturated fatty acids (PUFAs) found in fish oils provide cardiovascular benefits. Docosahexaenoic acid (DHA), a C22:6 PUFA, is the most abundant ω-3 fatty acid in neural tissues, especially in the retina and brain. It can be synthesized from other dietary ω-3 PUFAs or taken as a nutritional supplement. Docosahexaenoyl glycine consists of DHA with glycine attached at its carboxy terminus.
T79919 S-Adenosyl-L-methionine (1,4-butanedisulfonate)

Ademetionine (1,4-butanedisulfonate),S-Adenosyl methionine (1,4-butanedisulfonate),AdoMet (1,4-butanedisulfonate)

Endogenous Metabolite Metabolism
S-Adenosyl-L-methionine (S-Adenosyl methionine) 1,4-butanedisulfonate 作为一种口服活性的甲基供体,它是一种膳食补充剂,对抗抑郁和缓解疼痛具有显著功效。此化合物在癌症治疗中显示了抗增殖、促进凋亡和阻止转移的潜在作用。同时,S-Adenosyl-L-methionine 1,4-butanedisulfonate 也用于肝病和骨关节炎的相关研究。

化合物

Iron(II) fumarate
Cat.No: T0001
Synonym: Ferrous fumarate,Iron Fumarate,富马酸铁 (II),富马酸亚铁
Target: Others
(±)-Propionylcarnitine chloride
Cat.No: T22484
Synonym: Propionyl-DL-carnitine chloride
Target: Endogenous Metabolite
Acetyl-L-carnitine
Cat.No: T26551
Synonym: RO 447190,L-Acetylcarnitine,LAC,L-O-Acetylcarnitine,ALCAR,Acetyl L carnitine
Target: Endogenous Metabolite
Thiamine disulfide
Cat.No: T20062
Synonym: 二硫化硫胺,TDS,Daiomin,Algoneurina
Target: HIV Protease, Endogenous Metabolite
Hydroxocobalamin acetate
Cat.No: T13730
Synonym:
Target: Others
TMP-153
Cat.No: T36126
Synonym:
Target:
Propionylcarnitine
Cat.No: T19528
Synonym: Propionyl carnitine
Target: Others
Benfotiamine
Cat.No: T1129
Synonym: Benzoylthiamine monophosphate,S-Benzoylthiamine O-monophosphate,苯磷硫胺
Target: Others
Hydroxocobalamin hydrochloride
Cat.No: T75328
Synonym:
Target:
Docosahexaenoyl Glycine
Cat.No: T37532
Synonym:
Target:
S-Adenosyl-L-methionine (1,4-butanedisulfonate)
Cat.No: T79919
Synonym: Ademetionine (1,4-butanedisulfonate),S-Adenosyl methionine (1,4-butanedisulfonate),AdoMet (1,4-butanedisulfonate)
Target: Endogenous Metabolite
Cat. No. Product Name Target Signaling Pathways
T2207 Adrenosterone

肾上腺甾酮,11-ketoandrostenedione,11-oxoandrostenedione,Reichstein's substance G

Androgen Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Adrenosterone (11-ketoandrostenedione) 是一种人内源性代谢物,由肾上腺皮质产生。Adrenosterone 是一种竞争性羟基类固醇脱氢酶 1 抑制剂。它是一种的类固醇激素,具有较弱的雄激素特性。它是一种膳食补充剂,能够减少脂肪并提高肌肉质量。它能够抑制人类癌细胞的转移进展。
T1286 Vincamine

Angiopac,Oxybral,Devincan,Novicet,Equipur,长春胺,Perval

GPR; Others Endocrinology/Hormones; GPCR/G Protein; Others
Vincamine (Perval) 是从长春花中提取的单萜类吲哚生物碱,可作为外周血管扩张剂,对脑微血管循环有选择性的血管调节作用。它可改善体内葡萄糖稳态,对 2 型糖尿病具有研究潜力。它是GPR40激动剂,通过改善 β 细胞功能障碍和促进葡萄糖刺激型胰岛素分泌发挥 β 细胞保护作用。
T7475 S-Adenosyl-L-methionine

