11
5
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T9618 |
HeE1-2Tyr
|
SARS-CoV | Microbiology/Virology |
HeE1-2Tyr 是 一种pyridobenzothiazole,抑制黄病毒 RNA 依赖性 RNA 聚合酶。HeE1-2Tyr 在体外对Dengue, West Nile 和 SARS-CoV-2 RdRps 有显著的抑制活性(IC50为 27.6 µM) 。 | |||
T72041 |
Flaviviruses-IN-2
|
Virus Protease | Microbiology/Virology |
Flaviviruses-IN-2 是一种有效的 flaviviruses 抑制剂。 Flaviviruses-IN-2 可降低 西尼罗河病毒(WNV)蛋白酶活性,对西尼罗河病毒的抑制率为 56%。 | |||
T67777 |
Flaviviruses-IN-3
WAY-324593 |
Virus Protease | Microbiology/Virology |
Flaviviruses-IN-3(化合物87)是flaviviruse 的有效抑制剂。Flaviviruses-IN-3可降低西尼罗河病毒(WNV)蛋白酶活性,抑制率为54%。 | |||
TNU0060 |
3’-O-Methyladenosine
|
Antiviral; Adenosine deaminase | Immunology/Inflammation; Metabolism |
3’-O-Methyladenosine 是一种抗病毒化合物,对西尼罗河病毒具有抑制作用,可用于治疗病毒感染。3’-O-Methyladenosine 对腺苷脱氨酶VII型具有抑制作用,Ki 值为 493 µM。 | |||
TNU0007 |
3'-Deoxy-3'-fluoroadenosine
|
Nucleoside Antimetabolite/Analog | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
3'-Deoxy-3'-fluoroadenosine 是一种嘌呤核苷类似物,具有广泛的抗肿瘤活性和抗病毒活性,对蜱传脑炎病毒(TBEV),寨卡病毒和西尼罗河病毒(WNV)具有抑制作用,EC50分别为1.1μM、 0.1 μM和4.7 1.5 μM。3'-Deoxy-3'-fluoroadenosine可用于研究肿瘤疾病。 | |||
T4027 |
KIN1148
|
Influenza Virus | Microbiology/Virology |
KIN1148 是一种新型小分子佐剂,是IRF3激动剂,用于增强流感疫苗效率。 | |||
T33381 |
Micordilin
|
||
Micordilin is isolated from West Indian medicinal plant Mikania cordifolia. | |||
T81309 |
RCB16007
|
||
RCB16007为一种抗黄热病毒(YFV)化合物,对西尼罗河病毒显示出抑制活性,具体抑制浓度为EC50: 7.9 μM,细胞毒性浓度为CC50: 17 μM。 | |||
T70855 | Favipiravir sodium | ||
Favipiravir sodium is a selective inhibitor of viral RNA-dependent RNA polymerase with activity against many RNA viruses, influenza viruses, West Nile virus, yellow fever virus, foot-and-mouth disease virus as well as other flaviviruses, arenaviruses, bunyaviruses and alphaviruses. | |||
T38861 |
Tat-beclin 1
|
||
Tat-beclin 1, a peptide derived from the autophagy protein beclin 1, is a powerful inducer of autophagy. It interacts with GAPR-1 (GLIPR2), a negative regulator of autophagy. Tat-beclin 1 effectively reduces the buildup of polyglutamine expansion protein aggregates and inhibits the replication of various pathogens, such as HIV-1, in laboratory experiments. In addition, it has demonstrated the ability to decrease mortality in mice infected with chikungunya (CHIKV) or West Nile virus (WNV). | |||
T76058 |
Tat-beclin 1 TFA
|
||
Tat-beclin 1 TFA是一种来源于自噬蛋白区域(beclin 1)的肽,有效诱导自噬(autophagy)并与GAPR-1 (GLIPR2)发生相互作用,具有显著的自噬负调控作用。该化合物能有效减少体外聚谷氨酰胺扩增蛋白聚集体的积累,并抑制HIV-1等多种病原体的复制。同时,Tat-beclin 1 TFA能显著降低感染基孔肯雅病(CHIKV)或西尼罗河病毒(WNV)小鼠的死亡率。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2718 |
Palmatine chloride
|
Others; Indoleamine 2,3-Dioxygenase (IDO); Aurora Kinase | Cell Cycle/Checkpoint; Chromatin/Epigenetic; Metabolism; Others |
Palmatine chloride 是口服具有活力的不可逆 IDO-1抑制剂。它能够减轻结肠损伤,预防肠道菌群失调和调节色氨酸分解代谢,并改善 DSS 诱发的结肠炎。 | |||
T5S0802 |
Palmatine
巴马汀,Berbericinine,Burasaine |
Indoleamine 2,3-Dioxygenase (IDO); AChR; AChE; Aurora Kinase | Cell Cycle/Checkpoint; Chromatin/Epigenetic; Metabolism; Neuroscience |
Palmatine (Burasaine) 是口服具有活力的、不可逆IDO-1抑制剂。它可以减轻结肠损伤,预防肠道菌群失调和调节色氨酸分解代谢,从而改善DSS (Dextran Sulphate Sodium Salt) 诱发的结肠炎。它有用于结肠炎的研究潜力。 | |||
T3S0693 |
Blinin
|
Others | Others |
Blinin 是一种二萜,分离自植物 Conyza blinii 中。 | |||
T25789 |
Melianone
NSC 302037,NSC-302037,NSC302037 |
||
Melianone exhibits antiviral activity (EC50s: 3-11μM) against three important human pathogens, belonging to the Flaviviridae family, West Nile virus, Dengue virus, and Yellow Fever virus. | |||
T72508 | Palmatine hydroxide | ||
Palmatine hydroxide 是不可逆的口服活性IDO-1抑制剂,其对HEK 293-hIDO-1 和 rhIDO-1的IC50值分别为3 μM和157 μM。该化合物还能非竞争性抑制(WNV)NS2B-NS3蛋白酶,IC50值为96 μM。Palmatine hydroxide展现了抗癌、抗炎、神经保护、抗细菌和抗病毒的活性。 |