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Cat. No.	Product Name	Target	Signaling Pathways
T126501	Xanthone V1a
	Xanthone V1a 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T126501。
T11857	LIT-001	Oxytocin Receptor	Endocrinology/Hormones; GPCR/G Protein
	LIT-001 是非肽类催产素受体激动剂，EC50为55 nM，Ki 为226 nM。它可改善孤独症小鼠模型的社交互动。
T80160	ω-Hexatoxin-Hv1a ω-ACTX-Hv1,ω-Atracotoxin-HV1	Calcium Channel	Membrane transporter/Ion channel; Metabolism
	ω-Hexatoxin-Hv1a，一种从毒液蜘蛛 (Hadronyche versuta) 分离得到的神经毒素，能够阻断电压门控钙通道 (calcium channels)。
T6453	Conivaptan hydrochloride Vaprisol,盐酸考尼伐坦,Conivaptan HCl,YM 087	Vasopressin Receptor	GPCR/G Protein
	Conivaptan hydrochloride (Vaprisol) 是一种口服有效的加压素 V2 和 V1A 受体拮抗剂，用于治疗高血容量性低钠血症和正常血容量。
T4141	RG7713 RO 5028442	Vasopressin Receptor	GPCR/G Protein
	RG7713 (RO 5028442) 是一种高效且有选择性的脑-渗透加压素 1a (V1a) 受体拮抗剂，对人类 (hV1a) 和小鼠 (mV1a) 受体的 Ki 值分别为 1 和 39 nM，可用于研究自闭症的试验。
TP2082L	d[Cha4]-AVP acetate(500170-27-4 free base)	Vasopressin Receptor	GPCR/G Protein
	d[Cha4]-AVP acetate(500170-27-4 free base) 是一种有效的选择性人血管加压素 V1B 受体激动剂（V1B、V1A、催产素和 V2 受体的 Ki 值分别为 1.2、151、240 和 750 nM）。刺激 ACTH 和皮质酮分泌，并在体内表现出微不足道的血管加压活性。
T14494	Balovaptan RG7314	Vasopressin Receptor	GPCR/G Protein
	Balovaptan (RG7314) 是一种高效和选择性的脑渗透性血管加压素 1a (hV1a) 受体拮抗剂，对人类 (hV1a) 和小鼠 (mV1a) 受体的 Ki 值分别为 1 和 39 nM，可用于自闭症的研究。
T16934	SRX246	Others	Others
	SRX246 has no interaction at V1b and V2 receptors. SRX246 shows negligible binding at 64 other receptors classes, including 35 G-proteincoupled receptors. SRX246 is a potent and CNS-penetrant vasopressin 1a (V1a) receptor antagonist (Ki=0.3 nM for human V
T28629	RWJ 676070 RWJ676070,RWJ-676070
	RWJ 676070 is an antagonist of vasopressin V1A/V2 receptor.
T24625	PF-184563 PF184563,PF 184563
	PF-184563 is an effective and selective non-peptidic V1a receptor antagonist.
T28745	Selepressin FE 202158,FE202158
	Selepressin, an analog of vasopressin, is a potent, selective vasopressin V1a receptor agonist.
T17251	VNA-932 WAY-VNA 932	Others	Others
	VNA-932 is an agonist of the vasopressin V2-receptor (IC50: 80.3 nM and 778 nM in human-V2 binding and V1a binding assay).
T28854	SRX 251 SRX-251,SRX251
	SRX 251, a vasopressin V1a receptor antagonist, is used potentially for the treatment of primary dysmenorrhea.
T29177	YM 218 YM218,YM-218
	YM 218 is a novel, potent, selective antagonist of nonpeptide vasopressin V1A receptor.
T23393	SR 49059	Others	Others
	vasopressin V1A receptor antagonist
T80137	(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin d(CH2)5[Tyr(Me)2, Dab5]AVP	Vasopressin Receptor	GPCR/G Protein
	(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin (d(CH2)5[Tyr(Me)2, Dab5]AVP)作为针对加压素受体V1a的特异性拮抗剂，具有pA2值为6.71。
T15682	L-371,257	Oxytocin Receptor; Vasopressin Receptor	Endocrinology/Hormones; GPCR/G Protein
	L-371,257 是催产素受体的竞争性拮抗剂，pA2 为 8.4，Ki 为 19 nM。 L-371,257 对加压素受体 1a 的 Ki 值为 3.7 nM。
T25577	Khusimol
	Khusimol is a vasopressin V1a receptors non-peptide ligand that acts by inhibiting the binding of vasopressin.
T29178	YM 471 YM-471,YM471
	YM 471 is a non-peptide arginine vasopressin (AVP) V1A and V2 receptor antagonist with oral activity.
TP2136	(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
	Selective vasopressin V1A receptor antagonist. Inhibits vasopressin and oxytocin-induced increases in intracellular calcium concentrations in vitro (IC50 values are 5 and 30 nM respectively). Exhibits potent and prolonged antivasopressor activity and indu
T24370	L-368899 free base L 368899,L 368,899,L368,899,L-368899,L368899,L-368,899
	L-368899 is a non-peptide and orally active antagonist of oxytocin receptor (IC50: 8.9 nM). It displays 40-fold selectivity over vasopressin V1a and V2 receptors (IC50: 370 and 570 nM respectively).
T80270	Invopressin OCE-205	Vasopressin Receptor	GPCR/G Protein
	Invopressin (Compound 42)，一种vasopressin V1A 受体部分激动剂（EC50: 1.0 nM），主要应用于肝硬化相关症状如细菌性腹膜炎、HRS2 及难治性腹水的研究。
TP1927	d[Leu4,Lys8]-VP
	Selective vasopressin V1B receptor agonist (Ki values are 0.16, 64, 100 and 3800 nM for V1B, oxytocin, V2 and V1A receptors respectively). Displays weak antidiuretic, vasopressor and in vitro oxytocic activities.
T80136	Val9-Oxytocin	Vasopressin Receptor	GPCR/G Protein
	Val9-Oxytocin为完全抗拮抗加压素(1a)受体的化合物，其结构上是Oxytocin的衍生物，特点在于Gly9位点被Val9取代。
TP2082	d[Cha4]-AVP
	Potent and selective human vasopressin V1B receptor agonist (Ki values are 1.2, 151, 240 and 750 nM for V1B, V1A, Oxytocin and V2 receptors respectively). Stimulates ACTH and corticosterone secretion and exhibits negligible vasopressor activity in vivo.
T75933	d[Cha4]-AVP TFA
	d[Cha4]-AVP TFA 是一种有效的选择性加压素 (AVP)V1b 受体激动剂，对人V1b 受体的Ki 为 1.2 nM。d[Cha4]-AVP TFA 对 V1b 受体的选择性高于对人类 V1a 受体、V2 受体和催产素受体。
T21378	Conivaptan YM087,YM-087,YM 087,Vaprisol
	Conivaptan, a non-peptide inhibitor of antidiuretic hormone, was approved for hyponatremia caused by the syndrome of inappropriate antidiuretic hormone (SIADH), there is also some evidence that it may be effective in heart failure. Conivaptan inhibits sub
T75708	Argipressin diacetate
	Argipressin (diacetate) (AVP (diacetate)，又称antidiuretic hormone (ADH)) 是一种由垂体后叶分泌的含9个氨基酸的神经肽。通过作用于三种G蛋白偶联受体(GPCRs)，Avpr1a (V1a)、Avpr1b (V1b) 及Avpr2 (V2)，它调控体液平衡、渗透压及心血管系统的生理功能，并可能对中枢代谢过程产生重要影响。
T73654	Selepressin acetate
	Selepressin (FE 202158) acetate 是一种选择性的加压素 V1A 受体 (vasopressin V1Areceptor) 激动剂。Selepressin acetate 是一种有效的血管加压素。Selepressin acetate 可用于脓毒性休克的研究。
T28257	OPC-51803 SOU-003,SOU 003,SOU003,OPC51803,OPC 51803	Vasopressin Receptor	GPCR/G Protein
	OPC-51803是一种可口服的非肽加压素（AVP）V（2）受体选择性激动剂，可用于治疗尿失禁和夜尿。