AdoMet,Ademetionine,SAMe,S-Adenosyl methionine,S-腺苷-L-蛋氨酸

Others; Endogenous Metabolite Metabolism; Others
S-Adenosyl-L-methionine (Ademetionine) 是一种具有有效的抗抑郁和减轻疼痛作用的膳食补充剂,是通过蛋氨酸腺苷转移酶的作用由蛋氨酸和 ATP 内源性生产的,是一种重要的口服具有活力的甲基供体,能够用于肝病和骨关节炎的研究。
T22293 Chondroitine sulfate

Chondroitine sulfate (From cattle)

Others Others
Chondroitine sulfate 是软骨的重要结构成分,已被用作治疗关节不适的膳食补充剂。
T19608 Zinc sulfate heptahydrate

Others Others
Zinc sulfate heptahydrate 是七水合形式的硫酸锌,是一种膳食补充剂,可用于锌缺乏症和预防高危人群的锌缺乏症。
T0978 Pantethine

LBF disulfide,Pantosin,Pantetina,Bis-pantethine,泛硫乙胺(维生素B5),泛硫乙胺,Pantomin,D-Pantethine

Endogenous Metabolite Metabolism
D-Pantethine (Pantomin) 是泛酸的二聚体形式, 是生产辅酶 A 的中间体。D-Pantethine 能够作为膳食补充剂,用于改善血液胆固醇和研究痤疮。
T3578 Pyridoxal phosphate

PLP,PAL-P,磷酸吡哆醛,pyridoxal 5'-phosphate,Pyridoxyl phosphate,Pyridoxal 5′-phosphate,Vitamin B6 phosphate

Reverse Transcriptase; Endogenous Metabolite Metabolism; Microbiology/Virology
Pyridoxal phosphate (Vitamin B6 phosphate) 是维生素 B6 的活性形式,可抑制逆转录酶活性,用于研究迟发性运动障碍症。
T13731 Hydroxocobalamin monohydrochloride

Vitamin B12a monohydrochloride,盐酸羟钴胺

Others Others
Hydroxocobalamin monohydrochloride is an injectable naturally occurring form of vitamin B12. It is used as a dietary supplement in the treatment of vitamin B12 deficiency including pernicious anemia.
TN1590 DL-alpha-Tocopherylacetate

Dl-alpha-tocopheryl acetate is a dietary supplement.
T78476 Hydroxocobalamin

Vitamin B12a

Endogenous Metabolite Metabolism
Hydroxocobalamin(Vitamin B12a)为可注射型天然维生素B12,不良反应特性良好,适用于治疗维生素B12缺乏症(包括恶性贫血)的膳食补充。

天然产物

Adrenosterone
Cat.No: T2207
Synonym: 肾上腺甾酮,11-ketoandrostenedione,11-oxoandrostenedione,Reichstein's substance G
Target: Androgen Receptor, Endogenous Metabolite
Vincamine
Cat.No: T1286
Synonym: Angiopac,Oxybral,Devincan,Novicet,Equipur,长春胺,Perval
Target: GPR, Others
S-Adenosyl-L-methionine
Cat.No: T7475
Synonym: AdoMet,Ademetionine,SAMe,S-Adenosyl methionine,S-腺苷-L-蛋氨酸
Target: Others, Endogenous Metabolite
Chondroitine sulfate
Cat.No: T22293
Synonym: Chondroitine sulfate (From cattle)
Target: Others
Zinc sulfate heptahydrate
Cat.No: T19608
Synonym:
Target: Others
Pantethine
Cat.No: T0978
Synonym: LBF disulfide,Pantosin,Pantetina,Bis-pantethine,泛硫乙胺(维生素B5),泛硫乙胺,Pantomin,D-Pantethine
Target: Endogenous Metabolite
Pyridoxal phosphate
Cat.No: T3578
Synonym: PLP,PAL-P,磷酸吡哆醛,pyridoxal 5'-phosphate,Pyridoxyl phosphate,Pyridoxal 5′-phosphate,Vitamin B6 phosphate
Target: Reverse Transcriptase, Endogenous Metabolite
Hydroxocobalamin monohydrochloride
Cat.No: T13731
Synonym: Vitamin B12a monohydrochloride,盐酸羟钴胺
Target: Others
DL-alpha-Tocopherylacetate
Cat.No: TN1590
Synonym:
Target:
Hydroxocobalamin
Cat.No: T78476
Synonym: Vitamin B12a
Target: Endogenous Metabolite
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