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Cat. No. Product Name Target Signaling Pathways
T16156 MT 63-78

Apoptosis; AMPK; mTOR Apoptosis; Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
MT 63-78 是一种有效的直接AMPK 激活剂,EC50为 25 μM。它诱导细胞有丝分裂阻滞和细胞凋亡,通过抑制脂肪生成和mTORC1途径来阻止前列腺癌的生长,具有抗肿瘤作用。
T1838 Sapanisertib

沙帕色替,TAK-228,MLN0128,INK 128

PI3K; mTOR; Autophagy Autophagy; PI3K/Akt/mTOR signaling
Sapanisertib (INK 128) 是一种口服有效的 ATP 依赖性的mTOR1/2抑制剂,抑制 mTOR 激酶的IC50值为 1 nM,具有潜在抗肿瘤活性。
T31223 DCBCI0901

DCBCI-0901,DCBCI 0901

DCBCI0901 is an inhibitor of phosphatidylinositide 3-kinase (PI3K), raptor-mTOR (mTOR complex 1 or mTORC1) and rictor-mTOR (mTOR complex 2 or mTORC2) with potential antineoplastic activity.
T30441 BI-860585

BI860585

BI-860585 is an inhibitor of Raptor-Mammalian Target of Rapamycin (mTOR) Complex 1 (mTOR Complex 1; mTORC1) and rictor-mTOR Complex 2 (mTOR Complex 2; mTORC2), with potential Anti-tumor activity.

化合物

MT 63-78
Cat.No: T16156
Synonym:
Target: Apoptosis, AMPK, mTOR
Sapanisertib
Cat.No: T1838
Synonym: 沙帕色替,TAK-228,MLN0128,INK 128
Target: PI3K, mTOR, Autophagy
DCBCI0901
Cat.No: T31223
Synonym: DCBCI-0901,DCBCI 0901
Target:
BI-860585
Cat.No: T30441
Synonym: BI860585
Target:
TargetMol Loading
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