化合物

Cat.No: T126501

Cat.No: T11857

Target: Oxytocin Receptor

ω-Hexatoxin-Hv1a

Cat.No: T80160

Synonym: ω-ACTX-Hv1,ω-Atracotoxin-HV1

Target: Calcium Channel

Conivaptan hydrochloride

Cat.No: T6453

Synonym: Vaprisol,盐酸考尼伐坦,Conivaptan HCl,YM 087

Target: Vasopressin Receptor

Cat.No: T4141

Synonym: RO 5028442

Target: Vasopressin Receptor

d[Cha4]-AVP acetate(500170-27-4 free base)

Cat.No: TP2082L

Target: Vasopressin Receptor

Cat.No: T14494

Synonym: RG7314

Target: Vasopressin Receptor

Cat.No: T16934

Target: Others

Cat.No: T28629

Synonym: RWJ676070,RWJ-676070

Cat.No: T24625

Synonym: PF184563,PF 184563

Cat.No: T28745

Synonym: FE 202158,FE202158

Cat.No: T17251

Synonym: WAY-VNA 932

Target: Others

Cat.No: T28854

Synonym: SRX-251,SRX251

Cat.No: T29177

Synonym: YM218,YM-218

Cat.No: T23393

Target: Others

(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin

Cat.No: T80137

Synonym: d(CH2)5[Tyr(Me)2, Dab5]AVP

Target: Vasopressin Receptor

Cat.No: T15682

Target: Oxytocin Receptor, Vasopressin Receptor

Cat.No: T25577

Cat.No: T29178

Synonym: YM-471,YM471

(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin

Cat.No: TP2136

L-368899 free base

Cat.No: T24370

Synonym: L 368899,L 368,899,L368,899,L-368899,L368899,L-368,899

Cat.No: T80270

Synonym: OCE-205

Target: Vasopressin Receptor

d[Leu4,Lys8]-VP

Cat.No: TP1927

Cat.No: T80136

Target: Vasopressin Receptor

Cat.No: TP2082

d[Cha4]-AVP TFA

Cat.No: T75933

Cat.No: T21378

Synonym: YM087,YM-087,YM 087,Vaprisol

Argipressin diacetate

Cat.No: T75708

Selepressin acetate

Cat.No: T73654

Cat.No: T28257

Synonym: SOU-003,SOU 003,SOU003,OPC51803,OPC 51803

Target: Vasopressin Receptor

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