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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T35040 Vatiquinone

EPI-743,EPI743,alpha-Tocotrienol quinone. ATQ3,EPI 743

Vatiquinone, also known as EPI 743, is an orally bioavailable para-benzoquinone being developed for inherited mitochondrial diseases. The mechanism of action of EPI-743 involves augmenting the synthesis of glutathione, optimizing metabolic control, enhanc

化合物

Vatiquinone
Cat.No: T35040
Synonym: EPI-743,EPI743,alpha-Tocotrienol quinone. ATQ3,EPI 743
Target:
Cat. No. Product Name Target Signaling Pathways
T9675 α-Tocotrienol

Endogenous Metabolite Metabolism
α-Tocotrienol 是维生素 E 的一种亚型,存在于蔬菜、水果、种子、坚果、谷物和油脂中。α-Tocotrienol 是抗氧化剂,可以降低胆固醇和其他脂类,也是神经保护和抗癌剂,在心血管疾病的保护中发挥作用。
T19768 γ-Tocotrienol

gamma Tocotrienol,gammaTocotrienol,gamma-Tocotrienol,D-gamma-Tocotrienol,Plastochromanol,γ-生育三烯酚

Others Others
γ-Tocotrienol (Plastochromanol) 是一种维生素 E 的活性形式。
TMA2474 δ-Tocotrienol

Delta-Tocotrienol,δ-生育三烯酚

ERK; BCL; VEGFR; Akt; PI3K; PDK; p53 Angiogenesis; Apoptosis; Cytoskeletal Signaling; MAPK; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
δ-Tocotrienol (Delta-Tocotrienol) 是一种维生素 E,存在于蔬菜,水果,种子,坚果,谷物和油等。维生素 E 是抗氧化剂、神经保护剂和抗癌剂,可以降低胆固醇和其他脂质,保护心血管疾病。
T21523 β-Tocotrienol

Beta-Tocotrienol

Caspase Apoptosis; Proteases/Proteasome
Beta-Tocotrienol to serve as a new anticancer agent for treating human lung and brain cancers. It inhibits the growth of both A549 (GI50=1.38±0.334μM) and U87MG (GI50=2.53±0.604μM) cells at rather low concentrations.

天然产物

α-Tocotrienol
Cat.No: T9675
Synonym:
Target: Endogenous Metabolite
γ-Tocotrienol
Cat.No: T19768
Synonym: gamma Tocotrienol,gammaTocotrienol,gamma-Tocotrienol,D-gamma-Tocotrienol,Plastochromanol,γ-生育三烯酚
Target: Others
δ-Tocotrienol
Cat.No: TMA2474
Synonym: Delta-Tocotrienol,δ-生育三烯酚
Target: ERK, BCL, VEGFR, Akt, PI3K, PDK, p53
β-Tocotrienol
Cat.No: T21523
Synonym: Beta-Tocotrienol
Target: Caspase
TargetMol Loading
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