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Cat. No. Product Name Target Signaling Pathways
T0189 Pemetrexed

Pemetrexed acid,培美曲塞,LY231514,培美曲唑,LY-231514 Disodium Hydrate

DHFR; DNA/RNA Synthesis; Antifolate; Autophagy Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
Pemetrexed (LY-231514 Disodium Hydrate) acid 是一种鸟嘌呤衍生的抗肿瘤药物,可结合并抑制胸苷酸合酶、二氢叶酸还原酶和甘氨酰胺核苷酸甲酰转移酶的 Ki 分别为 1.3 nM、7.2 nM 和 65 nM。
T6226 Pemetrexed disodium hemipenta hydrate

培美曲塞二钠一水合物,Pemetrexed Disodium Hydrate,LY-231514 Disodium Hydrate,Pemetrexed sodium hydrate,培美曲塞二钠水合物

Apoptosis; DHFR; DNA/RNA Synthesis; Antifolate; Autophagy Apoptosis; Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
Pemetrexed disodium hemipenta hydrate (LY-231514 Disodium Hydrate) 是一种叶酸拮抗剂。抑制胸苷酸合成酶 (TS),二氢叶酸还原酶 (DHFR) 和甘氨酰胺核苷酸甲酰转移酶 (GARFT),Ki 分别为 1.3 nM,7.2 nM 和 65 nM。
T0189L Pemetrexed disodium

培美曲塞二钠盐,LY-231514,LY231514 disodium,培美曲塞二钠,Pemetrexed

Apoptosis; DHFR; DNA/RNA Synthesis; Antifolate; Autophagy Apoptosis; Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
Pemetrexed disodium (LY-231514) 是一种叶酸拮抗剂,用于治疗非小细胞肺癌和恶性间皮瘤。它抑制胸苷酸合成酶,二氢叶酸还原酶和甘氨酰胺核苷酸甲酰转移酶的Ki 分别为 1.3 nM,7.2 nM 和 65 nM。
T25929 Pemetrexed tromethamine

Pemetrexed ditromethamine dihydrate

Pemetrexed tromethamine is a chemotherapy drug used for pleural mesothelioma and non-small cell lung cancer.
T70583 Pemetrexed Diethyl Ester

Pemetrexed Diethyl Ester is a protected intermediate in the synthesis of Pemetrexed, a multi-targeted anti-folate that inhibits thymidylate synthase as well as other folate dependent enzymes.
T20355 LY-338979

Pemetrexed 6-oxo diacid impurity,LY338979

LY-338979 是培美曲塞酮的杂质。
T66032 Pemetrexed disodium heptahydrate

Pemetrexed disodium is a guanine-derived antineoplastic agent that functions as a nucleic acid synthesis inhibitor through its binding to, and inhibition of, thymidylate synthase.
T74111 N-Methyl pemetrexed

N-Methyl pemetrexedPemetrexed 的一种杂质,为抗叶酸细胞毒剂,应用于癌症研究。

化合物

Pemetrexed
Cat.No: T0189
Synonym: Pemetrexed acid,培美曲塞,LY231514,培美曲唑,LY-231514 Disodium Hydrate
Target: DHFR, DNA/RNA Synthesis, Antifolate, Autophagy
Pemetrexed disodium hemipenta hydrate
Cat.No: T6226
Synonym: 培美曲塞二钠一水合物,Pemetrexed Disodium Hydrate,LY-231514 Disodium Hydrate,Pemetrexed sodium hydrate,培美曲塞二钠水合物
Target: Apoptosis, DHFR, DNA/RNA Synthesis, Antifolate, Autophagy
Pemetrexed disodium
Cat.No: T0189L
Synonym: 培美曲塞二钠盐,LY-231514,LY231514 disodium,培美曲塞二钠,Pemetrexed
Target: Apoptosis, DHFR, DNA/RNA Synthesis, Antifolate, Autophagy
Pemetrexed tromethamine
Cat.No: T25929
Synonym: Pemetrexed ditromethamine dihydrate
Target:
Pemetrexed Diethyl Ester
Cat.No: T70583
Synonym:
Target:
LY-338979
Cat.No: T20355
Synonym: Pemetrexed 6-oxo diacid impurity,LY338979
Target:
Pemetrexed disodium heptahydrate
Cat.No: T66032
Synonym:
Target:
N-Methyl pemetrexed
Cat.No: T74111
Synonym:
Target:
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