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抑制剂 & 化合物

5

天然产物

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Cat. No. Product Name Target Signaling Pathways
T69207 Chelerythrine hydroxide

Chelerythrine hydroxide is the salt form of Chelerythrine, a benzophenanthridine alkaloid present in the plant Chelidonium majus (greater celandine). It is a potent, selective, and cell-permeable protein kinase C inhibitor in vitro. And an efficacious antagonist of G-protein-coupled CB1 receptors.]This molecule also exhibits anticancer qualities and it has served as a base for many potential novel drugs against cancer.

化合物

Chelerythrine hydroxide
Cat.No: T69207
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN1305 Ethoxysanguinarine

乙氧基血根碱,6-Ethoxydihydrosanguinarine

Apoptosis; AChR Apoptosis; Neuroscience
Ethoxysanguinarine (6-Ethoxydihydrosanguinarine) 是存在于龙葵中的一种苯并菲啶生物碱天然产物,通过抑制蛋白磷酸酶 2A,可抑制结直肠癌细胞活力,诱导细胞凋亡。
T0129 Sanguinarine chloride

Pseudochelerythrine chloride,血根碱,氯化血根碱,Sanguinarium chloride

Apoptosis; EGFR; VEGFR; Antibacterial; Parasite; Autophagy Angiogenesis; Apoptosis; Autophagy; JAK/STAT signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors
Sanguinarine chloride (Pseudochelerythrine chloride) 是一种来源于 Sanguinaria Canadensis 的生物碱,通过激活活性氧的产生,诱导细胞凋亡。
T8859 NITIDINE

Others Others
NITIDINE 是一种从花椒根中分离出来的具有生物活性的植物苯并菲啶生物碱。它具有抗癌、神经保护、抗疟疾、抗 HIV、镇痛、抗炎和抗真菌活性。
T3419 Chelerythrine chloride

白屈菜红碱,盐酸白屈菜红碱

Apoptosis; BCL; PKC; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling
Chelerythrine chloride 是一种可渗透细胞的蛋白激酶 C 抑制剂,对磷酸盐受体具有竞争性,而对 ATP 是非竞争性的。它诱导细胞凋亡和自噬。
T6S0052 Chelerythrine

Toddalin,Broussonpapyrine,白屈菜红碱,Cheleritrine

Apoptosis; BCL; PKC; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling
Chelerythrine (Broussonpapyrine) 是一种天然生物碱,为有效、选择性的 Ca2+/磷脂依赖性PKC 拮抗剂,IC50值为 0.7 μM。它具有抗肿瘤、抗糖尿病、抗炎的活性。它抑制BclXL-Bak BH3肽结合,IC50为 1.5 μM,并从 BclXL 取代了 Bax。它诱导细胞凋亡和自噬。

天然产物

Ethoxysanguinarine
Cat.No: TN1305
Synonym: 乙氧基血根碱,6-Ethoxydihydrosanguinarine
Target: Apoptosis, AChR
Sanguinarine chloride
Cat.No: T0129
Synonym: Pseudochelerythrine chloride,血根碱,氯化血根碱,Sanguinarium chloride
Target: Apoptosis, EGFR, VEGFR, Antibacterial, Parasite, Autophagy
NITIDINE
Cat.No: T8859
Synonym:
Target: Others
Chelerythrine chloride
Cat.No: T3419
Synonym: 白屈菜红碱,盐酸白屈菜红碱
Target: Apoptosis, BCL, PKC, Autophagy
Chelerythrine
Cat.No: T6S0052
Synonym: Toddalin,Broussonpapyrine,白屈菜红碱,Cheleritrine
Target: Apoptosis, BCL, PKC, Autophagy
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